2VWM.A | F10

General Structure Information 2vwm F10 aminopyrrolidine factor xa inhibitor 1.96Å AUTH K.G.ZBINDEN,L.ANSELM,D.W.BANNER,J.M.BENZ,F.BLASCO,AUTH 2 G.DECORET,J.HIMBER,B.KUHN,N.PANDAY,F.RICKLIN,AUTH 3 P.RISCH,D.SCHLATTER,M.STAHL,S.THOMI,R.UNGER,W.HAAPTITL DESIGN OF NOVEL AMINOPYRROLIDINE FACTOR XATITL 2 INHIBITORS FROM A SCREENING HIT.REF EUR.J.MED.CHEM. V. 44 2787 2009REFN ISSN 0223-5234PMID 19200624DOI 10.1016/J.EJMECH.2008.12.025 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2ANW.A | KLKB1

General Structure Information 2anw KLKB1 expression, crystallization and three-dimensional structure of the catalytic domain of human plasma kallikrein: implications for structure-based design of protease inhibitors 1.85Å AUTH J.TANG,C.L.YU,S.R.WILLIAMS,E.SPRINGMAN,D.JEFFERY,AUTH 2 P.A.SPRENGELER,A.ESTEVEZ,J.SAMPANG,W.SHRADER,AUTH 3 J.SPENCER,W.YOUNG,M.MCGRATH,B.A.KATZTITL EXPRESSION, CRYSTALLIZATION, AND THREE-DIMENSIONALTITL 2 STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN PLASMATITL 3 KALLIKREIN.REF J.BIOL.CHEM. V. 280 41077 2005REFN ISSN 0021-9258PMID 16199530DOI […]

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3GXM.A | GBA

General Structure Information 3gxm GBA crystal structure of acid-beta-glucosidase at ph 4.5, phosphate crystallization condition 2.2Å AUTH R.L.LIEBERMAN,J.A.DAQUINO,D.RINGE,G.A.PETSKOTITL EFFECTS OF PH AND IMINOSUGAR PHARMACOLOGICAL CHAPERONES ONTITL 2 LYSOSOMAL GLYCOSIDASE STRUCTURE AND STABILITY.REF BIOCHEMISTRY V. 48 4816 2009REFN ISSN 0006-2960PMID 19374450DOI 10.1021/BI9002265 Variant Set Distributions Pathogenic Proximity Analysis Mapped Variants

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1ZED.A | ALPP

General Structure Information 1zed ALPP alkaline phosphatase from human placenta in complex with p- nitrophenyl-phosphonate 1.57Å AUTH P.LLINAS,E.A.STURA,A.MENEZ,Z.KISS,T.STIGBRAND,J.L.MILLAN,AUTH 2 M.H.LE DUTITL STRUCTURAL STUDIES OF HUMAN PLACENTAL ALKALINE PHOSPHATASETITL 2 IN COMPLEX WITH FUNCTIONAL LIGANDS.REF J.MOL.BIOL. V. 350 441 2005REFN ISSN 0022-2836PMID 15946677DOI 10.1016/J.JMB.2005.04.068 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity […]

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2XRC.A | CFI

General Structure Information 2xrc CFI human complement factor i 2.69Å AUTH P.ROVERSI,S.JOHNSON,J.J.CAESAR,F.MCLEAN,K.J.LEATH,AUTH 2 S.A.TSIFTSOGLOU,B.P.MORGAN,C.L.HARRIS,R.B.SIM,S.M.LEATITL STRUCTURAL BASIS FOR COMPLEMENT FACTOR I CONTROL AND ITSTITL 2 DISEASE-ASSOCIATED SEQUENCE POLYMORPHISMS.REF PROC.NATL.ACAD.SCI.USA V. 108 12839 2011REFN ISSN 0027-8424PMID 21768352DOI 10.1073/PNAS.1102167108 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1MFV.A | AMY1B

General Structure Information 1mfv AMY1B probing the role of a mobile loop in human slaivary amylase: structural studies on the loop-deleted enzyme 2.0Å AUTH N.RAMASUBBU,C.RAGUNATH,P.J.MISHRATITL PROBING THE ROLE OF A MOBILE LOOP IN SUBSTRATETITL 2 BINDING AND ENZYME ACTIVITY OF HUMAN SALIVARYTITL 3 AMYLASE.REF J.MOL.BIOL. V. 325 1061 2003REFN ISSN 0022-2836PMID 12527308DOI 10.1016/S0022-2836(02)01326-8 Variant Set […]

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1MFV.A | AMY1C

General Structure Information 1mfv AMY1C probing the role of a mobile loop in human slaivary amylase: structural studies on the loop-deleted enzyme 2.0Å AUTH N.RAMASUBBU,C.RAGUNATH,P.J.MISHRATITL PROBING THE ROLE OF A MOBILE LOOP IN SUBSTRATETITL 2 BINDING AND ENZYME ACTIVITY OF HUMAN SALIVARYTITL 3 AMYLASE.REF J.MOL.BIOL. V. 325 1061 2003REFN ISSN 0022-2836PMID 12527308DOI 10.1016/S0022-2836(02)01326-8 Variant Set […]

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1MFV.A | AMY1A

General Structure Information 1mfv AMY1A probing the role of a mobile loop in human slaivary amylase: structural studies on the loop-deleted enzyme 2.0Å AUTH N.RAMASUBBU,C.RAGUNATH,P.J.MISHRATITL PROBING THE ROLE OF A MOBILE LOOP IN SUBSTRATETITL 2 BINDING AND ENZYME ACTIVITY OF HUMAN SALIVARYTITL 3 AMYLASE.REF J.MOL.BIOL. V. 325 1061 2003REFN ISSN 0022-2836PMID 12527308DOI 10.1016/S0022-2836(02)01326-8 Variant Set […]

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3IJ9.A | AMY2A

General Structure Information 3ij9 AMY2A directed in situ elongation as a strategy to characterize the covalent glycosyl-enzyme catalytic intermediate of human pancreatic a-amylase 1.85Å AUTH R.ZHANG,C.LI,L.K.WILLIAMS,B.P.REMPEL,G.D.BRAYER,AUTH 2 S.G.WITHERSTITL DIRECTED IN SITU INHIBITOR ELONGATION AS ATITL 2 STRATEGY TO STRUCTURALLY CHARACTERIZE THE COVALENTTITL 3 GLYCOSYL-ENZYME INTERMEDIATE OF HUMAN PANCREATICTITL 4 ALPHA-AMYLASEREF BIOCHEMISTRY V. 48 10752 2009REFN […]

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3BT1.A | PLAU

General Structure Information 3bt1 PLAU structure of urokinase receptor, urokinase and vitronectin complex 2.8Å AUTH Q.HUAI,A.ZHOU,L.LIN,A.P.MAZAR,G.C.PARRY,J.CALLAHAN,D.E.SHAW,AUTH 2 B.FURIE,B.C.FURIE,M.HUANGTITL CRYSTAL STRUCTURES OF TWO HUMAN VITRONECTIN, UROKINASE ANDTITL 2 UROKINASE RECEPTOR COMPLEXESREF NAT.STRUCT.MOL.BIOL. V. 15 422 2008REFN ISSN 1545-9993PMID 18376415DOI 10.1038/NSMB.1404 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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