2XAH.B | RCOR1

General Structure Information

PDB ID 2xah
HGNC Gene Label(s) RCOR1
Structure Name crystal structure of lsd1-corest in complex with (+)- trans-2-phenylcyclopropyl-1-amine
Resolution 3.1Å
Reference AUTH C.BINDA,S.VALENTE,M.ROMANENGHI,S.PILOTTO,R.CIRILLI,AUTH 2 A.KARYTINOS,G.CIOSSANI,O.A.BOTRUGNO,F.FORNERIS,AUTH 3 M.TARDUGNO,D.E.EDMONDSON,S.MINUCCI,A.MATTEVI,A.MAITITL BIOCHEMICAL, STRUCTURAL, AND BIOLOGICAL EVALUATIONTITL 2 OF TRANYLCYPROMINE DERIVATIVES AS INHIBITORS OFTITL 3 HISTONE DEMETHYLASES LSD1 AND LSD2.REF J.AM.CHEM.SOC. V. 132 6827 2010REFN ISSN 0002-7863PMID 20415477DOI 10.1021/JA101557K

Variant Set Distributions

ExAC Variants

Number Of Residues 133
Number Of SNVs 20
Number Of Permutations 8433
Optimal Distance Threshold 6.0
K Statistic 0.042
p-value 0.977

Mapped Variants

[+] ExAC Missense Variants