3BI6.A | WEE1

General Structure Information 3bi6 WEE1 wee1 kinase complex with inhibitor pd352396 2.2Å AUTH J.B.SMAILL,H.H.LEE,B.D.PALMER,A.M.THOMPSON,AUTH 2 C.J.SQUIRE,E.N.BAKER,R.J.BOOTH,A.KRAKER,K.HOOK,AUTH 3 W.A.DENNYTITL SYNTHESIS AND STRUCTURE-ACTIVITY RELATIONSHIPS OFTITL 2 SOLUBLE 8-SUBSTITUTEDTITL 3 4-(2-CHLOROPHENYL)-9-HYDROXYPYRROLO[3,4-TITL 4 C]CARBAZOLE-1,3(2H,6H)-DIONES AS INHIBITORS OF THETITL 5 WEE1 AND CHK1 CHECKPOINT KINASES.REF BIOORG.MED.CHEM.LETT. V. 18 929 2008REFN ISSN 0960-894XPMID 18191399DOI 10.1016/J.BMCL.2007.12.046 Variant Set Distributions Ripley’s K Analysis […]

See Details
1J55.A | S100P

General Structure Information 1j55 S100P the crystal structure of ca+-bound human s100p determined at 2.0a resolution by x-ray 2.0Å AUTH H.ZHANG,G.WANG,Y.DING,Z.WANG,R.BARRACLOUGH,P.S.RUDLAND,AUTH 2 D.G.FERNIG,Z.RAOTITL THE CRYSTAL STRUCTURE AT 2A RESOLUTION OF THE CA2+-BINDINGTITL 2 PROTEIN S100PREF J.MOL.BIOL. V. 325 785 2003REFN ISSN 0022-2836PMID 12507480DOI 10.1016/S0022-2836(02)01278-0 Variant Set Distributions Mapped Variants

See Details
3DPE.A | MMP8

General Structure Information 3dpe MMP8 crystal structure of the complex between mmp-8 and a non- zinc chelating inhibitor 1.6Å AUTH G.POCHETTI,R.MONTANARI,C.GEGE,C.CHEVRIER,AUTH 2 A.G.TAVERAS,F.MAZZATITL EXTRA BINDING REGION INDUCED BY NON-ZINC CHELATINGTITL 2 INHIBITORS INTO THE S(1) SUBSITE OF MATRIXTITL 3 METALLOPROTEINASE 8 (MMP-8)REF J.MED.CHEM. V. 52 1040 2009REFN ISSN 0022-2623PMID 19173605DOI 10.1021/JM801166J Variant Set Distributions Ripley’s […]

See Details
4HWT.B | TARS

General Structure Information 4hwt TARS crystal structure of human threonyl-trna synthetase bound to a novel inhibitor 2.3Å AUTH M.TENG,M.T.HILGERS,M.L.CUNNINGHAM,A.BORCHARDT,J.B.LOCKE,AUTH 2 S.ABRAHAM,G.HALEY,B.P.KWAN,C.HALL,G.W.HOUGH,K.J.SHAW,J.FINNTITL IDENTIFICATION OF BACTERIA-SELECTIVE THREONYL-TRNATITL 2 SYNTHETASE SUBSTRATE INHIBITORS BY STRUCTURE-BASED DESIGN.REF J.MED.CHEM. V. 56 1748 2013REFN ISSN 0022-2623PMID 23362938DOI 10.1021/JM301756M Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

See Details
1F4R.A | MPG

General Structure Information 1f4r MPG crystal structure of the human aag dna repair glycosylase complexed with 1,n6-ethenoadenine-dna 2.4Å AUTH A.Y.LAU,M.D.WYATT,B.J.GLASSNER,L.D.SAMSON,AUTH 2 T.ELLENBERGERTITL MOLECULAR BASIS FOR DISCRIMINATING BETWEEN NORMALTITL 2 AND DAMAGED BASES BY THE HUMAN ALKYLADENINETITL 3 GLYCOSYLASE, AAG.REF PROC.NATL.ACAD.SCI.USA V. 97 13573 2000REFN ISSN 0027-8424PMID 11106395DOI 10.1073/PNAS.97.25.13573 Variant Set Distributions Ripley’s K Analysis Plots […]

See Details
1K1A.A | BCL3

General Structure Information 1k1a BCL3 crystal structure of the ankyrin repeat domain of bcl-3: a unique member of the ikappab protein family 1.86Å AUTH F.MICHEL,M.SOLER-LOPEZ,C.PETOSA,P.CRAMER,AUTH 2 U.SIEBENLIST,C.W.MULLERTITL CRYSTAL STRUCTURE OF THE ANKYRIN REPEAT DOMAIN OFTITL 2 BCL-3: A UNIQUE MEMBER OF THE IKAPPAB PROTEINTITL 3 FAMILY.REF EMBO J. V. 20 6180 2001REFN ISSN 0261-4189PMID 11707390DOI […]

See Details
4GJ3.A | TYK2

General Structure Information 4gj3 TYK2 tyk2 (jh1) in complex with 2,6-dichloro-4-cyano-n-[2-({[(1r,2r)-2- fluorocyclopropyl]carbonyl}amino)pyridin-4-yl]benzamide 2.5Å AUTH J.LIANG,A.VAN ABBEMA,M.BALAZS,K.BARRETT,L.BEREZHKOVSKY,AUTH 2 W.BLAIR,C.CHANG,D.DELAROSA,J.DEVOSS,J.DRISCOLL,C.EIGENBROT,AUTH 3 N.GHILARDI,P.GIBBONS,J.HALLADAY,A.JOHNSON,P.B.KOHLI,Y.LAI,AUTH 4 Y.LIU,J.LYSSIKATOS,P.MANTIK,K.MENGHRAJANI,J.MURRAY,I.PENG,AUTH 5 A.SAMBRONE,S.SHIA,Y.SHIN,J.SMITH,S.SOHN,V.TSUI,M.ULTSCH,AUTH 6 L.C.WU,Y.XIAO,W.YANG,J.YOUNG,B.ZHANG,B.Y.ZHU,S.MAGNUSONTITL LEAD OPTIMIZATION OF A 4-AMINOPYRIDINE BENZAMIDE SCAFFOLD TOTITL 2 IDENTIFY POTENT, SELECTIVE, AND ORALLY BIOAVAILABLE TYK2TITL 3 INHIBITORS.REF J.MED.CHEM. V. 56 4521 2013REFN ISSN 0022-2623PMID 23668484DOI 10.1021/JM400266T Variant Set […]

See Details
1WER.A | RASA1

General Structure Information 1wer RASA1 ras-gtpase-activating domain of human p120gap 1.6Å AUTH K.SCHEFFZEK,A.LAUTWEIN,W.KABSCH,M.R.AHMADIAN,AUTH 2 A.WITTINGHOFERTITL CRYSTAL STRUCTURE OF THE GTPASE-ACTIVATING DOMAINTITL 2 OF HUMAN P120GAP AND IMPLICATIONS FOR THETITL 3 INTERACTION WITH RAS.REF NATURE V. 384 591 1996REFN ISSN 0028-0836PMID 8955277DOI 10.1038/384591A0 Variant Set Distributions Mapped Variants

See Details
3ICI.B | PPIB

General Structure Information 3ici PPIB crystal structure of cyclophilin b in complex with calmegin fragment 1.7Å AUTH G.KOZLOV,S.BASTOS-ARISTIZABAL,P.MAATTANEN,A.ROSENAUER,AUTH 2 F.ZHENG,A.KILLIKELLY,J.F.TREMPE,D.Y.THOMAS,K.GEHRINGTITL STRUCTURAL BASIS OF CYCLOPHILIN B BINDING BY THETITL 2 CALNEXIN/CALRETICULIN P-DOMAIN.REF J.BIOL.CHEM. V. 285 35551 2010REFN ISSN 0021-9258PMID 20801878DOI 10.1074/JBC.M110.160101 Variant Set Distributions Mapped Variants

See Details
2MAM.A | ARID4A

General Structure Information 2mam ARID4A solution structure of the interdigitated double tudor domain of rbbp1 -1.0Å AUTH W.GONG,J.WANG,S.PERRETT,Y.FENGTITL RETINOBLASTOMA-BINDING PROTEIN 1 HAS AN INTERDIGITATEDTITL 2 DOUBLE TUDOR DOMAIN WITH DNA-BINDING ACTIVITY.REF J.BIOL.CHEM. 2013REFN ESSN 1083-351XPMID 24379399DOI 10.1074/JBC.M113.501940 Variant Set Distributions Mapped Variants

See Details