1M9K.B | NOS3

General Structure Information 1m9k NOS3 human endothelial nitric oxide synthase with 7- nitroindazole bound 2.01Å AUTH R.J.ROSENFELD,E.D.GARCIN,K.PANDA,G.ANDERSSON,AUTH 2 A.ABERG,A.V.WALLACE,G.M.MORRIS,A.J.OLSON,AUTH 3 D.J.STUEHR,J.A.TAINER,E.D.GETZOFFTITL CONFORMATIONAL CHANGES IN NITRIC OXIDE SYNTHASESTITL 2 INDUCED BY CHLORZOXAZONE AND NITROINDAZOLES:TITL 3 CRYSTALLOGRAPHIC AND COMPUTATIONAL ANALYSES OFTITL 4 INHIBITOR POTENCYREF BIOCHEMISTRY V. 41 13915 2002REFN ISSN 0006-2960PMID 12437348DOI 10.1021/BI026313J Variant Set Distributions Ripley’s […]

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1IVH.A | IVD

General Structure Information 1ivh IVD structure of human isovaleryl-coa dehydrogenase at 2.6 angstroms resolution: structural basis for substrate specificity 2.6Å AUTH K.A.TIFFANY,D.L.ROBERTS,M.WANG,R.PASCHKE,AUTH 2 A.W.MOHSEN,J.VOCKLEY,J.J.KIMTITL STRUCTURE OF HUMAN ISOVALERYL-COA DEHYDROGENASE ATTITL 2 2.6 A RESOLUTION: STRUCTURAL BASIS FOR SUBSTRATETITL 3 SPECIFICITY,.REF BIOCHEMISTRY V. 36 8455 1997REFN ISSN 0006-2960PMID 9214289DOI 10.1021/BI970422U Variant Set Distributions Ripley’s K Analysis […]

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3UA5.B | CYP2B6

General Structure Information 3ua5 CYP2B6 crystal structure of p450 2b6 (y226h/k262r) in complex with two molecules of amlodipine 2.8Å AUTH M.B.SHAH,P.R.WILDERMAN,J.PASCUAL,Q.ZHANG,C.D.STOUT,AUTH 2 J.R.HALPERTTITL CONFORMATIONAL ADAPTATION OF HUMAN CYTOCHROME P450 2B6 ANDTITL 2 RABBIT CYTOCHROME P450 2B4 REVEALED UPON BINDING MULTIPLETITL 3 AMLODIPINE MOLECULES.REF BIOCHEMISTRY V. 51 7225 2012REFN ISSN 0006-2960PMID 22909231DOI 10.1021/BI300894Z Variant Set Distributions […]

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3SN5.B | CYP7A1

General Structure Information 3sn5 CYP7A1 crystal structure of human cyp7a1 in complex with cholest-4-en-3-one 2.75Å AUTH N.STRUSHKEVICH,W.TEMPEL,F.MACKENZIE,A.K.WERNIMONT,AUTH 2 C.H.ARROWSMITH,A.M.EDWARDS,C.BOUNTRA,J.WEIGELT,H.PARKTITL CRYSTAL STRUCTURE OF HUMAN CYP7A1 IN COMPLEX WITHTITL 2 CHOLEST-4-EN-3-ONEREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2R37.B | GPX3

General Structure Information 2r37 GPX3 crystal structure of human glutathione peroxidase 3 (selenocysteine to glycine mutant) 1.85Å AUTH E.S.PILKA,K.GUO,O.GILEADI,A.ROJKOWA,F.VON DELFT,A.C.W.PIKE,AUTH 2 K.L.KAVANAGH,C.JOHANNSON,M.SUNDSTROM,C.H.ARROWSMITH,AUTH 3 J.WEIGELT,A.M.EDWARDS,U.OPPERMANNTITL CRYSTAL STRUCTURE OF HUMAN GLUTATHIONE PEROXIDASE 3TITL 2 (SELENOCYSTEINE TO GLYCINE MUTANT).REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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1PJ2.A | ME2

General Structure Information 1pj2 ME2 crystal structure of human mitochondrial nad(p)+-dependent malic enzyme in a pentary complex with natural substrate malate, cofactor nadh, mn++, and allosteric activator fumarate 2.3Å AUTH X.TAO,Z.YANG,L.TONGTITL CRYSTAL STRUCTURES OF SUBSTRATE COMPLEXES OF MALICTITL 2 ENZYME AND INSIGHTS INTO THE CATALYTIC MECHANISM.REF STRUCTURE V. 11 1141 2003REFN ISSN 0969-2126PMID 12962632DOI 10.1016/S0969-2126(03)00168-0 […]

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2V60.A | MAOB

General Structure Information 2v60 MAOB structure of human mao b in complex with the selective inhibitor 7-(3-chlorobenzyloxy)-4-carboxaldehyde-coumarin 2.0Å AUTH C.BINDA,J.WANG,L.PISANI,C.CACCIA,A.CAROTTI,AUTH 2 P.SALVATI,D.E.EDMONDSON,A.MATTEVITITL STRUCTURES OF HUMAN MONOAMINE OXIDASE B COMPLEXESTITL 2 WITH SELECTIVE NONCOVALENT INHIBITORS: SAFINAMIDETITL 3 AND COUMARIN ANALOGS.REF J.MED.CHEM. V. 50 5848 2007REFN ISSN 0022-2623PMID 17915852DOI 10.1021/JM070677Y Variant Set Distributions Ripley’s K Analysis Plots […]

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2ACU.A | AKR1B1

General Structure Information 2acu AKR1B1 tyrosine-48 is the proton donor and histidine-110 directs substrate stereochemical selectivity in the reduction reaction of human aldose reductase: enzyme kinetics and the crystal structure of the y48h mutant enzyme 1.76Å AUTH K.M.BOHREN,C.E.GRIMSHAW,C.J.LAI,D.H.HARRISON,AUTH 2 D.RINGE,G.A.PETSKO,K.H.GABBAYTITL TYROSINE-48 IS THE PROTON DONOR AND HISTIDINE-110TITL 2 DIRECTS SUBSTRATE STEREOCHEMICAL SELECTIVITY INTITL 3 THE […]

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3QFC.A | POR

General Structure Information 3qfc POR crystal structure of human nadph-cytochrome p450 (v492e mutant) 1.8Å AUTH C.XIA,S.P.PANDA,C.C.MAROHNIC,P.MARTASEK,B.S.MASTERS,J.J.KIMTITL STRUCTURAL BASIS FOR HUMAN NADPH-CYTOCHROME P450TITL 2 OXIDOREDUCTASE DEFICIENCY.REF PROC.NATL.ACAD.SCI.USA V. 108 13486 2011REFN ISSN 0027-8424PMID 21808038DOI 10.1073/PNAS.1106632108 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1NFB.B | IMPDH2

General Structure Information 1nfb IMPDH2 ternary complex of the human type ii inosine monophosphate dedhydrogenase with 6cl-imp and nad 2.9Å AUTH D.RISAL,M.D.STRICKLER,B.M.GOLDSTEINTITL THE CONFORMATION OF NAD BOUND TO HUMAN INOSINE MONOPHOSPHATETITL 2 DEHYDROGENASE TYPE IIREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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