3R01.A | PIM1

General Structure Information 3r01 PIM1 the discovery of novel benzofuran-2-carboxylic acids as potent pim-1 inhibitors 2.6Å AUTH Y.XIANG,B.HIRTH,G.ASMUSSEN,H.P.BIEMANN,K.A.BISHOP,A.GOOD,AUTH 2 M.FITZGERALD,T.GLADYSHEVA,A.JAIN,K.JANCSICS,J.LIU,M.METZ,AUTH 3 A.PAPOULIS,R.SKERLJ,J.D.STEPP,R.R.WEITITL THE DISCOVERY OF NOVEL BENZOFURAN-2-CARBOXYLIC ACIDS ASTITL 2 POTENT PIM-1 INHIBITORS.REF BIOORG.MED.CHEM.LETT. V. 21 3050 2011REFN ISSN 0960-894XPMID 21507633DOI 10.1016/J.BMCL.2011.03.030 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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4DM9.A | UCHL1

General Structure Information 4dm9 UCHL1 the crystal structure of ubiquitin carboxy-terminal hydrolase l1 (uchl1) bound to a tripeptide fluoromethyl ketone z-vae(ome)-fmk 2.35Å AUTH C.W.DAVIES,J.CHANEY,G.KORBEL,D.RINGE,G.A.PETSKO,H.PLOEGH,AUTH 2 C.DASTITL THE CO-CRYSTAL STRUCTURE OF UBIQUITIN CARBOXY-TERMINALTITL 2 HYDROLASE L1 (UCHL1) WITH A TRIPEPTIDE FLUOROMETHYL KETONETITL 3 (Z-VAE(OME)-FMK).REF BIOORG.MED.CHEM.LETT. V. 22 3900 2012REFN ISSN 0960-894XPMID 22617491DOI 10.1016/J.BMCL.2012.04.124 Variant Set Distributions […]

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1PLS.A | PLEK

General Structure Information 1pls PLEK solution structure of a pleckstrin homology domain -1.0Å AUTH H.S.YOON,P.J.HAJDUK,A.M.PETROS,E.T.OLEJNICZAK,AUTH 2 R.P.MEADOWS,S.W.FESIKTITL SOLUTION STRUCTURE OF A PLECKSTRIN-HOMOLOGY DOMAIN.REF NATURE V. 369 672 1994REFN ISSN 0028-0836PMID 8208296DOI 10.1038/369672A0 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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2FGI.A | FGFR1

General Structure Information 2fgi FGFR1 crystal structure of the tyrosine kinase domain of fgf receptor 1 in complex with inhibitor pd173074 2.5Å AUTH M.MOHAMMADI,S.FROUM,J.M.HAMBY,M.C.SCHROEDER,AUTH 2 R.L.PANEK,G.H.LU,A.V.ELISEENKOVA,D.GREEN,AUTH 3 J.SCHLESSINGER,S.R.HUBBARDTITL CRYSTAL STRUCTURE OF AN ANGIOGENESIS INHIBITORTITL 2 BOUND TO THE FGF RECEPTOR TYROSINE KINASE DOMAIN.REF EMBO J. V. 17 5896 1998REFN ISSN 0261-4189PMID 9774334DOI 10.1093/EMBOJ/17.20.5896 Variant Set […]

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4GLP.A | CD14

General Structure Information 4glp CD14 the crystal structure of soluble human cd14 reveals a bent solenoid with a hydrophobic amino-terminal pocket. 4.0Å AUTH S.L.KELLEY,T.LUKK,S.K.NAIR,R.I.TAPPINGTITL THE CRYSTAL STRUCTURE OF HUMAN SOLUBLE CD14 REVEALS A BENTTITL 2 SOLENOID WITH A HYDROPHOBIC AMINO-TERMINAL POCKET.REF J.IMMUNOL. V. 190 1304 2013REFN ISSN 0022-1767PMID 23264655DOI 10.4049/JIMMUNOL.1202446 Variant Set Distributions Ripley’s K […]

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1XFB.D | ALDOC

General Structure Information 1xfb ALDOC human brain fructose 1,6-(bis)phosphate aldolase (c isozyme) 3.0Å AUTH T.L.ARAKAKI,J.A.PEZZA,M.A.CRONIN,C.E.HOPKINS,AUTH 2 D.B.ZIMMER,D.R.TOLAN,K.N.ALLENTITL STRUCTURE OF HUMAN BRAIN FRUCTOSETITL 2 1,6-(BIS)PHOSPHATE ALDOLASE: LINKING ISOZYMETITL 3 STRUCTURE WITH FUNCTIONREF PROTEIN SCI. V. 13 3077 2004REFN ISSN 0961-8368PMID 15537755DOI 10.1110/PS.04915904 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped […]

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2OBD.A | CETP

General Structure Information 2obd CETP crystal structure of cholesteryl ester transfer protein 2.1Å AUTH X.QIU,A.MISTRY,M.J.AMMIRATI,B.A.CHRUNYK,R.W.CLARK,AUTH 2 Y.CONG,J.S.CULP,D.E.DANLEY,T.B.FREEMAN,AUTH 3 K.F.GEOGHEGAN,M.C.GRIFFOR,S.J.HAWRYLIK,C.M.HAYWARD,AUTH 4 P.HENSLEY,L.R.HOTH,G.A.KARAM,M.E.LIRA,D.B.LLOYD,AUTH 5 K.M.MCGRATH,K.J.STUTZMAN-ENGWALL,A.K.SUBASHI,AUTH 6 T.A.SUBASHI,J.F.THOMPSON,I.K.WANG,H.ZHAO,A.P.SEDDONTITL CRYSTAL STRUCTURE OF CHOLESTERYL ESTER TRANSFERTITL 2 PROTEIN REVEALS A LONG TUNNEL AND FOUR BOUND LIPIDTITL 3 MOLECULES.REF NAT.STRUCT.MOL.BIOL. V. 14 106 2007REFN ISSN 1545-9993PMID 17237796DOI 10.1038/NSMB1197 Variant Set Distributions […]

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3E04.C | FH

General Structure Information 3e04 FH crystal structure of human fumarate hydratase 1.95Å AUTH K.L.KAVANAGH,S.PICAUD,E.S.PILKA,W.W.YUE,A.K.ROOS,AUTH 2 P.FILIPPAKOPOULOS,F.VON DELFT,C.H.ARROWSMITH,M.WIKSTROM,AUTH 3 A.M.EDWARDS,C.BOUNTRA,U.OPPERMANN,AUTH 4 STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL CRYSTAL STRUCTURE OF HUMAN FUMARATE HYDRATASEREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3RHK.B | MET

General Structure Information 3rhk MET crystal structure of the catalytic domain of c-met kinase in complex with arq 197 1.94Å AUTH S.EATHIRAJ,R.PALMA,E.VOLCKOVA,M.HIRSCHI,D.S.FRANCE,AUTH 2 M.A.ASHWELL,T.C.CHANTITL DISCOVERY OF A NOVEL MODE OF PROTEIN KINASE INHIBITIONTITL 2 CHARACTERIZED BY THE MECHANISM OF INHIBITION OF HUMANTITL 3 MESENCHYMAL-EPITHELIAL TRANSITION FACTOR (C-MET) PROTEINTITL 4 AUTOPHOSPHORYLATION BY ARQ 197.REF J.BIOL.CHEM. V. […]

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1HUP.A | MBL2

General Structure Information 1hup MBL2 human mannose binding protein carbohydrate recognition domain trimerizes through a triple alpha-helical coiled-coil 2.5Å AUTH S.SHERIFF,C.Y.CHANG,R.A.EZEKOWITZTITL HUMAN MANNOSE-BINDING PROTEIN CARBOHYDRATE RECOGNITIONTITL 2 DOMAIN TRIMERIZES THROUGH A TRIPLE ALPHA-HELICALTITL 3 COILED-COIL.REF NAT.STRUCT.BIOL. V. 1 789 1994REFN ISSN 1072-8368PMID 7634089DOI 10.1038/NSB1194-789 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped […]

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