3D3L.B | ALOX12

General Structure Information 3d3l ALOX12 the 2.6 a crystal structure of the lipoxygenase domain of human arachidonate 12-lipoxygenase, 12s-type (casp target) 2.6Å AUTH L.TRESAUGUES,M.MOCHE,C.H.ARROWSMITH,H.BERGLUND,AUTH 2 R.D.BUSAM,R.COLLINS,L.G.DAHLGREN,A.M.EDWARDS,AUTH 3 S.FLODIN,A.FLORES,S.GRASLUND,M.HAMMARSTROM,AUTH 4 M.D.HERMAN,A.JOHANSSON,I.JOHANSSON,A.KALLAS,AUTH 5 T.KARLBERG,T.KOTENYOVA,L.LEHTIO,M.E.NILSSON,AUTH 6 T.NYMAN,K.OLESEN,C.PERSSON,J.SAGEMARK,H.SCHUELER,AUTH 7 L.SVENSSON,A.G.THORSELL,S.VAN DEN BERG,M.WELIN,AUTH 8 J.WEIGELT,M.WIKSTROM,P.NORDLUNDTITL CRYSTAL STRUCTURE OF THE LIPOXYGENASE DOMAIN OFTITL 2 HUMAN ARACHIDONATE 12-LIPOXYGENASE, 12S-TYPE.REF TO BE PUBLISHEDREFN […]

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3OWH.A | NQO2

General Structure Information 3owh NQO2 x-ray structural study of quinone reductase ii inhibition by compounds with micromolar to nanomolar range ic50 values 2.28Å AUTH S.D.PEGAN,M.STURDY,G.FERRY,P.DELAGRANGE,J.A.BOUTIN,AUTH 2 A.D.MESECARTITL X-RAY STRUCTURAL STUDIES OF QUINONE REDUCTASE 2 NANOMOLARTITL 2 RANGE INHIBITORS.REF PROTEIN SCI. V. 20 1182 2011REFN ISSN 0961-8368PMID 21538647DOI 10.1002/PRO.647 Variant Set Distributions Ripley’s K Analysis Plots […]

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1MLW.A | TPH1

General Structure Information 1mlw TPH1 crystal structure of human tryptophan hydroxylase with bound 7,8-dihydro-l-biopterin cofactor and fe(iii) 1.71Å AUTH L.WANG,H.ERLANDSEN,J.HAAVIK,P.M.KNAPPSKOG,AUTH 2 R.C.STEVENSTITL THREE-DIMENSIONAL STRUCTURE OF HUMAN TRYPTOPHANTITL 2 HYDROXYLASE AND ITS IMPLICATIONS FOR THETITL 3 BIOSYNTHESIS OF THE NEUROTRANSMITTERS SEROTONINTITL 4 AND MELATONINREF BIOCHEMISTRY V. 41 12569 2002REFN ISSN 0006-2960PMID 12379098DOI 10.1021/BI026561F Variant Set Distributions […]

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1H66.D | NQO1

General Structure Information 1h66 NQO1 crystal structure of human nad[p]h-quinone oxidoreductase co with 2,5-diaziridinyl-3-hydroxyl-6-methyl-1,4-benzoquinone 2.0Å AUTH M.FAIG,M.A.BIANCHET,S.WINSKI,R.HARGREAVES,C.J.MOODY,AUTH 2 A.R.HUDNOTT,D.ROSS,L.M.AMZELTITL STRUCTURE-BASED DEVELOPMENT OF ANTICANCER DRUGS: COMPLEXESTITL 2 OF NAD(P)H:QUINONE OXIDOREDUCTASE 1 WITH CHEMOTHERAPEUTICTITL 3 QUINONESREF STRUCTURE V. 9 659 2001REFN ISSN 0969-2126PMID 11587640DOI 10.1016/S0969-2126(01)00636-0 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity […]

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4BTA.B | P4HA1

General Structure Information 4bta P4HA1 crystal structure of the peptide(pro-pro-gly)3 bound complex of n-terminal domain and peptide substrate binding domain of prolyl-4 hydroxylase (residues 1-244) type i from human 2.95Å AUTH J.ANANTHARAJAN,M.K.KOSKI,P.KURSULA,R.HIETA,U.BERGMANN,AUTH 2 J.MYLLYHARJU,R.K.WIERENGATITL THE STRUCTURAL MOTIFS FOR SUBSTRATE BINDING ANDTITL 2 DIMERIZATION OF THE ALPHA SUBUNIT OF COLLAGEN PROLYLTITL 3 4-HYDROXYLASEREF STRUCTURE V. 21 […]

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3BHM.A | CBR1

General Structure Information 3bhm CBR1 crystal structure of human carbonyl reductase 1 in complex with s-hydroxymethylglutathione 1.8Å AUTH R.L.BATEMAN,D.RAUH,B.TAVSHANJIAN,K.M.SHOKATTITL HUMAN CARBONYL REDUCTASE 1 IS ANTITL 2 S-NITROSOGLUTATHIONE REDUCTASEREF J.BIOL.CHEM. V. 283 35756 2008REFN ISSN 0021-9258PMID 18826943DOI 10.1074/JBC.M807125200 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3MPH.B | AOC1

General Structure Information 3mph AOC1 the structure of human diamine oxidase complexed with an inhibitor aminoguanidine 2.05Å AUTH A.P.MCGRATH,T.CARADOC-DAVIES,C.A.COLLYER,J.M.GUSSTITL CORRELATION OF ACTIVE SITE METAL CONTENT IN HUMAN DIAMINETITL 2 OXIDASE WITH TRIHYDROXYPHENYLALANINE QUINONE COFACTORTITL 3 BIOGENESISREF BIOCHEMISTRY V. 49 8316 2010REFN ISSN 0006-2960PMID 20722416DOI 10.1021/BI1010915 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

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2VIG.H | ACADS

General Structure Information 2vig ACADS crystal structure of human short-chain acyl coa dehydrogenase 1.9Å AUTH A.C.W.PIKE,N.PANTIC,E.PARIZOTTO,O.GILEADI,AUTH 2 E.UGOCHUKWU,F.VON DELFT,J.WEIGELT,C.H.ARROWSMITH,AUTH 3 A.EDWARDS,U.OPPERMANNTITL CRYSTAL STRUCTURE OF HUMAN SHORT-CHAIN ACYL COATITL 2 DEHYDROGENASEREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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1V16.A | BCKDHA

General Structure Information 1v16 BCKDHA crosstalk between cofactor binding and the phosphorylation loop conformation in the bckd machine 1.9Å AUTH J.LI,R.M.WYNN,M.MACHIUS,J.L.CHUANG,S.KARTHIKEYAN,AUTH 2 D.R.TOMCHICK,D.T.CHUANGTITL CROSS-TALK BETWEEN THIAMIN DIPHOSPHATE BINDING ANDTITL 2 PHOSPHORYLATION LOOP CONFORMATION IN HUMAN BRANCHED-CHAINTITL 3 {ALPHA}-KETO ACID DECARBOXYLASE/DEHYDROGENASEREF J.BIOL.CHEM. V. 279 32968 2004REFN ISSN 0021-9258PMID 15166214DOI 10.1074/JBC.M403611200 Variant Set Distributions Pathogenic Proximity Analysis […]

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2GDZ.A | HPGD

General Structure Information 2gdz HPGD crystal structure of 15-hydroxyprostaglandin dehydrogenase type1, complexed with nad+ 1.65Å AUTH F.H.NIESEN,L.SCHULTZ,A.JADHAV,C.BHATIA,K.GUO,D.J.MALONEY,AUTH 2 E.S.PILKA,M.WANG,U.OPPERMANN,T.D.HEIGHTMAN,A.SIMEONOVTITL HIGH-AFFINITY INHIBITORS OF HUMAN NAD-DEPENDENTTITL 2 15-HYDROXYPROSTAGLANDIN DEHYDROGENASE: MECHANISMS OFTITL 3 INHIBITION AND STRUCTURE-ACTIVITY RELATIONSHIPS.REF PLOS ONE V. 5 E1371 2010REFN ESSN 1932-6203PMID 21072165DOI 10.1371/JOURNAL.PONE.0013719 Variant Set Distributions Mapped Variants

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