3RCD.A | ERBB2

General Structure Information 3rcd ERBB2 her2 kinase domain complexed with tak-285 3.21Å AUTH T.ISHIKAWA,M.SETO,H.BANNO,Y.KAWAKITA,M.OORUI,T.TANIGUCHI,AUTH 2 Y.OHTA,T.TAMURA,A.NAKAYAMA,H.MIKI,H.KAMIGUCHI,T.TANAKA,AUTH 3 N.HABUKA,S.SOGABE,J.YANO,K.AERTGEERTS,K.KAMIYAMATITL DESIGN AND SYNTHESIS OF NOVEL HUMAN EPIDERMAL GROWTH FACTORTITL 2 RECEPTOR 2 (HER2)/EPIDERMAL GROWTH FACTOR RECEPTOR (EGFR)TITL 3 DUAL INHIBITORS BEARING A PYRROLO[3,2-D]PYRIMIDINE SCAFFOLD.REF J.MED.CHEM. V. 54 8030 2011REFN ISSN 0022-2623PMID 22003817DOI 10.1021/JM2008634 Variant Set Distributions Ripley’s […]

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2Y3I.A | PGK1

General Structure Information 2y3i PGK1 the structure of the fully closed conformation of human pgk in complex with l-adp, 3pg and the tsa aluminium tetrafluoride 2.9Å AUTH P.LALLEMAND,L.CHALOIN,B.ROY,T.BARMAN,M.W.BOWLER,C.LIONNETITL INTERACTION OF HUMAN 3-PHOSPHOGLYCERATE KINASE WITH ITS TWOTITL 2 SUBSTRATES: IS SUBSTRATE ANTAGONISM A KINETIC ADVANTAGE?REF J.MOL.BIOL. V. 409 742 2011REFN ISSN 0022-2836PMID 21549713DOI 10.1016/J.JMB.2011.04.048 Variant Set […]

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3KLS.B | C5

General Structure Information 3kls C5 structure of complement c5 in complex with ssl7 3.6Å AUTH N.S.LAURSEN,N.GORDON,S.HERMANS,N.LORENZ,N.JACKSON,B.WINES,AUTH 2 E.SPILLNER,J.B.CHRISTENSEN,M.JENSEN,F.FREDSLUND,M.BJERRE,AUTH 3 L.SOTTRUP-JENSEN,J.D.FRASER,G.R.ANDERSENTITL STRUCTURAL BASIS FOR INHIBITION OF COMPLEMENT C5 BY THE SSL7TITL 2 PROTEIN FROM STAPHYLOCOCCUS AUREUSREF PROC.NATL.ACAD.SCI.USA V. 107 3681 2010REFN ISSN 0027-8424PMID 20133685DOI 10.1073/PNAS.0910565107 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped […]

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3Q91.D | NUDT14

General Structure Information 3q91 NUDT14 crystal structure of human uridine diphosphate glucose pyrophosphatase (nudt14) 2.7Å AUTH L.TRESAUGUES,M.I.SIPONEN,C.H.ARROWSMITH,H.BERGLUND,AUTH 2 C.BOUNTRA,R.COLLINS,A.M.EDWARDS,T.EKBLAD,S.FLODIN,A.FLORES,AUTH 3 S.GRASLUND,M.HAMMARSTROM,I.JOHANSSON,T.KARLBERG,S.KOL,AUTH 4 T.KOTENYOVA,E.KOUZNETSOVA,M.MOCHE,T.NYMAN,C.PERSSON,AUTH 5 H.SCHULER,P.SCHUTZ,A.G.THORSELL,S.VAN DER BERG,E.WAHLBERG,AUTH 6 J.WEIGELT,M.WELIN,P.NORDLUNDTITL CRYSTAL STRUCTURE OF HUMAN URIDINE DIPHOSPHATE GLUCOSETITL 2 PYROPHOSPHATASE (NUDT14)REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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1JMO.A | SERPIND1

General Structure Information 1jmo SERPIND1 crystal structure of the heparin cofactor ii-s195a thrombin complex 2.2Å AUTH T.P.BAGLIN,R.W.CARRELL,F.C.CHURCH,C.T.ESMON,J.A.HUNTINGTONTITL CRYSTAL STRUCTURES OF NATIVE AND THROMBIN-COMPLEXED HEPARINTITL 2 COFACTOR II REVEAL A MULTISTEP ALLOSTERIC MECHANISM.REF PROC.NATL.ACAD.SCI.USA V. 99 11079 2002REFN ISSN 0027-8424PMID 12169660DOI 10.1073/PNAS.162232399 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped […]

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1B9G.A | IGF1

General Structure Information 1b9g IGF1 insulin-like-growth-factor-1 -1.0Å AUTH E.DE WOLF,R.GILL,S.GEDDES,J.PITTS,A.WOLLMER,AUTH 2 J.GROTZINGERTITL SOLUTION STRUCTURE OF A MINI IGF-1.REF PROTEIN SCI. V. 5 2193 1996REFN ISSN 0961-8368PMID 8931138 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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2NZ2.A | ASS1

General Structure Information 2nz2 ASS1 crystal structure of human argininosuccinate synthase in complex with aspartate and citrulline 2.4Å AUTH T.KARLBERG,R.COLLINS,S.VAN DEN BERG,A.FLORES,M.HAMMARSTROM,AUTH 2 M.HOGBOM,L.HOLMBERG SCHIAVONE,J.UPPENBERGTITL STRUCTURE OF HUMAN ARGININOSUCCINATE SYNTHETASE.REF ACTA CRYSTALLOGR.,SECT.D V. 64 279 2008REFN ISSN 0907-4449PMID 18323623DOI 10.1107/S0907444907067455 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2F83.A | F11

General Structure Information 2f83 F11 crystal structure at 2.9 angstroms resolution of human plasma coagulation factor xi zymogen 2.87Å AUTH E.PAPAGRIGORIOU,P.A.MCEWAN,P.N.WALSH,J.EMSLEYTITL CRYSTAL STRUCTURE OF THE FACTOR XI ZYMOGEN REVEALS A PATHWAYTITL 2 FOR TRANSACTIVATION.REF NAT.STRUCT.MOL.BIOL. V. 13 557 2006REFN ISSN 1545-9993PMID 16699514DOI 10.1038/NSMB1095 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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4L1M.A | HERC2

General Structure Information 4l1m HERC2 structure of the first rcc1-like domain of herc2 2.6Å AUTH W.TEMPEL,M.B.KHAN,A.DONG,J.HU,Y.LI,C.BOUNTRA,C.H.ARROWSMITH,AUTH 2 A.M.EDWARDS,Y.TONGTITL STRUCTURE OF THE FIRST RCC1-LIKE DOMAIN OF HERC2REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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1RTF.B | PLAT

General Structure Information 1rtf PLAT complex of benzamidine with the catalytic domain of human two chain tissue plasminogen activator [(tc)-t-pa] 2.3Å AUTH D.LAMBA,M.BAUER,R.HUBER,S.FISCHER,R.RUDOLPH,AUTH 2 U.KOHNERT,W.BODETITL THE 2.3 A CRYSTAL STRUCTURE OF THE CATALYTICTITL 2 DOMAIN OF RECOMBINANT TWO-CHAIN HUMAN TISSUE-TYPETITL 3 PLASMINOGEN ACTIVATORREF J.MOL.BIOL. V. 258 117 1996REFN ISSN 0022-2836PMID 8613982DOI 10.1006/JMBI.1996.0238 Variant Set Distributions […]

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