3LJU.X | ADAP1

General Structure Information 3lju ADAP1 crystal structure of full length centaurin alpha-1 bound with the head group of pip3 1.7Å AUTH Y.TONG,W.TEMPEL,H.WANG,K.YAMADA,L.SHEN,G.A.SENISTERRA,AUTH 2 F.MACKENZIE,A.H.CHISHTI,H.W.PARKTITL PHOSPHORYLATION-INDEPENDENT DUAL-SITE BINDING OF THE FHATITL 2 DOMAIN OF KIF13 MEDIATES PHOSPHOINOSITIDE TRANSPORT VIATITL 3 CENTAURIN ALPHA1.REF PROC.NATL.ACAD.SCI.USA V. 107 20346 2010REFN ISSN 0027-8424PMID 21057110DOI 10.1073/PNAS.1009008107 Variant Set Distributions Ripley’s K […]

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2OX0.A | KDM4A

General Structure Information 2ox0 KDM4A crystal structure of jmjd2a complexed with histone h3 peptide dimethylated at lys9 1.95Å AUTH S.S.NG,K.L.KAVANAGH,M.A.MCDONOUGH,D.BUTLER,E.S.PILKA,AUTH 2 B.M.LIENARD,J.E.BRAY,P.SAVITSKY,O.GILEADI,F.VON DELFT,AUTH 3 N.R.ROSE,J.OFFER,J.C.SCHEINOST,T.BOROWSKI,M.SUNDSTROM,AUTH 4 C.J.SCHOFIELD,U.OPPERMANNTITL CRYSTAL STRUCTURES OF HISTONE DEMETHYLASE JMJD2A REVEALTITL 2 BASIS FOR SUBSTRATE SPECIFICITY.REF NATURE V. 448 87 2007REFN ISSN 0028-0836PMID 17589501DOI 10.1038/NATURE05971 Variant Set Distributions Mapped Variants

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2I4I.A | DDX3X

General Structure Information 2i4i DDX3X crystal structure of human dead-box rna helicase ddx3x 2.2Å AUTH M.HOGBOM,R.COLLINS,S.VAN DEN BERG,R.-M.JENVERT,T.KARLBERG,AUTH 2 T.KOTENYOVA,A.FLORES,G.B.KARLSSON HEDESTAM,AUTH 3 L.H.HOLMBERG SCHIAVONETITL CRYSTAL STRUCTURE OF CONSERVED DOMAINS 1 AND 2 OF THE HUMANTITL 2 DEAD-BOX HELICASE DDX3X IN COMPLEX WITH THE MONONUCLEOTIDETITL 3 AMPREF J.MOL.BIOL. V. 372 150 2007REFN ISSN 0022-2836PMID 17631897DOI 10.1016/J.JMB.2007.06.050 […]

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2P0A.A | SYN3

General Structure Information 2p0a SYN3 the crystal structure of human synapsin iii (syn3) in complex with amppnp 1.9Å AUTH A.P.TURNBULL,C.PHILLIPS,A.C.W.PIKE,J.M.ELKINS,C.GILEADI,AUTH 2 E.SALAH,F.H.NIESEN,N.BURGESS,O.GILEADI,F.GORREC,C.UMEANO,AUTH 3 F.VON DELFT,J.WEIGELT,A.EDWARDS,C.H.ARROWSMITH,M.SUNDSTROM,AUTH 4 D.DOYLETITL THE CRYSTAL STRUCTURE OF HUMAN SYNAPSIN III (SYN3) INTITL 2 COMPLEX WITH AMPPNPREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity […]

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2P0R.B | CAPN9

General Structure Information 2p0r CAPN9 structure of human calpain 9 in complex with leupeptin 2.5Å AUTH T.L.DAVIS,R.PARAMANATHAN,J.R.WALKER,C.BUTLER-COLE,AUTH 2 P.J.FINERTY JR.,J.WEIGELT,M.SUNDSTROM,C.H.ARROWSMITH,AUTH 3 A.M.EDWARDS,A.BOCHKAREV,S.DHE-PAGANONTITL STRUCTURES OF HUMAN MINICALPAINS BOUND TO INHIBITORSREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3MDY.A | BMPR1B

General Structure Information 3mdy BMPR1B crystal structure of the cytoplasmic domain of the bone morphogenetic protein receptor type-1b (bmpr1b) in complex with fkbp12 and ldn- 193189 2.05Å AUTH A.CHAIKUAD,C.SANVITALE,P.MAHAJAN,N.DAGA,C.COOPER,T.KROJER,AUTH 2 I.ALFANO,S.KNAPP,F.VON DELFT,J.WEIGELT,C.H.ARROWSMITH,AUTH 3 A.M.EDWARDS,C.BOUNTRA,A.BULLOCK,AUTH 4 STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL CRYSTAL STRUCTURE OF THE CYTOPLASMIC DOMAIN OF THE BONETITL 2 MORPHOGENETIC PROTEIN RECEPTOR TYPE-1B (BMPR1B) IN […]

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3BQR.A | DAPK3

General Structure Information 3bqr DAPK3 crystal structure of human death associated protein kinase 3 (dapk3) in complex with an imidazo-pyridazine ligand 1.75Å AUTH P.FILIPPAKOPOULOS,P.RELLOS,O.FEDOROV,F.NIESEN,A.C.W.PIKE,AUTH 2 E.S.PILKA,F.VON DELFT,C.H.ARROWSMITH,A.M.EDWARDS,J.WEIGELT,AUTH 3 S.KNAPPTITL CRYSTAL STRUCTURE OF HUMAN DEATH ASSOCIATED PROTEIN KINASE 3TITL 2 (DAPK3) IN COMPLEX WITH AN IMIDAZO-PYRIDAZINE LIGAND.REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis […]

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4AVX.A | HGS

General Structure Information 4avx HGS hepatocyte growth factor-regulated tyrosine kinase substrate (hgs-hrs) bound to an ip2 compound at 1.68 a resolution 1.68Å AUTH E.WILLIAMS,P.CANNING,L.SHRESTHA,T.KROJER,M.VOLLMAR,A.SLOWEY,AUTH 2 S.CONWAY,F.VON DELFT,C.H.ARROWSMITH,A.M.EDWARDS,J.WEIGELT,AUTH 3 C.BOUNTRA,A.BULLOCKTITL CRYSTAL STRUCTURE OF THE TANDEM VHS AND FYVE DOMAINS OFTITL 2 HEPATOCYTE GROWTH FACTOR-REGULATED TYROSINE KINASETITL 3 SUBSTRATE (HGS-HRS) BOUND TO AN IP2 COMPOUND AT 1.68 […]

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2F7S.A | RAB27B

General Structure Information 2f7s RAB27B the crystal structure of human rab27b bound to gdp 2.7Å AUTH J.WANG,S.ISMAIL,Y.SHEN,W.TEMPEL,C.H.ARROWSMITH,AUTH 2 A.M.EDWARDS,M.SUNDSTROM,A.BOCHKAREV,H.W.PARKTITL THE CRYSTAL STRUCTURE OF HUMAN RAB27BREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2IHB.B | RGS10

General Structure Information 2ihb RGS10 crystal structure of the heterodimeric complex of human rgs10 and activated gi alpha 3 2.71Å AUTH M.SOUNDARARAJAN,F.S.WILLARD,A.J.KIMPLE,A.P.TURNBULL,AUTH 2 L.J.BALL,G.A.SCHOCH,C.GILEADI,O.Y.FEDOROV,E.F.DOWLER,AUTH 3 V.A.HIGMAN,S.Q.HUTSELL,M.SUNDSTROM,D.A.DOYLE,D.P.SIDEROVSKITITL STRUCTURAL DIVERSITY IN THE RGS DOMAIN AND ITS INTERACTIONTITL 2 WITH HETEROTRIMERIC G PROTEIN ALPHA-SUBUNITS.REF PROC.NATL.ACAD.SCI.USA V. 105 6457 2008REFN ISSN 0027-8424PMID 18434541DOI 10.1073/PNAS.0801508105 Variant Set Distributions Mapped Variants

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