4ACH.A | GSK3B

General Structure Information 4ach GSK3B gsk3b in complex with inhibitor 2.6Å AUTH S.BERG,M.BERGH,S.HELLBERG,K.HOGDIN,Y.LO-ALFREDSSON,AUTH 2 P.SODERMAN,S.VON BERG,T.WEIGELT,M.ORMO,Y.XUE,J.TUCKER,AUTH 3 J.NEELISSEN,E.JERNING,Y.NILSSON,R.BHATTITL DISCOVERY OF NOVEL POTENT AND HIGHLY SELECTIVE GLYCOGENTITL 2 SYNTHASE KINASE-3BETA (GSK3BETA) INHIBITORS FOR ALZHEIMERSTITL 3 DISEASE: DESIGN, SYNTHESIS, AND CHARACTERIZATION OFTITL 4 PYRAZINES.REF J.MED.CHEM. V. 55 9107 2012REFN ISSN 0022-2623PMID 22489897DOI 10.1021/JM201724M Variant Set Distributions Ripley’s […]

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3HHD.C | FASN

General Structure Information 3hhd FASN structure of the human fatty acid synthase ks-mat didomain as a framework for inhibitor design. 2.15Å AUTH G.PAPPENBERGER,J.BENZ,B.GSELL,M.HENNIG,A.RUF,AUTH 2 M.STIHLE,R.THOMA,M.G.RUDOLPHTITL STRUCTURE OF THE HUMAN FATTY ACID SYNTHASE KS-MATTITL 2 DIDOMAIN AS A FRAMEWORK FOR INHIBITOR DESIGN.REF J.MOL.BIOL. V. 397 508 2010REFN ISSN 0022-2836PMID 20132826DOI 10.1016/J.JMB.2010.01.066 Variant Set Distributions Ripley’s K […]

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2C9Y.A | AK2

General Structure Information 2c9y AK2 structure of human adenylate kinase 2 2.1Å AUTH G.BUNKOCZI,P.FILIPPAKOPOULOS,J.E.DEBRECZENI,A.TURNBULL,AUTH 2 E.PAPAGRIGORIOU,P.SAVITSKY,S.COLEBROOK,F.VON DELFT,AUTH 3 C.ARROWSMITH,A.EDWARDS,M.SUNDSTROM,J.WEIGELT,S.KNAPPTITL STRUCTURE OF HUMAN ADENYLATE KINASE 2REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3MX0.D | EFNA5

General Structure Information 3mx0 EFNA5 crystal structure of epha2 ectodomain in complex with ephrin-a5 3.51Å AUTH J.P.HIMANEN,L.YERMEKBAYEVA,P.W.JANES,J.R.WALKER,K.XU,AUTH 2 L.ATAPATTU,K.R.RAJASHANKAR,A.MENSINGA,M.LACKMANN,AUTH 3 D.B.NIKOLOV,S.DHE-PAGANONTITL ARCHITECTURE OF EPH RECEPTOR CLUSTERS.REF PROC.NATL.ACAD.SCI.USA V. 107 10860 2010REFN ISSN 0027-8424PMID 20505120DOI 10.1073/PNAS.1004148107 Variant Set Distributions Mapped Variants

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2WYA.C | HMGCS2

General Structure Information 2wya HMGCS2 crystal structure of human mitochondrial 3-hydroxy-3- methylglutaryl-coenzyme a synthase 2 (hmgcs2) 1.7Å AUTH N.SHAFQAT,A.TURNBULL,J.ZSCHOCKE,U.OPPERMANN,AUTH 2 W.W.YUETITL CRYSTAL STRUCTURES OF HUMAN HMG-COA SYNTHASETITL 2 ISOFORMS PROVIDE INSIGHTS INTO INHERITEDTITL 3 KETOGENESIS DISORDERS AND INHIBITOR DESIGN.REF J.MOL.BIOL. V. 398 497 2010REFN ISSN 0022-2836PMID 20346956DOI 10.1016/J.JMB.2010.03.034 Variant Set Distributions Ripley’s K Analysis Plots […]

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2COJ.B | BCAT1

General Structure Information 2coj BCAT1 crystal structure of reduced human cytosolic branched-chain aminotransferase complexed with gabapentin 2.4Å AUTH M.GOTO,I.MIYAHARA,K.HIROTSU,M.CONWAY,N.YENNAWAR,M.M.ISLAM,AUTH 2 S.M.HUTSONTITL STRUCTURAL DETERMINANTS FOR BRANCHED-CHAIN AMINOTRANSFERASETITL 2 ISOZYME-SPECIFIC INHIBITION BY THE ANTICONVULSANT DRUGTITL 3 GABAPENTINREF J.BIOL.CHEM. V. 280 37246 2005REFN ISSN 0021-9258PMID 16141215DOI 10.1074/JBC.M506486200 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic […]

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2H11.B | TPMT

General Structure Information 2h11 TPMT amino-terminal truncated thiopurine s-methyltransferase complexed with s-adenosyl-l-homocysteine 1.89Å AUTH J.R.HORTON,X.CHENGTITL AMINO-TERMINAL TRUNCATED THIOPURINETITL 2 S-METHYLTRANSFERASE COMPLEXED WITHTITL 3 S-ADENOSYL-L-HOMOCYSTEINEREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3E37.A | FNTA

General Structure Information 3e37 FNTA protein farnesyltransferase complexed with bisubstrate ethylenediamine scaffold inhibitor 5 1.8Å AUTH M.A.HAST,S.FLETCHER,C.G.CUMMINGS,E.E.PUSATERI,AUTH 2 M.A.BLASKOVICH,K.RIVAS,M.H.GELB,W.C.VAN VOORHIS,AUTH 3 S.M.SEBTI,A.D.HAMILTON,L.S.BEESETITL STRUCTURAL BASIS FOR BINDING AND SELECTIVITY OFTITL 2 ANTIMALARIAL AND ANTICANCER ETHYLENEDIAMINETITL 3 INHIBITORS TO PROTEIN FARNESYLTRANSFERASE.REF CHEM.BIOL. V. 16 181 2009REFN ISSN 1074-5521PMID 19246009DOI 10.1016/J.CHEMBIOL.2009.01.014 Variant Set Distributions Ripley’s K Analysis Plots […]

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3PFF.A | ACLY

General Structure Information 3pff ACLY truncated human atp-citrate lyase with adp and tartrate bound 2.3Å AUTH T.SUN,K.HAYAKAWA,M.E.FRASERTITL ADP-MG2+ BOUND TO THE ATP-GRASP DOMAIN OF ATP-CITRATE LYASE.REF ACTA CRYSTALLOGR.,SECT.F V. 67 1168 2011REFN ESSN 1744-3091PMID 22102020DOI 10.1107/S1744309111028363 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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1KO6.A | NUP98

General Structure Information 1ko6 NUP98 crystal structure of c-terminal autoproteolytic domain of nucleoporin nup98 3.0Å AUTH A.E.HODEL,M.R.HODEL,E.R.GRIFFIS,K.A.HENNIG,AUTH 2 G.A.RATNER,S.XU,M.A.POWERSTITL THE THREE-DIMENSIONAL STRUCTURE OF THETITL 2 AUTOPROTEOLYTIC, NUCLEAR PORE-TARGETING DOMAIN OFTITL 3 THE HUMAN NUCLEOPORIN NUP98.REF MOL.CELL V. 10 347 2002REFN ISSN 1097-2765PMID 12191480DOI 10.1016/S1097-2765(02)00589-0 Variant Set Distributions Mapped Variants

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