3HNG.A | FLT1

General Structure Information 3hng FLT1 crystal structure of vegfr1 in complex with n-(4-chlorophenyl)-2- ((pyridin-4-ylmethyl)amino)benzamide 2.7Å AUTH L.TRESAUGUES,A.ROOS,C.H.ARROWSMITH,H.BERGLUND,C.BOUNTRA,AUTH 2 R.COLLINS,A.M.EDWARDS,S.FLODIN,A.FLORES,S.GRASLUND,AUTH 3 M.HAMMARSTROM,A.JOHANSSON,I.JOHANSSON,T.KARLBERG,AUTH 4 T.KOTENYOVA,M.MOCHE,T.NYMAN,C.PERSSON,T.KRAGH-NIELSEN,AUTH 5 A.KOTZCH,J.SAGEMARK,H.SCHUELER,P.SCHUTZ,M.I.SIPONEN,AUTH 6 L.SVENSSON,A.G.THORSELL,S.VAN DER BERG,J.WEIGELT,M.WELIN,AUTH 7 M.WISNIEWSKA,P.NORDLUNDTITL CRYSTAL STRUCTURE OF VEGFR1 IN COMPLEX WITHTITL 2 N-(4-CHLOROPHENYL)-2-((PYRIDIN-4-YLMETHYL)AMINO)BENZAMIDEREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity […]

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2FN4.A | RRAS

General Structure Information 2fn4 RRAS the crystal structure of human ras-related protein, rras, in the gdp- bound state 1.65Å AUTH A.P.TURNBULL,J.M.ELKINS,C.GILEADI,N.BURGESS,E.SALAH,AUTH 2 E.PAPAGRIGORIOU,J.DEBRECZENI,F.VON DELFT,J.WEIGELT,AUTH 3 A.EDWARDS,C.ARROWSMITH,M.SUNDSTROM,D.DOYLETITL THE CRYSTAL STRUCTURE OF HUMAN RAS-RELATED PROTEIN, RRAS, INTITL 2 THE GDP-BOUND STATEREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2PFR.A | NAT2

General Structure Information 2pfr NAT2 human n-acetyltransferase 2 1.92Å AUTH H.WU,W.TEMPEL,L.DOMBROVSKI,P.LOPPNAU,J.WEIGELT,M.SUNDSTROM,AUTH 2 C.H.ARROWSMITH,A.M.EDWARDS,A.BOCHKAREV,D.M.GRANT,AUTH 3 A.N.PLOTNIKOV,STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL THE CRYSTAL STRUCTURE OF HUMAN N-ACETYLTRANSFERASE 2 INTITL 2 COMPLEX WITH COAREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3TF2.B | EIF4E

General Structure Information 3tf2 EIF4E crystal structure of the cap free human translation initiation factor eif4e 2.1Å AUTH N.SIDDIQUI,W.TEMPEL,L.NEDYALKOVA,L.VOLPON,A.K.WERNIMONT,AUTH 2 M.J.OSBORNE,H.W.PARK,K.L.BORDENTITL STRUCTURAL INSIGHTS INTO THE ALLOSTERIC EFFECTS OF 4EBP1 ONTITL 2 THE EUKARYOTIC TRANSLATION INITIATION FACTOR EIF4E.REF J.MOL.BIOL. V. 415 781 2012REFN ISSN 0022-2836PMID 22178476DOI 10.1016/J.JMB.2011.12.002 Variant Set Distributions Mapped Variants

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3E04.C | FH

General Structure Information 3e04 FH crystal structure of human fumarate hydratase 1.95Å AUTH K.L.KAVANAGH,S.PICAUD,E.S.PILKA,W.W.YUE,A.K.ROOS,AUTH 2 P.FILIPPAKOPOULOS,F.VON DELFT,C.H.ARROWSMITH,M.WIKSTROM,AUTH 3 A.M.EDWARDS,C.BOUNTRA,U.OPPERMANN,AUTH 4 STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL CRYSTAL STRUCTURE OF HUMAN FUMARATE HYDRATASEREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3P1M.C | FDX1

General Structure Information 3p1m FDX1 crystal structure of human ferredoxin-1 (fdx1) in complex with iron- sulfur cluster 2.54Å AUTH A.CHAIKUAD,C.JOHANSSON,T.KROJER,W.W.YUE,C.PHILLIPS,J.E.BRAY,AUTH 2 A.C.W.PIKE,J.R.C.MUNIZ,M.VOLLMAR,J.WEIGELT,C.H.ARROWSMITH,AUTH 3 A.M.EDWARDS,C.BOUNTRA,K.KAVANAGH,U.OPPERMANNTITL CRYSTAL STRUCTURE OF HUMAN FERREDOXIN-1 (FDX1) IN COMPLEXTITL 2 WITH IRON-SULFUR CLUSTERREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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3COS.D | ADH4

General Structure Information 3cos ADH4 crystal structure of human class ii alcohol dehydrogenase (adh4) in complex with nad and zn 2.1Å AUTH K.L.KAVANAGH,N.SHAFQAT,W.YUE,F.VON DELFT,S.BISHOP,A.ROOS,AUTH 2 J.MURRAY,A.M.EDWARDS,C.H.ARROWSMITH,C.BOUNTRA,U.OPPERMANNTITL CRYSTAL STRUCTURE OF HUMAN CLASS II ALCOHOL DEHYDROGENASETITL 2 (ADH4) IN COMPLEX WITH NAD AND ZN.REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

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2IIK.B | ACAA1

General Structure Information 2iik ACAA1 crystal structure of human peroxisomal acetyl-coa acyl transferase 1 (acaa1) 2.55Å AUTH E.PAPAGRIGORIOU,C.JOHANSSON,C.SMEE,K.KAVANAGH,A.C.W.PIKE,AUTH 2 M.SUNDSTROM,J.WEIGELT,A.EDWARDS,C.H.ARROWSMITH,O.GILEADI,AUTH 3 F.GORREC,C.UMEANO,F.VON DELFT,U.OPPERMANN,AUTH 4 STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL CRYSTAL STRUCTURE OF HUMAN PEROXISOMAL ACETYL-COA ACYLTITL 2 TRANSFERASE 1 (ACAA1)REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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4DYL.A | FES

General Structure Information 4dyl FES f-bar domain of human fes tyrosine kinase 2.18Å AUTH E.UGOCHUKWU,E.SALAH,J.ELKINS,A.BARR,T.KROJER,AUTH 2 FILIPPAKOPOULOS P.,J.WEIGELT,C.H.ARROWSMITH,A.EDWARDS,AUTH 3 C.BOUNTRA,F.VON DELFT,S.KNAPP,AUTH 4 STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL F-BAR DOMAIN OF HUMAN FES TYROSINE KINASEREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2F8A.B | GPX1

General Structure Information 2f8a GPX1 crystal structure of the selenocysteine to glycine mutant of human glutathione peroxidase 1 1.5Å AUTH K.L.KAVANAGH,C.JOHANSSON,C.SMEE,O.GILEADI,F.VON DELFT,AUTH 2 U.OPPERMANNTITL CRYSTAL STRUCTURE OF THE SELENOCYSTEINE TO GLYCINE MUTANT OFTITL 2 HUMAN GLUTATHIONE PEROXIDASE 1REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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