4DHF.A | AURKA

General Structure Information 4dhf AURKA structure of aurora a mutant bound to biogenidec cpd 15 2.8Å AUTH J.Y.LE BRAZIDEC,A.PASIS,B.TAM,C.BOYKIN,D.WANG,D.J.MARCOTTE,AUTH 2 G.CLAASSEN,J.H.CHONG,J.CHAO,J.FAN,K.NGUYEN,L.SILVIAN,L.LING,AUTH 3 L.ZHANG,M.CHOI,M.TENG,N.PATHAN,S.ZHAO,T.LI,A.TAVERASTITL STRUCTURE-BASED DESIGN OFTITL 2 2,6,7-TRISUBSTITUTED-7H-PYRROLO[2,3-D]PYRIMIDINES AS AURORATITL 3 KINASES INHIBITORS.REF BIOORG.MED.CHEM.LETT. V. 22 4033 2012REFN ISSN 0960-894XPMID 22607669DOI 10.1016/J.BMCL.2012.04.085 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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3OL2.B | PLXNB1

General Structure Information 3ol2 PLXNB1 receptor-ligand structure of human semaphorin 4d with plexin b1. 2.99Å AUTH B.J.JANSSEN,R.A.ROBINSON,F.PEREZ-BRANGULI,C.H.BELL,AUTH 2 K.J.MITCHELL,C.SIEBOLD,E.Y.JONESTITL STRUCTURAL BASIS OF SEMAPHORIN-PLEXIN SIGNALLING.REF NATURE V. 467 1118 2010REFN ISSN 0028-0836PMID 20877282DOI 10.1038/NATURE09468 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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4GMJ.C | CNOT1

General Structure Information 4gmj CNOT1 structure of human not1 mif4g domain co-crystallized with caf1 2.7Å AUTH A.P.PETIT,L.WOHLBOLD,P.BAWANKAR,E.HUNTZINGER,S.SCHMIDT,AUTH 2 E.IZAURRALDE,O.WEICHENRIEDERTITL THE STRUCTURAL BASIS FOR THE INTERACTION BETWEEN THE CAF1TITL 2 NUCLEASE AND THE NOT1 SCAFFOLD OF THE HUMAN CCR4-NOTTITL 3 DEADENYLASE COMPLEXREF NUCLEIC ACIDS RES. V. 40 11058 2012REFN ISSN 0305-1048PMID 22977175DOI 10.1093/NAR/GKS883 Variant Set Distributions […]

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2P0R.B | CAPN9

General Structure Information 2p0r CAPN9 structure of human calpain 9 in complex with leupeptin 2.5Å AUTH T.L.DAVIS,R.PARAMANATHAN,J.R.WALKER,C.BUTLER-COLE,AUTH 2 P.J.FINERTY JR.,J.WEIGELT,M.SUNDSTROM,C.H.ARROWSMITH,AUTH 3 A.M.EDWARDS,A.BOCHKAREV,S.DHE-PAGANONTITL STRUCTURES OF HUMAN MINICALPAINS BOUND TO INHIBITORSREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3UKM.D | KCNK1

General Structure Information 3ukm KCNK1 crystal structure of the human two pore domain potassium ion channel k2p1 (twik-1) 3.4Å AUTH A.N.MILLER,S.B.LONGTITL CRYSTAL STRUCTURE OF THE HUMAN TWO-PORE DOMAIN POTASSIUMTITL 2 CHANNEL K2P1.REF SCIENCE V. 335 432 2012REFN ISSN 0036-8075PMID 22282804DOI 10.1126/SCIENCE.1213274 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped […]

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1G55.A | TRDMT1

General Structure Information 1g55 TRDMT1 structure of human dnmt2, an enigmatic dna methyltransferase homologue 1.8Å AUTH A.DONG,J.A.YODER,X.ZHANG,L.ZHOU,T.H.BESTOR,X.CHENGTITL STRUCTURE OF HUMAN DNMT2, AN ENIGMATIC DNA METHYLTRANSFERASETITL 2 HOMOLOG THAT DISPLAYS DENATURANT-RESISTANT BINDING TO DNA.REF NUCLEIC ACIDS RES. V. 29 439 2001REFN ISSN 0305-1048PMID 11139614DOI 10.1093/NAR/29.2.439 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped […]

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4E3C.E | IKBKB

General Structure Information 4e3c IKBKB x-ray crystal structure of human ikk2 in an active conformation 3.98Å AUTH S.POLLEY,D.B.HUANG,A.V.HAUENSTEIN,A.J.FUSCO,X.ZHONG,D.VU,AUTH 2 A.HOFFMANN,I.V.VERMA,G.GHOSH,T.HUAFORDTITL X-RAY CRYSTAL STRUCTURE OF HUMAN IKK2 IN AN ACTIVETITL 2 CONFORMATIONREF PLOS.BIOL. 2013REFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2CZH.B | IMPA2

General Structure Information 2czh IMPA2 crystal structure of human myo-inositol monophosphatase 2 (impa2) with phosphate ion (orthorhombic form) 2.7Å AUTH R.ARAI,K.ITO,T.OHNISHI,H.OHBA,R.AKASAKA,Y.BESSHO,AUTH 2 K.HANAWA-SUETSUGU,T.YOSHIKAWA,M.SHIROUZU,S.YOKOYAMATITL CRYSTAL STRUCTURE OF HUMAN MYO-INOSITOLTITL 2 MONOPHOSPHATASE 2, THE PRODUCT OF THE PUTATIVETITL 3 SUSCEPTIBILITY GENE FOR BIPOLAR DISORDER,TITL 4 SCHIZOPHRENIA, AND FEBRILE SEIZURESREF PROTEINS V. 67 732 2007REFN ISSN 0887-3585PMID 17340635DOI […]

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1GUM.D | GSTA4

General Structure Information 1gum GSTA4 human glutathione transferase a4-4 without ligands 3.0Å AUTH C.M.BRUNS,I.HUBATSCH,M.RIDDERSTROM,B.MANNERVIK,AUTH 2 J.A.TAINERTITL HUMAN GLUTATHIONE TRANSFERASE A4-4 CRYSTALTITL 2 STRUCTURES AND MUTAGENESIS REVEAL THE BASIS OFTITL 3 HIGH CATALYTIC EFFICIENCY WITH TOXIC LIPIDTITL 4 PEROXIDATION PRODUCTSREF J.MOL.BIOL. V. 288 427 1999REFN ISSN 0022-2836PMID 10329152DOI 10.1006/JMBI.1999.2697 Variant Set Distributions Ripley’s K Analysis Plots […]

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2Q5E.C | CTDSP2

General Structure Information 2q5e CTDSP2 crystal structure of human carboxy-terminal domain rna polymerase ii polypeptide a small phosphatase 2 2.51Å AUTH S.C.ALMO,J.B.BONANNO,J.M.SAUDER,S.EMTAGE,AUTH 2 T.P.DILORENZO,V.MALASHKEVICH,S.R.WASSERMAN,AUTH 3 S.SWAMINATHAN,S.ESWARAMOORTHY,R.AGARWAL,D.KUMARAN,AUTH 4 M.MADEGOWDA,S.RAGUMANI,Y.PATSKOVSKY,J.ALVARADO,AUTH 5 U.A.RAMAGOPAL,J.FABER-BARATA,M.R.CHANCE,A.SALI,AUTH 6 A.FISER,Z.Y.ZHANG,D.S.LAWRENCE,S.K.BURLEYTITL STRUCTURAL GENOMICS OF PROTEIN PHOSPHATASES.REF J.STRUCT.FUNCT.GENOM. V. 8 121 2007REFN ISSN 1345-711XPMID 18058037DOI 10.1007/S10969-007-9036-1 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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