1JIQ.B | GPI

General Structure Information 1jiq GPI crystal structure of human autocrine motility factor 1.9Å AUTH N.TANAKA,A.HAGA,H.UEMURA,H.AKIYAMA,T.FUNASAKA,AUTH 2 H.NAGASE,A.RAZ,K.T.NAKAMURATITL INHIBITION MECHANISM OF CYTOKINE ACTIVITY OF HUMANTITL 2 AUTOCRINE MOTILITY FACTOR EXAMINED BY CRYSTALTITL 3 STRUCTURE ANALYSES AND SITE-DIRECTED MUTAGENESISTITL 4 STUDIES.REF J.MOL.BIOL. V. 318 985 2002REFN ISSN 0022-2836PMID 12054796DOI 10.1016/S0022-2836(02)00186-9 Variant Set Distributions Ripley’s K Analysis Plots […]

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2X2M.B | RET

General Structure Information 2x2m RET crystal structure of phosphorylated ret tyrosine kinase domain with inhibitor 2.5Å AUTH L.MOLOGNI,R.ROSTAGNO,S.BRUSSOLO,P.P.KNOWLES,AUTH 2 S.KJAER,J.MURRAY-RUST,E.ROSSO,A.ZAMBON,L.SCAPOZZA,AUTH 3 N.Q.MCDONALD,V.LUCCHINI,C.GAMBACORTI-PASSERINITITL SYNTHESIS, STRUCTURE-ACTIVITY RELATIONSHIP ANDTITL 2 CRYSTALLOGRAPHIC STUDIES OF 3-SUBSTITUTED INDOLIN-TITL 3 2-ONE RET INHIBITORS.REF BIOORG.MED.CHEM. V. 18 1482 2010REFN ISSN 0968-0896PMID 20117004DOI 10.1016/J.BMC.2010.01.011 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

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1BHG.A | GUSB

General Structure Information 1bhg GUSB human beta-glucuronidase at 2.6 a resolution 2.53Å AUTH S.JAIN,W.B.DRENDEL,Z.W.CHEN,F.S.MATHEWS,W.S.SLY,J.H.GRUBBTITL STRUCTURE OF HUMAN BETA-GLUCURONIDASE REVEALS CANDIDATETITL 2 LYSOSOMAL TARGETING AND ACTIVE-SITE MOTIFS.REF NAT.STRUCT.BIOL. V. 3 375 1996REFN ISSN 1072-8368PMID 8599764DOI 10.1038/NSB0496-375 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1EGD.A | ACADM

General Structure Information 1egd ACADM structure of t255e, e376g mutant of human medium chain acyl- coa dehydrogenase 2.4Å AUTH H.J.LEE,M.WANG,R.PASCHKE,A.NANDY,S.GHISLA,J.J.KIMTITL CRYSTAL STRUCTURES OF THE WILD TYPE AND THETITL 2 GLU376GLY/THR255GLU MUTANT OF HUMAN MEDIUM-CHAINTITL 3 ACYL-COA DEHYDROGENASE: INFLUENCE OF THE LOCATIONTITL 4 OF THE CATALYTIC BASE ON SUBSTRATE SPECIFICITY.REF BIOCHEMISTRY V. 35 12412 1996REFN ISSN […]

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1KF9.C | GHR

General Structure Information 1kf9 GHR phage display derived variant of human growth hormone complexed with two copies of the extracellular domain of its receptor 2.6Å AUTH C.A.SCHIFFER,M.ULTSCH,S.WALSH,W.SOMERS,A.M.DE VOS,AUTH 2 A.A.KOSSIAKOFFTITL STRUCTURE OF A PHAGE DISPLAY DERIVED VARIANT OFTITL 2 HUMAN GROWTH HORMONE COMPLEXED TO TWO COPIES OFTITL 3 THE EXTRACELLULAR DOMAIN OF ITS RECEPTOR: EVIDENCETITL […]

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1TRN.A | PRSS1

General Structure Information 1trn PRSS1 crystal structure of human trypsin 1: unexpected phosphorylation of tyrosine 151 2.2Å AUTH C.GABORIAUD,L.SERRE,O.GUY-CROTTE,E.FOREST,AUTH 2 J.C.FONTECILLA-CAMPSTITL CRYSTAL STRUCTURE OF HUMAN TRYPSIN 1: UNEXPECTEDTITL 2 PHOSPHORYLATION OF TYR151.REF J.MOL.BIOL. V. 259 995 1996REFN ISSN 0022-2836PMID 8683601DOI 10.1006/JMBI.1996.0376 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped […]

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1QKI.D | G6PD

General Structure Information 1qki G6PD x-ray structure of human glucose 6-phosphate dehydrogenase (variant canton r459l) complexed with structural nadp+ 3.0Å AUTH S.W.N.AU,S.GOVER,V.M.S.LAM,M.J.ADAMSTITL HUMAN GLUCOSE-6-PHOSPHATE DEHYDROGENASE: THETITL 2 CRYSTAL STRUCTURE REVEALS A STRUCTURAL NADP+TITL 3 MOLECULE AND PROVIDES INSIGHTS INTO ENZYMETITL 4 DEFICIENCYREF STRUCTURE V. 8 293 2000REFN ISSN 0969-2126PMID 10745013DOI 10.1016/S0969-2126(00)00104-0 Variant Set Distributions Ripley’s […]

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1B0F.A | ELANE

General Structure Information 1b0f ELANE crystal structure of human neutrophil elastase with mdl 101, 146 3.0Å AUTH R.J.CREGGE,S.L.DURHAM,R.A.FARR,S.L.GALLION,C.M.HARE,AUTH 2 R.V.HOFFMAN,M.J.JANUSZ,H.O.KIM,J.R.KOEHL,S.MEHDI,W.A.METZ,AUTH 3 N.P.PEET,J.T.PELTON,H.A.SCHREUDER,S.SUNDER,C.TARDIFTITL INHIBITION OF HUMAN NEUTROPHIL ELASTASE. 4. DESIGN,TITL 2 SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, ANDTITL 3 STRUCTURE-ACTIVITY RELATIONSHIPS FOR A SERIES OFTITL 4 P2-MODIFIED, ORALLY ACTIVE PEPTIDYL PENTAFLUOROETHYLTITL 5 KETONES.REF J.MED.CHEM. V. 41 2461 1998REFN […]

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1NR1.C | GLUD1

General Structure Information 1nr1 GLUD1 crystal structure of the r463a mutant of human glutamate dehydrogenase 3.3Å AUTH S.BANERJEE,T.SCHMIDT,J.FANG,C.A.STANLEY,T.J.SMITHTITL STRUCTURAL STUDIES ON ADP ACTIVATION OF MAMMALIANTITL 2 GLUTAMATE DEHYDROGENASE AND THE EVOLUTION OFTITL 3 REGULATIONREF BIOCHEMISTRY V. 42 3446 2003REFN ISSN 0006-2960PMID 12653548DOI 10.1021/BI0206917 Variant Set Distributions Pathogenic Proximity Analysis Mapped Variants

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1UMK.A | CYB5R3

General Structure Information 1umk CYB5R3 the structure of human erythrocyte nadh-cytochrome b5 reductase 1.75Å AUTH S.BANDO,T.TAKANO,T.YUBISUI,K.SHIRABE,M.TAKESHITA,AUTH 2 A.NAKAGAWATITL STRUCTURE OF HUMAN ERYTHROCYTE NADH-CYTOCHROME B5TITL 2 REDUCTASE.REF ACTA CRYSTALLOGR.,SECT.D V. 60 1929 2004REFN ISSN 0907-4449PMID 15502298DOI 10.1107/S0907444904020645 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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