4JZ1.A | ST14

General Structure Information 4jz1 ST14 crystal structure of matriptase in complex with inhibitor 1.9Å AUTH R.GOSWAMI,S.MUKHERJEE,G.WOHLFAHRT,C.GHADIYARAM,J.NAGARAJ,AUTH 2 B.R.CHANDRA,R.K.SISTLA,L.K.SATYAM,D.S.SAMIULLA,A.MOILANEN,AUTH 3 H.S.SUBRAMANYA,M.RAMACHANDRATITL DISCOVERY OF PYRIDYL BIS(OXY)DIBENZIMIDAMIDE DERIVATIVES ASTITL 2 SELECTIVE MATRIPTASE INHIBITORSREF ACS MED.CHEM.LETT. V. 4 1152 2013REFN ISSN 1948-5875PMID 24900621DOI 10.1021/ML400213V Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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4DL3.A | POLH

General Structure Information 4dl3 POLH human dna polymerase eta inserting dcmpnpp opposite gg template (gg0b). 2.1Å AUTH Y.ZHAO,C.BIERTUMPFEL,M.T.GREGORY,Y.J.HUA,F.HANAOKA,W.YANGTITL STRUCTURAL BASIS FOR CHEMORESISTANCE TO CISPLATIN MEDIATEDTITL 2 BY DNA POLYMERASE ETAREF PROC.NATL.ACAD.SCI.USA V. 109 7269 2012REFN ISSN 0027-8424PMID 22529383DOI 10.1073/PNAS.1202681109 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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2PID.A | YARS2

General Structure Information 2pid YARS2 crystal structure of human mitochondrial tyrosyl-trna synthetase in complex with an adenylate analog 2.2Å AUTH L.BONNEFOND,M.FRUGIER,E.TOUZE,B.LORBER,C.FLORENTZ,R.GIEGE,AUTH 2 C.SAUTER,J.RUDINGER-THIRIONTITL CRYSTAL STRUCTURE OF HUMAN MITOCHONDRIAL TYROSYL-TRNATITL 2 SYNTHETASE REVEALS COMMON AND IDIOSYNCRATIC FEATURES.REF STRUCTURE V. 15 1505 2007REFN ISSN 0969-2126PMID 17997975DOI 10.1016/J.STR.2007.09.018 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

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4L7R.A | PARP3

General Structure Information 4l7r PARP3 human artd3 (parp3) – catalytic domain in complex with inhibitor me0400 2.2Å AUTH A.E.LINDGREN,T.KARLBERG,T.EKBLAD,S.SPJUT,A.G.THORSELL,AUTH 2 C.D.ANDERSSON,T.T.NHAN,V.HELLSTEN,J.WEIGELT,A.LINUSSON,AUTH 3 H.SCHULER,M.ELOFSSONTITL CHEMICAL PROBES TO STUDY ADP-RIBOSYLATION: SYNTHESIS ANDTITL 2 BIOCHEMICAL EVALUATION OF INHIBITORS OF THE HUMANTITL 3 ADP-RIBOSYLTRANSFERASE ARTD3/PARP3.REF J.MED.CHEM. V. 56 9556 2013REFN ISSN 0022-2623PMID 24188023DOI 10.1021/JM401394U Variant Set Distributions Ripley’s K […]

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1V27.A | RIMS2

General Structure Information 1v27 RIMS2 solution structure of the first c2 domain of rim2 -1.0Å AUTH T.NAGASHIMA,F.HAYASHI,S.YOKOYAMATITL SOLUTION STRUCTURE OF THE FIRST C2 DOMAIN OF RIM2REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3RPN.E | GSTK1

General Structure Information 3rpn GSTK1 crystal structure of human kappa class glutathione transferase in complex with s-hexylglutathione 1.9Å AUTH B.WANG,Y.PENG,T.ZHANG,J.DINGTITL CRYSTAL STRUCTURES AND KINETIC STUDIES OF HUMAN KAPPA CLASSTITL 2 GLUTATHIONE TRANSFERASE PROVIDE INSIGHTS INTO THE CATALYTICTITL 3 MECHANISM.REF BIOCHEM.J. V. 439 215 2011REFN ISSN 0264-6021PMID 21728995DOI 10.1042/BJ20110753 Variant Set Distributions Ripley’s K Analysis Plots […]

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2EKF.A | AUP1

General Structure Information 2ekf AUP1 solution structure of ruh-075, a human cue domain -1.0Å AUTH A.Z.M.RUHUL MOMEN,H.HIROTA,F.HAYASHI,S.YOKOYAMATITL SOLUTION STRUCTURE OF RUH-075, A HUMAN CUE DOMAINREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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4NH3.A | DICER1

General Structure Information 4nh3 DICER1 structure of human dicer platform-paz-connector helix cassette in complex with 13-mer sirna having 5-pu and uu-3 ends (2.6 angstrom resolution) 2.62Å AUTH Y.TIAN,D.K.SIMANSHU,J.B.MA,J.E.PARK,I.HEO,V.N.KIM,D.J.PATELTITL A PHOSPHATE-BINDING POCKET WITHIN THE PLATFORM-PAZ-CONNECTORTITL 2 HELIX CASSETTE OF HUMAN DICER.REF MOL.CELL V. 53 606 2014REFN ISSN 1097-2765PMID 24486018DOI 10.1016/J.MOLCEL.2014.01.003 Variant Set Distributions Ripley’s K Analysis […]

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3ENP.B | TPRKB

General Structure Information 3enp TPRKB crystal structure of human cgi121 2.48Å AUTH D.Y.MAO,D.NECULAI,M.DOWNEY,S.ORLICKY,Y.Z.HAFFANI,AUTH 2 D.F.CECCARELLI,J.S.HO,R.K.SZILARD,W.ZHANG,C.S.HO,L.WAN,AUTH 3 C.FARES,S.RUMPEL,I.KURINOV,C.H.ARROWSMITH,D.DUROCHER,AUTH 4 F.SICHERITITL ATOMIC STRUCTURE OF THE KEOPS COMPLEX: AN ANCIENT PROTEINTITL 2 KINASE-CONTAINING MOLECULAR MACHINE.REF MOL.CELL V. 32 259 2008REFN ISSN 1097-2765PMID 18951093DOI 10.1016/J.MOLCEL.2008.10.002 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped […]

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1LB6.A | TRAF6

General Structure Information 1lb6 TRAF6 traf6-cd40 complex 1.8Å AUTH H.YE,J.R.ARRON,B.LAMOTHE,M.CIRILLI,T.KOBAYASHI,AUTH 2 N.K.SHEVDE,D.SEGAL,O.K.DZIVENU,M.VOLOGODSKAIA,AUTH 3 M.YIM,K.DU,S.SINGH,J.W.PIKE,B.G.DARNAY,Y.CHOI,H.WUTITL DISTINCT MOLECULAR MECHANISM FOR INITIATING TRAF6TITL 2 SIGNALLING.REF NATURE V. 418 443 2002REFN ISSN 0028-0836PMID 12140561DOI 10.1038/NATURE00888 Variant Set Distributions Mapped Variants

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