3TXO.A | PRKCH

General Structure Information 3txo PRKCH pkc eta kinase in complex with a naphthyridine 2.05Å AUTH M.J.VAN EIS,J.P.EVENOU,P.FLOERSHEIM,C.GAUL,S.W.COWAN-JACOB,AUTH 2 L.MONOVICH,G.RUMMEL,W.SCHULER,W.STARK,A.STRAUSS,A.MATT,AUTH 3 E.VANGREVELINGHE,J.WAGNER,N.SOLDERMANNTITL 2,6-NAPHTHYRIDINES AS POTENT AND SELECTIVE INHIBITORS OF THETITL 2 NOVEL PROTEIN KINASE C ISOZYMES.REF BIOORG.MED.CHEM.LETT. V. 21 7367 2011REFN ISSN 0960-894XPMID 22078216DOI 10.1016/J.BMCL.2011.10.025 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped […]

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4BGC.A | KCNA3

General Structure Information 4bgc KCNA3 t1 domain of the renal potassium channel kv1.3 1.2Å AUTH W.KREMER,M.WEYAND,A.WINKLMEIER,C.SCHREIER,H.R.KALBITZERTITL 1.2 A X-RAY STRUCTURE OF THE RENAL POTASSIUM CHANNEL KV1.3TITL 2 T1 DOMAIN.REF PROTEIN J. V. 32 533 2013REFN ISSN 1572-3887PMID 24114469DOI 10.1007/S10930-013-9513-2 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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4HC7.A | GATA3

General Structure Information 4hc7 GATA3 crystal structure of the full dna binding domain of gata3-complex 2 2.65Å AUTH Y.CHEN,D.L.BATES,R.DEY,P.H.CHEN,A.C.MACHADO,AUTH 2 I.A.LAIRD-OFFRINGA,R.ROHS,L.CHENTITL DNA BINDING BY GATA TRANSCRIPTION FACTOR SUGGESTS MECHANISMSTITL 2 OF DNA LOOPING AND LONG-RANGE GENE REGULATION.REF CELL REP V. 2 1197 2012REFN ESSN 2211-1247PMID 23142663DOI 10.1016/J.CELREP.2012.10.012 Variant Set Distributions Ripley’s K Analysis Plots Variant […]

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1FGU.B | RPA1

General Structure Information 1fgu RPA1 ssdna-binding domain of the large subunit of replication protein a 2.5Å AUTH E.BOCHKAREVA,V.BELEGU,S.KOROLEV,A.BOCHKAREVTITL STRUCTURE OF THE MAJOR SINGLE-STRANDED DNA-BINDINGTITL 2 DOMAIN OF REPLICATION PROTEIN A SUGGESTS A DYNAMICTITL 3 MECHANISM FOR DNA BINDING.REF EMBO J. V. 20 612 2001REFN ISSN 0261-4189PMID 11157767DOI 10.1093/EMBOJ/20.3.612 Variant Set Distributions Ripley’s K Analysis Plots […]

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4AWN.A | DNASE1

General Structure Information 4awn DNASE1 structure of recombinant human dnase i (rhdnasei) in complex with magnesium and phosphate. 1.95Å AUTH G.PARSIEGLA,C.NOGUERE,L.SANTELL,R.A.LAZARUS,Y.BOURNETITL THE STRUCTURE OF HUMAN DNASE I BOUND TO MAGNESIUM ANDTITL 2 PHOSPHATE IONS POINTS TO A CATALYTIC MECHANISM COMMON TOTITL 3 MEMBERS OF THE DNASE I-LIKE SUPERFAMILY.REF BIOCHEMISTRY V. 51 10250 2012REFN ISSN 0006-2960PMID […]

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2NPP.A | PPP2R1A

General Structure Information 2npp PPP2R1A structure of the protein phosphatase 2a holoenzyme 3.3Å AUTH Y.XU,Y.XING,Y.CHEN,Y.CHAO,Z.LIN,E.FAN,J.W.YU,S.STRACK,AUTH 2 P.D.JEFFREY,Y.SHITITL STRUCTURE OF THE PROTEIN PHOSPHATASE 2A HOLOENZYMEREF CELL(CAMBRIDGE,MASS.) V. 127 1239 2006REFN ISSN 0092-8674PMID 17174897DOI 10.1016/J.CELL.2006.11.033 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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1M9K.B | NOS3

General Structure Information 1m9k NOS3 human endothelial nitric oxide synthase with 7- nitroindazole bound 2.01Å AUTH R.J.ROSENFELD,E.D.GARCIN,K.PANDA,G.ANDERSSON,AUTH 2 A.ABERG,A.V.WALLACE,G.M.MORRIS,A.J.OLSON,AUTH 3 D.J.STUEHR,J.A.TAINER,E.D.GETZOFFTITL CONFORMATIONAL CHANGES IN NITRIC OXIDE SYNTHASESTITL 2 INDUCED BY CHLORZOXAZONE AND NITROINDAZOLES:TITL 3 CRYSTALLOGRAPHIC AND COMPUTATIONAL ANALYSES OFTITL 4 INHIBITOR POTENCYREF BIOCHEMISTRY V. 41 13915 2002REFN ISSN 0006-2960PMID 12437348DOI 10.1021/BI026313J Variant Set Distributions Ripley’s […]

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3V4P.D | ITGB7

General Structure Information 3v4p ITGB7 crystal structure of a4b7 headpiece complexed with fab act-1 3.15Å AUTH Y.YU,J.ZHU,L.Z.MI,T.WALZ,H.SUN,J.CHEN,T.A.SPRINGERTITL STRUCTURAL SPECIALIZATIONS OF A4B7, AN INTEGRIN THATTITL 2 MEDIATES ROLLING ADHESIONREF J.CELL BIOL. V. 196 131 2012REFN ISSN 0021-9525PMID 22232704DOI 10.1083/JCB.201110023 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1APY.A | AGA

General Structure Information 1apy AGA human aspartylglucosaminidase 2.0Å AUTH C.OINONEN,R.TIKKANEN,J.ROUVINEN,L.PELTONENTITL THREE-DIMENSIONAL STRUCTURE OF HUMAN LYSOSOMALTITL 2 ASPARTYLGLUCOSAMINIDASE.REF NAT.STRUCT.BIOL. V. 2 1102 1995REFN ISSN 1072-8368PMID 8846222DOI 10.1038/NSB1295-1102 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1IVH.A | IVD

General Structure Information 1ivh IVD structure of human isovaleryl-coa dehydrogenase at 2.6 angstroms resolution: structural basis for substrate specificity 2.6Å AUTH K.A.TIFFANY,D.L.ROBERTS,M.WANG,R.PASCHKE,AUTH 2 A.W.MOHSEN,J.VOCKLEY,J.J.KIMTITL STRUCTURE OF HUMAN ISOVALERYL-COA DEHYDROGENASE ATTITL 2 2.6 A RESOLUTION: STRUCTURAL BASIS FOR SUBSTRATETITL 3 SPECIFICITY,.REF BIOCHEMISTRY V. 36 8455 1997REFN ISSN 0006-2960PMID 9214289DOI 10.1021/BI970422U Variant Set Distributions Ripley’s K Analysis […]

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