3KVQ.A | KDR

General Structure Information 3kvq KDR crystal structure of vegfr2 extracellular domain d7 2.7Å AUTH Y.YANG,P.XIE,Y.OPATOWSKY,J.SCHLESSINGERTITL DIRECT CONTACTS BETWEEN EXTRACELLULARTITL 2 MEMBRANE-PROXIMAL DOMAINS ARE REQUIRED FOR VEGFTITL 3 RECEPTOR ACTIVATION AND CELL SIGNALINGREF PROC.NATL.ACAD.SCI.USA V. 107 1906 2010REFN ISSN 0027-8424PMID 20080685DOI 10.1073/PNAS.0914052107 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped […]

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3EAC.A | CSK

General Structure Information 3eac CSK crystal structure of sh2 domain of human csk (carboxyl-terminal src kinase), oxidized form. 1.37Å AUTH D.LIU,R.D.SEIDEL,D.COWBURNTITL OBSERVATION OF DOMAIN INTERACTIONS IN PROTEIN TYROSINETITL 2 KINASE CSK BY SEGMENTAL LABELING NMRREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2XYN.B | ABL2

General Structure Information 2xyn ABL2 human abl2 in complex with aurora kinase inhibitor vx-680 2.81Å AUTH E.SALAH,E.UGOCHUKWU,A.J.BARR,F.VON DELFT,S.KNAPP,AUTH 2 J.M.ELKINSTITL CRYSTAL STRUCTURES OF ABL-RELATED GENE (ABL2) INTITL 2 COMPLEX WITH IMATINIB, TOZASERTIB (VX-680), AND ATITL 3 TYPE I INHIBITOR OF THE TRIAZOLE CARBOTHIOAMIDETITL 4 CLASS.REF J.MED.CHEM. V. 54 2359 2011REFN ISSN 0022-2623PMID 21417343DOI 10.1021/JM101506N Variant […]

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3NYO.A | GRK6

General Structure Information 3nyo GRK6 crystal structure of g protein-coupled receptor kinase 6 in complex with amp 2.92Å AUTH C.A.BOGUTH,P.SINGH,C.C.HUANG,J.J.TESMERTITL MOLECULAR BASIS FOR ACTIVATION OF G PROTEIN-COUPLED RECEPTORTITL 2 KINASES.REF EMBO J. V. 29 3249 2010REFN ISSN 0261-4189PMID 20729810DOI 10.1038/EMBOJ.2010.206 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3IU2.A | NMT1

General Structure Information 3iu2 NMT1 crystal structure of human type-i n-myristoyltransferase with bound myristoyl-coa and inhibitor ddd90096 1.73Å AUTH W.QIU,A.HUTCHINSON,A.WERNIMONT,Y.-H.LIN,A.KANIA,AUTH 2 M.RAVICHANDRAN,I.KOZIERADZKI,D.COSSAR,M.SCHAPIRA,AUTH 3 C.H.ARROWSMITH,C.BOUNTRA,J.WEIGELT,A.M.EDWARDS,P.G.WYATT,AUTH 4 M.A.J.FERGUSON,J.A.FREARSON,S.Y.BRAND,D.A.ROBINSON,AUTH 5 A.BOCHKAREV,R.HUITITL CRYSTAL STRUCTURE OF HUMAN TYPE-I N-MYRISTOYLTRANSFERASETITL 2 WITH BOUND MYRISTOYL-COA AND INHIBITOR DDD90096REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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4MLE.A | GCK

General Structure Information 4mle GCK human glucokinase in complex with novel amino thiazole activator 2.6Å AUTH R.J.HINKLIN,S.A.BOYD,M.J.CHICARELLI,K.R.CONDROSKI,AUTH 2 W.E.DEWOLF,P.A.LEE,W.LEE,A.SINGH,L.THOMAS,W.C.VOEGTLI,AUTH 3 L.WILLIAMS,T.D.AICHERTITL IDENTIFICATION OF A NEW CLASS OF GLUCOKINASE ACTIVATORSTITL 2 THROUGH STRUCTURE-BASED DESIGN.REF J.MED.CHEM. V. 56 7669 2013REFN ISSN 0022-2623PMID 24015910DOI 10.1021/JM401116K Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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3US4.A | MATK

General Structure Information 3us4 MATK crystal structure of a sh2 domain of a megakaryocyte-associated tyrosine kinase (matk) from homo sapiens at 1.50 a resolution 1.5Å AUTH JOINT CENTER FOR STRUCTURAL GENOMICS (JCSG),AUTH 2 PARTNERSHIP FOR T-CELL BIOLOGY (TCELL)TITL CRYSTAL STRUCTURE OF A SH2 DOMAIN OF ATITL 2 MEGAKARYOCYTE-ASSOCIATED TYROSINE KINASE (MATK) FROM HOMOTITL 3 SAPIENS […]

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2V9Y.A | GART

General Structure Information 2v9y GART human aminoimidazole ribonucleotide synthetase 2.1Å AUTH M.WELIN,J.G.GROSSMANN,S.FLODIN,T.NYMAN,P.STENMARK,AUTH 2 L.TRESAUGUES,T.KOTENYOVA,I.JOHANSSON,P.NORDLUND,L.LEHTIOTITL STRUCTURAL STUDIES OF TRI-FUNCTIONAL HUMAN GART.REF NUCLEIC ACIDS RES. V. 38 7308 2010REFN ISSN 0305-1048PMID 20631005DOI 10.1093/NAR/GKQ595 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3GTU.B | GSTM3

General Structure Information 3gtu GSTM3 ligand-free heterodimeric human glutathione s-transferase m2-3 (ec 2.5.1.18), monoclinic crystal form 2.8Å AUTH Y.V.PATSKOVSKY,L.N.PATSKOVSKA,I.LISTOWSKYTITL AN ASPARAGINE-PHENYLALANINE SUBSTITUTION ACCOUNTSTITL 2 FOR CATALYTIC DIFFERENCES BETWEEN HGSTM3-3 ANDTITL 3 OTHER HUMAN CLASS MU GLUTATHIONE S-TRANSFERASES.REF BIOCHEMISTRY V. 38 16187 1999REFN ISSN 0006-2960PMID 10587441DOI 10.1021/BI991714T Variant Set Distributions Mapped Variants

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2IB9.A | ACAT1

General Structure Information 2ib9 ACAT1 crystallographic and kinetic studies of human mitochondrial acetoacetyl-coa thiolase (t2): the importance of potassium and chloride for its structure and function 2.05Å AUTH A.M.HAAPALAINEN,G.MERILAINEN,P.L.PIRILA,N.KONDO,T.FUKAO,AUTH 2 R.K.WIERENGATITL CRYSTALLOGRAPHIC AND KINETIC STUDIES OF HUMAN MITOCHONDRIALTITL 2 ACETOACETYL-COA THIOLASE: THE IMPORTANCE OF POTASSIUM ANDTITL 3 CHLORIDE IONS FOR ITS STRUCTURE AND FUNCTIONREF BIOCHEMISTRY […]

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