2XAH.B | RCOR1

General Structure Information 2xah RCOR1 crystal structure of lsd1-corest in complex with (+)- trans-2-phenylcyclopropyl-1-amine 3.1Å AUTH C.BINDA,S.VALENTE,M.ROMANENGHI,S.PILOTTO,R.CIRILLI,AUTH 2 A.KARYTINOS,G.CIOSSANI,O.A.BOTRUGNO,F.FORNERIS,AUTH 3 M.TARDUGNO,D.E.EDMONDSON,S.MINUCCI,A.MATTEVI,A.MAITITL BIOCHEMICAL, STRUCTURAL, AND BIOLOGICAL EVALUATIONTITL 2 OF TRANYLCYPROMINE DERIVATIVES AS INHIBITORS OFTITL 3 HISTONE DEMETHYLASES LSD1 AND LSD2.REF J.AM.CHEM.SOC. V. 132 6827 2010REFN ISSN 0002-7863PMID 20415477DOI 10.1021/JA101557K Variant Set Distributions Mapped Variants

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3HD6.A | RHCG

General Structure Information 3hd6 RHCG crystal structure of the human rhesus glycoprotein rhcg 2.1Å AUTH F.GRUSWITZ,S.CHAUDHARY,J.D.HO,A.SCHLESSINGER,B.PEZESHKI,AUTH 2 C.M.HO,A.SALI,C.M.WESTHOFF,R.M.STROUDTITL FUNCTION OF HUMAN RH BASED ON STRUCTURE OF RHCG AT 2.1 A.REF PROC.NATL.ACAD.SCI.USA V. 107 9638 2010REFN ISSN 0027-8424PMID 20457942DOI 10.1073/PNAS.1003587107 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2CP3.A | CLIP2

General Structure Information 2cp3 CLIP2 solution structure of the 2nd cap-gly domain in human clip- 115/cyln2 -1.0Å AUTH K.SAITO,S.KOSHIBA,M.INOUE,T.KIGAWA,S.YOKOYAMATITL SOLUTION STRUCTURE OF THE 2ND CAP-GLY DOMAIN INTITL 2 HUMAN CLIP-115/CYLN2REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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4IR4.A | BAZ2B

General Structure Information 4ir4 BAZ2B crystal structure of the bromodomain of human baz2b in complex with 1- [7-(morpholin-4-yl)-1-(pyridin-2-yl)indolizin-3-yl]ethanone (gsk2834113a) 2.05Å AUTH P.CHEN,A.CHAIKUAD,P.BAMBOROUGH,M.BANTSCHEFF,C.BOUNTRA,AUTH 2 C.W.CHUNG,O.FEDOROV,P.GRANDI,D.JUNG,R.LESNIAK,M.LINDON,AUTH 3 S.MULLER,M.PHILPOTT,R.PRINJHA,C.ROGERS,C.SELENSKI,C.TALLANT,AUTH 4 T.WERNER,T.M.WILLSON,S.KNAPP,D.H.DREWRYTITL DISCOVERY AND CHARACTERIZATION OF GSK2801, A SELECTIVETITL 2 CHEMICAL PROBE FOR THE BROMODOMAINS BAZ2A AND BAZ2B.REF J.MED.CHEM. 2015REFN ISSN 0022-2623PMID 25799074DOI 10.1021/ACS.JMEDCHEM.5B00209 Variant Set Distributions Mapped Variants

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4I6H.A | PLK2

General Structure Information 4i6h PLK2 selective & brain-permeable polo-like kinase-2 (plk-2) inhibitors that reduce alpha-synuclein phosphorylation in rat brain 1.91Å AUTH D.L.AUBELE,R.K.HOM,M.ADLER,R.A.GALEMMO,S.BOWERS,A.P.TRUONG,AUTH 2 H.PAN,P.BEROZA,R.J.NEITZ,N.YAO,M.LIN,G.TONN,H.ZHANG,AUTH 3 M.P.BOVA,Z.REN,D.TAM,L.RUSLIM,J.BAKER,L.DIEP,K.FITZGERALD,AUTH 4 J.HOFFMAN,R.MOTTER,D.FAUSS,P.TANAKA,M.DAPPEN,J.JAGODZINSKI,AUTH 5 W.CHAN,A.W.KONRADI,L.LATIMER,Y.L.ZHU,H.L.SHAM,J.P.ANDERSON,AUTH 6 M.BERGERON,D.R.ARTISTITL SELECTIVE & BRAIN-PERMEABLE POLO-LIKE KINASE-2 (PLK-2)TITL 2 INHIBITORS THAT REDUCE ALPHA-SYNUCLEIN PHOSPHORYLATION INTITL 3 RAT BRAINREF CHEMMEDCHEM V. 8 1295 2013REFN ISSN 1860-7179PMID […]

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2D86.A | VAV3

General Structure Information 2d86 VAV3 solution structure of the ch domain from human vav-3 protein -1.0Å AUTH T.TOMIZAWA,T.KIGAWA,S.KOSHIBA,M.INOUE,S.YOKOYAMATITL SOLUTION STRUCTURE OF THE CH DOMAIN FROM HUMANTITL 2 VAV-3 PROTEINREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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4F3T.A | AGO2

General Structure Information 4f3t AGO2 human argonaute-2 – mir-20a complex 2.25Å AUTH E.ELKAYAM,C.D.KUHN,A.TOCILJ,A.D.HAASE,E.M.GREENE,G.J.HANNON,AUTH 2 L.JOSHUA-TORTITL THE STRUCTURE OF HUMAN ARGONAUTE-2 IN COMPLEX WITH MIR-20A.REF CELL(CAMBRIDGE,MASS.) V. 150 100 2012REFN ISSN 0092-8674PMID 22682761DOI 10.1016/J.CELL.2012.05.017 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3K0W.A | MALT1

General Structure Information 3k0w MALT1 crystal structure of the tandem ig-like c2-type 2 domains of the human mucosa-associated lymphoid tissue lymphoma translocation protein 1 2.8Å AUTH J.R.WALKER,L.QIU,C.BUTLER-COLE,C.BOUNTRA,J.WEIGELT,AUTH 2 C.H.ARROWSMITH,A.M.EDWARDS,A.BOCHKAREV,AUTH 3 S.DHE-PAGANONTITL STRUCTURE OF THE TANDEM IG-LIKE C2-TYPE 2 DOMAINSTITL 2 OF THE HUMAN MUCOSA-ASSOCIATED LYMPHOID TISSUETITL 3 LYMPHOMA TRANSLOCATION PROTEIN 1.REF TO BE PUBLISHEDREFN Variant […]

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4KRF.A | AGO1

General Structure Information 4krf AGO1 structure of human argonaute-1 let-7 complex 2.1Å AUTH C.R.FAEHNLE,E.ELKAYAM,A.D.HAASE,G.J.HANNON,L.JOSHUA-TORTITL THE MAKING OF A SLICER: ACTIVATION OF HUMAN ARGONAUTE-1.REF CELL REP V. 3 1901 2013REFN ESSN 2211-1247PMID 23746446DOI 10.1016/J.CELREP.2013.05.033 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3G5C.B | ADAM22

General Structure Information 3g5c ADAM22 structural and biochemical studies on the ectodomain of human adam22 2.36Å AUTH H.LIU,A.SHIM,X.CHEN,X.HETITL STRUCTURAL AND BIOCHEMICAL STUDIES ON THE ECTODOMAIN OFTITL 2 HUMAN ADAM22REF J.BIOL.CHEM. 2009REFN ESSN 1083-351X Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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