3EPZ.B | DNMT1

General Structure Information 3epz DNMT1 structure of the replication foci-targeting sequence of human dna cytosine methyltransferase dnmt1 2.31Å AUTH F.SYEDA,R.L.FAGAN,M.WEAN,G.V.AVVAKUMOV,J.R.WALKER,S.XUE,AUTH 2 S.DHE-PAGANON,C.BRENNERTITL THE REPLICATION FOCUS TARGETING SEQUENCE (RFTS) DOMAIN IS ATITL 2 DNA-COMPETITIVE INHIBITOR OF DNMT1.REF J.BIOL.CHEM. V. 286 15344 2011REFN ISSN 0021-9258PMID 21389349DOI 10.1074/JBC.M110.209882 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

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1R6T.A | WARS

General Structure Information 1r6t WARS crystal structure of human tryptophanyl-trna synthetase 2.1Å AUTH X.-L.YANG,F.J.OTERO,R.J.SKENE,D.E.MCREE,P.SCHIMMEL,AUTH 2 L.RIBAS DE POUPLANATITL CRYSTAL STRUCTURES THAT SUGGEST LATE DEVELOPMENT OF GENETICTITL 2 CODE COMPONENTS FOR DIFFERENTIATING AROMATIC SIDE CHAINSREF PROC.NATL.ACAD.SCI.USA V. 100 15376 2003REFN ISSN 0027-8424PMID 14671330DOI 10.1073/PNAS.2136794100 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity […]

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2M6I.A | GLRA1

General Structure Information 2m6i GLRA1 putative pentameric open-channel structure of full-length transmembrane domains of human glycine receptor alpha1 subunit -1.0Å AUTH D.D.MOWREY,T.CUI,Y.JIA,D.MA,A.M.MAKHOV,P.ZHANG,P.TANG,Y.XUTITL OPEN-CHANNEL STRUCTURES OF THE HUMAN GLYCINE RECEPTOR ALPHATITL 2 1 FULL-LENGTH TRANSMEMBRANE DOMAIN.REF STRUCTURE V. 21 1897 2013REFN ISSN 0969-2126PMID 23994010DOI 10.1016/J.STR.2013.07.014 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic […]

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2IFV.A | CDC25B

General Structure Information 2ifv CDC25B crystal structure of an active site mutant, c473d, of cdc25b phosphatase catalytic domain 1.6Å AUTH J.SOHN,G.BUHRMAN,J.RUDOLPHTITL KINETIC AND STRUCTURAL STUDIES OF SPECIFICTITL 2 PROTEIN-PROTEIN INTERACTIONS IN SUBSTRATETITL 3 CATALYSIS BY CDC25B PHOSPHATASE.REF BIOCHEMISTRY V. 46 807 2007REFN ISSN 0006-2960PMID 17223702DOI 10.1021/BI061257Y Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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1PJ2.A | ME2

General Structure Information 1pj2 ME2 crystal structure of human mitochondrial nad(p)+-dependent malic enzyme in a pentary complex with natural substrate malate, cofactor nadh, mn++, and allosteric activator fumarate 2.3Å AUTH X.TAO,Z.YANG,L.TONGTITL CRYSTAL STRUCTURES OF SUBSTRATE COMPLEXES OF MALICTITL 2 ENZYME AND INSIGHTS INTO THE CATALYTIC MECHANISM.REF STRUCTURE V. 11 1141 2003REFN ISSN 0969-2126PMID 12962632DOI 10.1016/S0969-2126(03)00168-0 […]

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2V60.A | MAOB

General Structure Information 2v60 MAOB structure of human mao b in complex with the selective inhibitor 7-(3-chlorobenzyloxy)-4-carboxaldehyde-coumarin 2.0Å AUTH C.BINDA,J.WANG,L.PISANI,C.CACCIA,A.CAROTTI,AUTH 2 P.SALVATI,D.E.EDMONDSON,A.MATTEVITITL STRUCTURES OF HUMAN MONOAMINE OXIDASE B COMPLEXESTITL 2 WITH SELECTIVE NONCOVALENT INHIBITORS: SAFINAMIDETITL 3 AND COUMARIN ANALOGS.REF J.MED.CHEM. V. 50 5848 2007REFN ISSN 0022-2623PMID 17915852DOI 10.1021/JM070677Y Variant Set Distributions Ripley’s K Analysis Plots […]

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2NLK.A | PTPRG

General Structure Information 2nlk PTPRG crystal structure of d1 and d2 catalytic domains of human protein tyrosine phosphatase gamma (d1+d2 ptprg) 2.4Å AUTH A.J.BARR,E.UGOCHUKWU,W.H.LEE,O.N.KING,P.FILIPPAKOPOULOS,AUTH 2 I.ALFANO,P.SAVITSKY,N.A.BURGESS-BROWN,S.MULLER,S.KNAPPTITL LARGE-SCALE STRUCTURAL ANALYSIS OF THE CLASSICAL HUMANTITL 2 PROTEIN TYROSINE PHOSPHATOME.REF CELL(CAMBRIDGE,MASS.) V. 136 352 2009REFN ISSN 0092-8674PMID 19167335DOI 10.1016/J.CELL.2008.11.038 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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3QAK.A | ADORA2A

General Structure Information 3qak ADORA2A agonist bound structure of the human adenosine a2a receptor 2.71Å AUTH F.XU,H.WU,V.KATRITCH,G.W.HAN,K.A.JACOBSON,Z.G.GAO,AUTH 2 V.CHEREZOV,R.C.STEVENSTITL STRUCTURE OF AN AGONIST-BOUND HUMAN A2A ADENOSINE RECEPTOR.REF SCIENCE V. 332 322 2011REFN ISSN 0036-8075PMID 21393508DOI 10.1126/SCIENCE.1202793 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3SZR.A | MX1

General Structure Information 3szr MX1 crystal structure of modified nucleotide-free human mxa 3.5Å AUTH S.GAO,A.VON DER MALSBURG,A.DICK,K.FAELBER,G.F.SCHRODER,AUTH 2 O.HALLER,G.KOCHS,O.DAUMKETITL STRUCTURE OF MYXOVIRUS RESISTANCE PROTEIN A REVEALS INTRA-TITL 2 AND INTERMOLECULAR DOMAIN INTERACTIONS REQUIRED FOR THETITL 3 ANTIVIRAL FUNCTION.REF IMMUNITY V. 35 514 2011REFN ISSN 1074-7613PMID 21962493DOI 10.1016/J.IMMUNI.2011.07.012 Variant Set Distributions Ripley’s K Analysis Plots Variant […]

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1RY7.B | FGFR3

General Structure Information 1ry7 FGFR3 crystal structure of the 3 ig form of fgfr3c in complex with fgf1 3.2Å AUTH S.K.OLSEN,O.A.IBRAHIMI,A.RAUCCI,F.ZHANG,AUTH 2 A.V.ELISEENKOVA,A.YAYON,C.BASILICO,R.J.LINHARDT,AUTH 3 J.SCHLESSINGER,M.MOHAMMADITITL INSIGHTS INTO THE MOLECULAR BASIS FOR FIBROBLASTTITL 2 GROWTH FACTOR RECEPTOR AUTOINHIBITION ANDTITL 3 LIGAND-BINDING PROMISCUITY.REF PROC.NATL.ACAD.SCI.USA V. 101 935 2004REFN ISSN 0027-8424PMID 14732692DOI 10.1073/PNAS.0307287101 Variant Set Distributions Ripley’s K […]

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