1JUJ.C | TYMS

General Structure Information 1juj TYMS human thymidylate synthase bound to dump and ly231514, a pyrrolo(2,3-d)pyrimidine-based antifolate 3.0Å AUTH P.H.SAYRE,J.S.FINER-MOORE,T.A.FRITZ,D.BIERMANN,AUTH 2 S.B.GATES,W.C.MACKELLAR,V.F.PATEL,R.M.STROUDTITL MULTI-TARGETED ANTIFOLATES AIMED AT AVOIDING DRUGTITL 2 RESISTANCE FORM COVALENT CLOSED INHIBITORYTITL 3 COMPLEXES WITH HUMAN AND ESCHERICHIA COLITITL 4 THYMIDYLATE SYNTHASES.REF J.MOL.BIOL. V. 313 813 2001REFN ISSN 0022-2836PMID 11697906DOI 10.1006/JMBI.2001.5074 Variant Set Distributions […]

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1LQ8.G | SERPINA5

General Structure Information 1lq8 SERPINA5 crystal structure of cleaved protein c inhibitor 2.4Å AUTH J.A.HUNTINGTON,M.KJELLBERG,J.STENFLOTITL CRYSTAL STRUCTURE OF PROTEIN C INHIBITOR PROVIDES INSIGHTSTITL 2 INTO HORMONE BINDING AND HEPARIN ACTIVATIONREF STRUCTURE V. 11 205 2003REFN ISSN 0969-2126PMID 12575940DOI 10.1016/S0969-2126(02)00944-9 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2UZP.B | PRKCG

General Structure Information 2uzp PRKCG crystal structure of the c2 domain of human protein kinase c gamma. 2.0Å AUTH A.C.W.PIKE,A.AMOS,C.JOHANSSON,F.SOBOTT,P.SAVITSKY,AUTH 2 G.BERRIDGE,O.FEDOROV,C.UMEANO,F.GORREC,G.BUNKOCZI,AUTH 3 J.DEBRECZENI,F.VON DELFT,C.H.ARROWSMITH,A.EDWARDS,J.WEIGELT,AUTH 4 M.SUNDSTROM,S.KNAPPTITL CRYSTAL STRUCTURE OF C2 DOMAIN OF PROTEIN KINASE C GAMMAREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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4F0X.H | MLYCD

General Structure Information 4f0x MLYCD crystal structure of human malonyl-coa decarboxylase (peroxisomal isoform) 3.29Å AUTH D.APARICIO,R.PEREZ-LUQUE,X.CARPENA,M.DIAZ,J.C.FERRER,AUTH 2 P.C.LOEWEN,I.FITATITL STRUCTURAL ASYMMETRY AND DISULFIDE BRIDGES AMONG SUBUNITSTITL 2 MODULATE THE ACTIVITY OF HUMAN MALONYL-COA DECARBOXYLASE.REF J.BIOL.CHEM. V. 288 11907 2013REFN ISSN 0021-9258PMID 23482565DOI 10.1074/JBC.M112.443846 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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3RUK.C | CYP17A1

General Structure Information 3ruk CYP17A1 human cytochrome p450 cyp17a1 in complex with abiraterone 2.6Å AUTH N.M.DEVORE,E.E.SCOTTTITL STRUCTURES OF CYTOCHROME P450 17A1 WITH PROSTATE CANCERTITL 2 DRUGS ABIRATERONE AND TOK-001.REF NATURE V. 482 116 2012REFN ISSN 0028-0836PMID 22266943DOI 10.1038/NATURE10743 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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2OAY.A | SERPING1

General Structure Information 2oay SERPING1 crystal structure of latent human c1-inhibitor 2.35Å AUTH L.BEINROHR,V.HARMAT,J.DOBO,Z.LORINCZ,P.GAL,P.ZAVODSZKYTITL C1 INHIBITOR SERPIN DOMAIN STRUCTURE REVEALS THE LIKELYTITL 2 MECHANISM OF HEPARIN POTENTIATION AND CONFORMATIONAL DISEASEREF J.BIOL.CHEM. V. 282 21100 2007REFN ISSN 0021-9258PMID 17488724DOI 10.1074/JBC.M700841200 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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1AFO.B | GYPA

General Structure Information 1afo GYPA dimeric transmembrane domain of human glycophorin a, nmr, 20 structures -1.0Å AUTH K.R.MACKENZIE,J.H.PRESTEGARD,D.M.ENGELMANTITL A TRANSMEMBRANE HELIX DIMER: STRUCTURE ANDTITL 2 IMPLICATIONS.REF SCIENCE V. 276 131 1997REFN ISSN 0036-8075PMID 9082985DOI 10.1126/SCIENCE.276.5309.131 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2WEF.A | BPNT1

General Structure Information 2wef BPNT1 human 3(2), 5-bisphosphate nucleotidase 1 (bpnt1) in complex with amp, po4 and magnesium 1.8Å AUTH M.MOCHE,P.SCHUTZ,C.H.ARROWSMITH,H.BERGLUND,AUTH 2 C.BOUNTRA,R.COLLINS,L.G.DAHLGREN,A.M.EDWARDS,AUTH 3 S.FLODIN,A.FLORES,S.GRASLUND,M.HAMMARSTROM,AUTH 4 A.JOHANSSON,I.JOHANSSON,T.KARLBERG,T.KOTENYOVA,AUTH 5 M.E.NILSSON,T.NYMAN,C.PERSSON,J.SAGEMARK,AUTH 6 H.SCHUELER,M.I.SIPONEN,A.G.THORSELL,L.TRESAUGUES,AUTH 7 S.VAN DEN BERG,J.WEIGELT,M.WELIN,M.WISNIEWSKA,AUTH 8 P.NORDLUNDTITL HUMAN 3(2), 5-BISPHOSPHATE NUCLEOTIDASE 1 (TITL 2 BPNT1) IN COMPLEX WITH AMP, PO4 AND MAGNESIUMREF TO BE PUBLISHEDREFN […]

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1HIG.D | IFNG

General Structure Information 1hig IFNG three-dimensional structure of recombinant human interferon- gamma. 3.5Å AUTH S.E.EALICK,W.J.COOK,S.VIJAY-KUMAR,M.CARSON,AUTH 2 T.L.NAGABHUSHAN,P.P.TROTTA,C.E.BUGGTITL THREE-DIMENSIONAL STRUCTURE OF RECOMBINANT HUMANTITL 2 INTERFERON-GAMMA.REF SCIENCE V. 252 698 1991REFN ISSN 0036-8075PMID 1902591 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2JWA.A | ERBB2

General Structure Information 2jwa ERBB2 erbb2 transmembrane segment dimer spatial structure -1.0Å AUTH E.V.BOCHAROV,K.S.MINEEV,P.E.VOLYNSKY,Y.S.ERMOLYUK,AUTH 2 E.N.TKACH,A.G.SOBOL,V.V.CHUPIN,M.P.KIRPICHNIKOV,AUTH 3 R.G.EFREMOV,A.S.ARSENIEVTITL SPATIAL STRUCTURE OF THE DIMERIC TRANSMEMBRANETITL 2 DOMAIN OF THE GROWTH FACTOR RECEPTOR ERBB2TITL 3 PRESUMABLY CORRESPONDING TO THE RECEPTOR ACTIVETITL 4 STATEREF J.BIOL.CHEM. V. 283 6950 2008REFN ISSN 0021-9258PMID 18178548DOI 10.1074/JBC.M709202200 Variant Set Distributions Ripley’s K […]

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