2QC8.F | GLUL

General Structure Information 2qc8 GLUL crystal structure of human glutamine synthetase in complex with adp and methionine sulfoximine phosphate 2.6Å AUTH W.W.KRAJEWSKI,R.COLLINS,L.HOLMBERG-SCHIAVONE,T.A.JONES,AUTH 2 T.KARLBERG,S.L.MOWBRAYTITL CRYSTAL STRUCTURES OF MAMMALIAN GLUTAMINE SYNTHETASESTITL 2 ILLUSTRATE SUBSTRATE-INDUCED CONFORMATIONAL CHANGES ANDTITL 3 PROVIDE OPPORTUNITIES FOR DRUG AND HERBICIDE DESIGN.REF J.MOL.BIOL. V. 375 217 2008REFN ISSN 0022-2836PMID 18005987DOI 10.1016/J.JMB.2007.10.029 Variant Set […]

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2WK3.B | IDE

General Structure Information 2wk3 IDE crystal structure of human insulin-degrading enzyme in complex with amyloid-beta (1-42) 2.59Å AUTH Q.GUO,M.MANOLOPOULOU,Y.BIAN,A.B.SCHILLING,W.J.TANGTITL MOLECULAR BASIS FOR THE RECOGNITION AND CLEAVAGESTITL 2 OF IGF-II, TGF-ALPHA, AND AMYLIN BY HUMAN INSULINTITL 3 DEGRADING ENZYME.REF J.MOL.BIOL. V. 395 430 2010REFN ISSN 0022-2836PMID 19896952DOI 10.1016/J.JMB.2009.10.072 Variant Set Distributions Ripley’s K Analysis Plots Variant […]

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4H27.A | SDS

General Structure Information 4h27 SDS modulating the function of human serine racemase and human serine dehydratase by protein engineering 1.3Å AUTH C.Y.WANG,S.C.KU,C.C.LEE,A.H.WANGTITL MODULATING THE FUNCTION OF HUMAN SERINE RACEMASE AND HUMANTITL 2 SERINE DEHYDRATASE BY PROTEIN ENGINEERING.REF PROTEIN ENG.DES.SEL. V. 25 741 2012REFN ISSN 1741-0126PMID 23112234DOI 10.1093/PROTEIN/GZS078 Variant Set Distributions Ripley’s K Analysis Plots Variant […]

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1AVF.A | PGC

General Structure Information 1avf PGC activation intermediate 2 of human gastricsin from human stomach 2.36Å AUTH A.R.KHAN,M.M.CHERNEY,N.I.TARASOVA,M.N.JAMESTITL STRUCTURAL CHARACTERIZATION OF ACTIVATIONTITL 2 INTERMEDIATE 2 ON THE PATHWAY TO HUMANTITL 3 GASTRICSIN.REF NAT.STRUCT.BIOL. V. 4 1010 1997REFN ISSN 1072-8368PMID 9406551DOI 10.1038/NSB1297-1010 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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4DVQ.J | CYP11B2

General Structure Information 4dvq CYP11B2 structure of human aldosterone synthase, cyp11b2, in complex with deoxycorticosterone 2.49Å AUTH N.STRUSHKEVICH,A.A.GILEP,L.SHEN,C.H.ARROWSMITH,A.M.EDWARDS,AUTH 2 S.A.USANOV,H.W.PARKTITL STRUCTURAL INSIGHTS INTO ALDOSTERONE SYNTHASE SUBSTRATETITL 2 SPECIFICITY AND TARGETED INHIBITION.REF MOL.ENDOCRINOL. V. 27 315 2013REFN ISSN 0888-8809PMID 23322723DOI 10.1210/ME.2012-1287 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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4FYS.A | ANPEP

General Structure Information 4fys ANPEP human aminopeptidase n (cd13) in complex with angiotensin iv 2.01Å AUTH A.H.WONG,D.ZHOU,J.M.RINITITL THE X-RAY CRYSTAL STRUCTURE OF HUMAN AMINOPEPTIDASE NTITL 2 REVEALS A NOVEL DIMER AND THE BASIS FOR PEPTIDE PROCESSING.REF J.BIOL.CHEM. V. 287 36804 2012REFN ISSN 0021-9258PMID 22932899DOI 10.1074/JBC.M112.398842 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

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3II5.A | BRAF

General Structure Information 3ii5 BRAF the complex of wild-type b-raf with pyrazolo pyrimidine inhibitor 2.79Å AUTH D.M.BERGER,N.TORRES,M.DUTIA,D.POWELL,G.CISZEWSKI,AUTH 2 A.GOPALSAMY,J.I.LEVIN,K.H.KIM,W.XU,J.WILHELM,Y.HU,AUTH 3 K.COLLINS,L.FELDBERG,S.KIM,E.FROMMER,AUTH 4 D.WOJCIECHOWICZ,R.MALLONTITL NON-HINGE-BINDING PYRAZOLO[1,5-A]PYRIMIDINES ASTITL 2 POTENT B-RAF KINASE INHIBITORS.REF BIOORG.MED.CHEM.LETT. V. 19 6519 2009REFN ISSN 0960-894XPMID 19864136DOI 10.1016/J.BMCL.2009.10.049 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2FVL.B | AKR1C4

General Structure Information 2fvl AKR1C4 crystal structure of human 3-alpha hydroxysteroid/dihydrodiol dehydrogenase (akr1c4) complexed with nadp+ 2.4Å AUTH E.UGOCHUKWU,C.SMEE,K.GUO,P.LUKACIK,K.KAVANAGH,AUTH 2 J.E.DEBRECZENI,F.VON DELFT,J.WEIGELT,M.SUNDSTROM,AUTH 3 C.ARROWSMITH,A.EDWARDS,U.OPPERMANNTITL CRYSTAL STRUCTURE OF HUMAN 3-ALPHATITL 2 HYDROXYSTEROID/DIHYDRODIOL DEHYDROGENASE (AKR1C4) COMPLEXEDTITL 3 WITH NADP+REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1EXT.A | TNFRSF1A

General Structure Information 1ext TNFRSF1A extracellular domain of the 55kda tumor necrosis factor receptor. crystallized at ph3.7 in p 21 21 21. 1.85Å AUTH J.H.NAISMITH,T.Q.DEVINE,T.KOHNO,S.R.SPRANGTITL STRUCTURES OF THE EXTRACELLULAR DOMAIN OF THE TYPETITL 2 I TUMOR NECROSIS FACTOR RECEPTOR.REF STRUCTURE V. 4 1251 1996REFN ISSN 0969-2126PMID 8939750DOI 10.1016/S0969-2126(96)00134-7 Variant Set Distributions Pathogenic Proximity Analysis Mapped […]

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1OP8.F | GZMA

General Structure Information 1op8 GZMA crystal structure of human granzyme a 2.5Å AUTH C.HINK-SCHAUER,E.ESTEBANEZ-PERPINA,F.KURSCHUS,AUTH 2 W.BODE,D.JENNETITL CRYSTAL STRUCTURE OF THE APOPTOSIS-INDUCING HUMANTITL 2 GRANZYME A DIMERREF NAT.STRUCT.BIOL. V. 10 535 2003REFN ISSN 1072-8368PMID 12819770DOI 10.1038/NSB945 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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