3II5.A | BRAF

General Structure Information 3ii5 BRAF the complex of wild-type b-raf with pyrazolo pyrimidine inhibitor 2.79Å AUTH D.M.BERGER,N.TORRES,M.DUTIA,D.POWELL,G.CISZEWSKI,AUTH 2 A.GOPALSAMY,J.I.LEVIN,K.H.KIM,W.XU,J.WILHELM,Y.HU,AUTH 3 K.COLLINS,L.FELDBERG,S.KIM,E.FROMMER,AUTH 4 D.WOJCIECHOWICZ,R.MALLONTITL NON-HINGE-BINDING PYRAZOLO[1,5-A]PYRIMIDINES ASTITL 2 POTENT B-RAF KINASE INHIBITORS.REF BIOORG.MED.CHEM.LETT. V. 19 6519 2009REFN ISSN 0960-894XPMID 19864136DOI 10.1016/J.BMCL.2009.10.049 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2FVL.B | AKR1C4

General Structure Information 2fvl AKR1C4 crystal structure of human 3-alpha hydroxysteroid/dihydrodiol dehydrogenase (akr1c4) complexed with nadp+ 2.4Å AUTH E.UGOCHUKWU,C.SMEE,K.GUO,P.LUKACIK,K.KAVANAGH,AUTH 2 J.E.DEBRECZENI,F.VON DELFT,J.WEIGELT,M.SUNDSTROM,AUTH 3 C.ARROWSMITH,A.EDWARDS,U.OPPERMANNTITL CRYSTAL STRUCTURE OF HUMAN 3-ALPHATITL 2 HYDROXYSTEROID/DIHYDRODIOL DEHYDROGENASE (AKR1C4) COMPLEXEDTITL 3 WITH NADP+REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1YK0.B | NPR3

General Structure Information 1yk0 NPR3 structure of natriuretic peptide receptor-c complexed with atrial natriuretic peptide 2.4Å AUTH X.L.HE,A.DUKKIPATI,K.C.GARCIATITL STRUCTURAL DETERMINANTS OF NATRIURETIC PEPTIDE RECEPTORTITL 2 SPECIFICITY AND DEGENERACY.REF J.MOL.BIOL. V. 361 698 2006REFN ISSN 0022-2836PMID 16870210DOI 10.1016/J.JMB.2006.06.060 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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1OP8.F | GZMA

General Structure Information 1op8 GZMA crystal structure of human granzyme a 2.5Å AUTH C.HINK-SCHAUER,E.ESTEBANEZ-PERPINA,F.KURSCHUS,AUTH 2 W.BODE,D.JENNETITL CRYSTAL STRUCTURE OF THE APOPTOSIS-INDUCING HUMANTITL 2 GRANZYME A DIMERREF NAT.STRUCT.BIOL. V. 10 535 2003REFN ISSN 1072-8368PMID 12819770DOI 10.1038/NSB945 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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4KKI.A | TCN1

General Structure Information 4kki TCN1 crystal structure of haptocorrin in complex with cncbl 2.35Å AUTH E.FURGER,D.C.FREI,R.SCHIBLI,E.FISCHER,A.E.PROTATITL STRUCTURAL BASIS FOR UNIVERSAL CORRINOID RECOGNITION BY THETITL 2 COBALAMIN TRANSPORT PROTEIN HAPTOCORRIN.REF J.BIOL.CHEM. V. 288 25466 2013REFN ISSN 0021-9258PMID 23846701DOI 10.1074/JBC.M113.483271 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1PV8.B | ALAD

General Structure Information 1pv8 ALAD crystal structure of a low activity f12l mutant of human porphobilinogen synthase 2.2Å AUTH S.BREINIG,J.KERVINEN,L.STITH,A.S.WASSON,R.FAIRMAN,AUTH 2 A.WLODAWER,A.ZDANOV,E.K.JAFFETITL CONTROL OF TETRAPYRROLE BIOSYNTHESIS BY ALTERNATE QUATERNARYTITL 2 FORMS OF PORPHOBILINOGEN SYNTHASE.REF NAT.STRUCT.BIOL. V. 10 757 2003REFN ISSN 1072-8368PMID 12897770DOI 10.1038/NSB963 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity […]

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3W4I.D | DAO

General Structure Information 3w4i DAO crystal structure of human daao in complex with coumpound 8 2.5Å AUTH T.HONDO,M.WARIZAYA,T.NIIMI,I.NAMATAME,T.YAMAGUCHI,AUTH 2 K.NAKANISHI,T.HAMAJIMA,K.HARADA,H.SAKASHITA,Y.MATSUMOTO,AUTH 3 M.ORITA,M.TAKEUCHITITL 4-HYDROXYPYRIDAZIN-3(2H)-ONE DERIVATIVES AS NOVEL D-AMINOTITL 2 ACID OXIDASE INHIBITORS.REF J.MED.CHEM. V. 56 3582 2013REFN ISSN 0022-2623PMID 23566269DOI 10.1021/JM400095B Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3V4V.A | ITGA4

General Structure Information 3v4v ITGA4 crystal structure of a4b7 headpiece complexed with fab act-1 and ro0505376 3.1Å AUTH Y.YU,J.ZHU,L.Z.MI,T.WALZ,H.SUN,J.CHEN,T.A.SPRINGERTITL STRUCTURAL SPECIALIZATIONS OF A4B7, AN INTEGRIN THATTITL 2 MEDIATES ROLLING ADHESIONREF J.CELL BIOL. V. 196 131 2012REFN ISSN 0021-9525PMID 22232704DOI 10.1083/JCB.201110023 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3DZU.A | RXRA

General Structure Information 3dzu RXRA intact ppar gamma – rxr alpha nuclear receptor complex on dna bound with bvt.13, 9-cis retinoic acid and ncoa2 peptide 3.2Å AUTH V.CHANDRA,P.HUANG,Y.HAMURO,S.RAGHURAM,Y.WANG,T.P.BURRIS,AUTH 2 F.RASTINEJADTITL STRUCTURE OF THE INTACT PPAR-GAMMA-RXR- NUCLEAR RECEPTORTITL 2 COMPLEX ON DNA.REF NATURE V. 456 350 2008REFN ISSN 0028-0836PMID 19043829DOI 10.1038/NATURE07413 Variant Set Distributions Ripley’s K […]

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2NSM.A | CPN1

General Structure Information 2nsm CPN1 crystal structure of the human carboxypeptidase n (kininase i) catalytic domain 2.1Å AUTH C.KEIL,K.MASKOS,M.THAN,J.T.HOOPES,R.HUBER,F.TAN,P.A.DEDDISH,AUTH 2 E.G.ERDOES,R.A.SKIDGEL,W.BODETITL CRYSTAL STRUCTURE OF THE HUMAN CARBOXYPEPTIDASE N (KININASETITL 2 I) CATALYTIC DOMAINREF J.MOL.BIOL. V. 366 504 2007REFN ISSN 0022-2836PMID 17157876DOI 10.1016/J.JMB.2006.11.025 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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