4L01.A | JAK1

General Structure Information 4l01 JAK1 crystal structure of the v658f apo jak1 pseudokinase domain 1.9Å AUTH A.V.TOMS,A.DESHPANDE,R.MCNALLY,Y.JEONG,J.M.ROGERS,C.U.KIM,AUTH 2 S.M.GRUNER,S.B.FICARRO,J.A.MARTO,M.SATTLER,J.D.GRIFFIN,AUTH 3 M.J.ECKTITL STRUCTURE OF A PSEUDOKINASE-DOMAIN SWITCH THAT CONTROLSTITL 2 ONCOGENIC ACTIVATION OF JAK KINASES.REF NAT.STRUCT.MOL.BIOL. V. 20 1221 2013REFN ISSN 1545-9993PMID 24013208DOI 10.1038/NSMB.2673 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3ZFM.A | EPHB2

General Structure Information 3zfm EPHB2 crystal structure of ephb2 2.27Å AUTH R.C.OVERMAN,J.E.DEBRECZENI,C.M.TRUMAN,M.S.MCALISTER,AUTH 2 T.K.ATTWOODTITL COMPLETING THE STRUCTURAL FAMILY PORTRAIT OF THE HUMAN EPHBTITL 2 TYROSINE KINASE DOMAINSREF PROTEIN SCI. V. 23 627 2014REFN ISSN 0961-8368PMID 24677421DOI 10.1002/PRO.2445 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2PVY.D | FGFR2

General Structure Information 2pvy FGFR2 crystal strucure of fgf receptor 2 (fgfr2) kinase domain harboring the pathogenic k659n mutation responsible for an unclassified craniosynostosis syndrome. 2.2Å AUTH H.CHEN,J.MA,W.LI,A.V.ELISEENKOVA,C.XU,T.A.NEUBERT,AUTH 2 W.T.MILLER,M.MOHAMMADITITL A MOLECULAR BRAKE IN THE KINASE HINGE REGION REGULATES THETITL 2 ACTIVITY OF RECEPTOR TYROSINE KINASES.REF MOL.CELL V. 27 717 2007REFN ISSN 1097-2765PMID 17803937DOI 10.1016/J.MOLCEL.2007.06.028 […]

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4L45.A | RPS6KB1

General Structure Information 4l45 RPS6KB1 crystal structures of human p70s6k1-t389e 2.9Å AUTH J.WANG,C.ZHONG,F.WANG,F.QU,J.DINGTITL CRYSTAL STRUCTURES OF S6K1 PROVIDE INSIGHTS INTO THETITL 2 REGULATION MECHANISM OF S6K1 BY THE HYDROPHOBIC MOTIFREF BIOCHEM.J. V. 454 39 2013REFN ISSN 0264-6021PMID 23731517DOI 10.1042/BJ20121863 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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4FV2.A | MAPK1

General Structure Information 4fv2 MAPK1 crystal structure of the erk2 complexed with ek5 2.0Å AUTH Y.N.KANG,J.A.STUCKEY,X.XIETITL CRYSTAL STRUCTURE OF THE ERK2 COMPLEXED WITH EK5REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3BBB.D | NME2

General Structure Information 3bbb NME2 crystal structure of the nm23-h2 transcription factor complex with dinucleotide d(ag) 1.3Å AUTH T.S.DEXHEIMER,S.S.CAREY,S.ZUOHE,V.M.GOKHALE,X.HU,L.B.MURATA,AUTH 2 E.M.MAES,A.WEICHSEL,D.SUN,E.J.MEUILLET,W.R.MONTFORT,AUTH 3 L.H.HURLEYTITL NM23-H2 MAY PLAY AN INDIRECT ROLE IN TRANSCRIPTIONALTITL 2 ACTIVATION OF C-MYC GENE EXPRESSION BUT DOES NOT CLEAVE THETITL 3 NUCLEASE HYPERSENSITIVE ELEMENT III1.REF MOL.CANCER THER. V. 8 1363 2009REFN ISSN 1535-7163PMID […]

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4K33.A | FGFR3

General Structure Information 4k33 FGFR3 crystal strucure of fgf receptor 3 (fgfr3) kinase domain harboring the k650e mutation, a gain-of-function mutation responsible for thanatophoric dysplasia type ii and spermatocytic seminoma 2.34Å AUTH Z.HUANG,H.CHEN,S.BLAIS,T.A.NEUBERT,X.LI,M.MOHAMMADITITL STRUCTURAL MIMICRY OF A-LOOP TYROSINE PHOSPHORYLATION BY ATITL 2 PATHOGENIC FGF RECEPTOR 3 MUTATION.REF STRUCTURE V. 21 1889 2013REFN ISSN 0969-2126PMID 23972473DOI […]

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1W2C.A | ITPKA

General Structure Information 1w2c ITPKA human inositol (1,4,5) trisphosphate 3-kinase complexed with mn2+/amppnp/ins(1,4,5)p3 1.95Å AUTH B.GONZALEZ,M.J.SCHELL,A.J.LETCHER,D.B.VEPRINTSEV,R.F.IRVINE,AUTH 2 R.L.WILLIAMSTITL STRUCTURE OF A HUMAN INOSITOL 1,4,5-TRISPHOSPHATE 3-KINASE;TITL 2 SUBSTRATE BINDING REVEALS WHY IT IS NOT A PHOSPHOINOSITIDETITL 3 3-KINASEREF MOL.CELL V. 15 689 2004REFN ISSN 1097-2765PMID 15350214DOI 10.1016/J.MOLCEL.2004.08.004 Variant Set Distributions Mapped Variants

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2E8N.A | EPHA2

General Structure Information 2e8n EPHA2 solution structure of the c-terminal sam-domain of ephaa2: ephrin type-a receptor 2 precursor (ec 2.7.10.1) -1.0Å AUTH A.K.GORONCY,M.SATO,S.KOSHIBA,M.INOUE,T.KIGAWA,AUTH 2 S.YOKOYAMATITL SOLUTION STRUCTURE OF THE C-TERMINAL SAM-DOMAIN OFTITL 2 EPHAA2: EPHRIN TYPE-A RECEPTOR 2 PRECURSOR (ECTITL 3 2.7.10.1)REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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1UCV.A | EPHA8

General Structure Information 1ucv EPHA8 sterile alpha motif (sam) domain of ephrin type-a receptor 8 -1.0Å AUTH A.GORONCY,T.KIGAWA,S.KOSHIBA,N.KOBAYASHI,N.TOCHIO,AUTH 2 M.INOUE,S.YOKOYAMATITL NMR STRUCTURE OF STERILE ALPHA MOTIF (SAM) DOMAINTITL 2 OF EPHRIN TYPE-A RECEPTOR 8REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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