3KXO.A | HPGDS

General Structure Information 3kxo HPGDS an orally active inhibitor bound at the active site of hpgds 2.1Å AUTH C.P.CARRON,J.I.TRUJILLO,K.L.OLSON,W.HUANG,B.C.HAMPER,T.DICE,AUTH 2 B.E.NEAL,M.J.PELC,J.DAY,D.C.ROHRER,J.R.KIEFER,J.B.MOON,AUTH 3 B.A.SCHWEITZER,T.D.BLAKE,S.R.TURNER,R.WOERNDLE,B.L.CASE,AUTH 4 C.P.BONO,V.M.DILWORTH,C.L.FUNCKES-SHIPPY,B.L.HOOD,AUTH 5 G.M.JEROME,C.M.KORNMEIER,M.R.RADABAUGH,M.L.WILLIAMS,AUTH 6 M.S.DAVIES,C.D.WEGNER,D.J.WELSCH,W.M.ABRAHAM,C.J.WARREN,AUTH 7 M.E.DOWTY,F.HUA,A.ZUTSHI,J.Z.YANG,A.THORARENSENTITL DISCOVERY OF AN ORAL POTENT SELECTIVE INHIBITOR OFTITL 2 HEMATOPOIETIC PROSTAGLANDIN D SYNTHASEREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant […]

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4L6Q.A | ROCK2

General Structure Information 4l6q ROCK2 rock2 in complex with benzoxaborole 2.79Å AUTH T.AKAMA,C.DONG,C.VIRTUCIO,D.SULLIVAN,Y.ZHOU,Y.K.ZHANG,AUTH 2 F.ROCK,Y.FREUND,L.LIU,W.BU,A.WU,X.Q.FAN,K.JARNAGINTITL LINKING PHENOTYPE TO KINASE: IDENTIFICATION OF A NOVELTITL 2 BENZOXABOROLE HINGE-BINDING MOTIF FOR KINASE INHIBITION ANDTITL 3 DEVELOPMENT OF HIGH-POTENCY RHO KINASE INHIBITORS.REF J.PHARMACOL.EXP.THER. V. 347 615 2013REFN ISSN 0022-3565PMID 24049062DOI 10.1124/JPET.113.207662 Variant Set Distributions Ripley’s K Analysis Plots Variant […]

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3AP1.B | TPST2

General Structure Information 3ap1 TPST2 crystal structure of human tyrosylprotein sulfotransferase-2 complexed with pap and c4 peptide 1.9Å AUTH T.TERAMOTO,Y.FUJIKAWA,Y.KAWAGUCHI,K.KUROGI,M.SOEJIMA,AUTH 2 R.ADACHI,Y.NAKANISHI,E.MISHIRO-SATO,M.C.LIU,Y.SAKAKIBARA,AUTH 3 M.SUIKO,M.KIMURA,Y.KAKUTATITL CRYSTAL STRUCTURE OF HUMAN TYROSYLPROTEIN SULFOTRANSFERASE-2TITL 2 REVEALS THE MECHANISM OF PROTEIN TYROSINE SULFATIONTITL 3 REACTION.REF NAT COMMUN V. 4 1572 2013REFN ESSN 2041-1723PMID 23481380DOI 10.1038/NCOMMS2593 Variant Set Distributions Ripley’s K […]

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4F91.B | SNRNP200

General Structure Information 4f91 SNRNP200 brr2 helicase region 2.7Å AUTH K.F.SANTOS,S.M.JOVIN,G.WEBER,V.PENA,R.LUHRMANN,M.C.WAHLTITL STRUCTURAL BASIS FOR FUNCTIONAL COOPERATION BETWEEN TANDEMTITL 2 HELICASE CASSETTES IN BRR2-MEDIATED REMODELING OF THETITL 3 SPLICEOSOME.REF PROC.NATL.ACAD.SCI.USA V. 109 17418 2012REFN ISSN 0027-8424PMID 23045696DOI 10.1073/PNAS.1208098109 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2I3Y.A | GPX5

General Structure Information 2i3y GPX5 crystal structure of human glutathione peroxidase 5 2.0Å AUTH K.L.KAVANAGH,U.OPPERMANNTITL CRYSTAL STRUCTURE OF HUMAN GLUTATHIONE PEROXIDASE 5REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1WRY.A | SH3BGRL

General Structure Information 1wry SH3BGRL solution structure of the sh3 domain-binding glutamic acid- rich-like protein -1.0Å AUTH K.INOUE,K.MIYAMOTO,T.NAGASHIMA,F.HAYASHI,T.KIGAWA,AUTH 2 S.YOKOYAMATITL SOLUTION STRUCTURE OF THE SH3 DOMAIN-BINDINGTITL 2 GLUTAMIC ACID-RICH-LIKE PROTEINREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3PU8.B | PHF2

General Structure Information 3pu8 PHF2 phf2 jumonji-nog-fe(ii) complex 1.94Å AUTH J.R.HORTON,A.K.UPADHYAY,H.HASHIMOTO,X.ZHANG,X.CHENGTITL STRUCTURAL BASIS FOR HUMAN PHF2 JUMONJI DOMAIN INTERACTIONTITL 2 WITH METAL IONS.REF J.MOL.BIOL. V. 406 1 2011REFN ISSN 0022-2836PMID 21167174DOI 10.1016/J.JMB.2010.12.013 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3EG9.B | SEC24D

General Structure Information 3eg9 SEC24D crystal structure of the mammalian copii-coat protein sec23/24 bound to the transport signal sequence of membrin 3.0Å AUTH J.D.MANCIAS,J.GOLDBERGTITL STRUCTURAL BASIS OF CARGO MEMBRANE PROTEIN DISCRIMINATION BYTITL 2 THE HUMAN COPII COAT MACHINERY.REF EMBO J. V. 27 2918 2008REFN ISSN 0261-4189PMID 18843296DOI 10.1038/EMBOJ.2008.208 Variant Set Distributions Ripley’s K Analysis Plots […]

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3LFV.B | PDE5A

General Structure Information 3lfv PDE5A crystal structure of unliganded pde5a gaf domain 2.8Å AUTH H.WANG,H.ROBINSON,H.KETITL CONFORMATION CHANGES, N-TERMINAL INVOLVEMENT, AND CGMPTITL 2 SIGNAL RELAY IN THE PHOSPHODIESTERASE-5 GAF DOMAIN.REF J.BIOL.CHEM. V. 285 38149 2010REFN ISSN 0021-9258PMID 20861010DOI 10.1074/JBC.M110.141614 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3HU6.A | SPOP

General Structure Information 3hu6 SPOP structures of spop-substrate complexes: insights into molecular architectures of btb-cul3 ubiquitin ligases: spopmathx/btb/3-box-pucsbc1 2.7Å AUTH M.ZHUANG,M.F.CALABRESE,J.LIU,M.B.WADDELL,A.NOURSE,AUTH 2 M.HAMMEL,D.J.MILLER,H.WALDEN,D.M.DUDA,S.N.SEYEDIN,AUTH 3 T.HOGGARD,J.W.HARPER,K.P.WHITE,B.A.SCHULMANTITL STRUCTURES OF SPOP-SUBSTRATE COMPLEXES: INSIGHTSTITL 2 INTO MOLECULAR ARCHITECTURES OF BTB-CUL3 UBIQUITINTITL 3 LIGASES.REF MOL.CELL V. 36 39 2009REFN ISSN 1097-2765PMID 19818708DOI 10.1016/J.MOLCEL.2009.09.022 Variant Set Distributions Ripley’s K Analysis Plots […]

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