2XAH.B | RCOR1

General Structure Information 2xah RCOR1 crystal structure of lsd1-corest in complex with (+)- trans-2-phenylcyclopropyl-1-amine 3.1Å AUTH C.BINDA,S.VALENTE,M.ROMANENGHI,S.PILOTTO,R.CIRILLI,AUTH 2 A.KARYTINOS,G.CIOSSANI,O.A.BOTRUGNO,F.FORNERIS,AUTH 3 M.TARDUGNO,D.E.EDMONDSON,S.MINUCCI,A.MATTEVI,A.MAITITL BIOCHEMICAL, STRUCTURAL, AND BIOLOGICAL EVALUATIONTITL 2 OF TRANYLCYPROMINE DERIVATIVES AS INHIBITORS OFTITL 3 HISTONE DEMETHYLASES LSD1 AND LSD2.REF J.AM.CHEM.SOC. V. 132 6827 2010REFN ISSN 0002-7863PMID 20415477DOI 10.1021/JA101557K Variant Set Distributions Mapped Variants

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4IR4.A | BAZ2B

General Structure Information 4ir4 BAZ2B crystal structure of the bromodomain of human baz2b in complex with 1- [7-(morpholin-4-yl)-1-(pyridin-2-yl)indolizin-3-yl]ethanone (gsk2834113a) 2.05Å AUTH P.CHEN,A.CHAIKUAD,P.BAMBOROUGH,M.BANTSCHEFF,C.BOUNTRA,AUTH 2 C.W.CHUNG,O.FEDOROV,P.GRANDI,D.JUNG,R.LESNIAK,M.LINDON,AUTH 3 S.MULLER,M.PHILPOTT,R.PRINJHA,C.ROGERS,C.SELENSKI,C.TALLANT,AUTH 4 T.WERNER,T.M.WILLSON,S.KNAPP,D.H.DREWRYTITL DISCOVERY AND CHARACTERIZATION OF GSK2801, A SELECTIVETITL 2 CHEMICAL PROBE FOR THE BROMODOMAINS BAZ2A AND BAZ2B.REF J.MED.CHEM. 2015REFN ISSN 0022-2623PMID 25799074DOI 10.1021/ACS.JMEDCHEM.5B00209 Variant Set Distributions Mapped Variants

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2ECB.A | ZHX1

General Structure Information 2ecb ZHX1 the solution structure of the third homeobox domain of human zinc fingers and homeoboxes protein -1.0Å AUTH S.OHNISHI,N.TOCHIO,A.SASAGAWA,K.SAITO,S.KOSHIBA,AUTH 2 M.INOUE,T.KIGAWA,S.YOKOYAMATITL THE SOLUTION STRUCTURE OF THE THIRD HOMEOBOXTITL 2 DOMAIN OF HUMAN ZINC FINGERS AND HOMEOBOXES PROTEINREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic […]

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3RSN.A | ASH2L

General Structure Information 3rsn ASH2L crystal structure of the n-terminal region of human ash2l 2.1Å AUTH Y.CHEN,B.WAN,K.C.WANG,F.CAO,Y.YANG,A.PROTACIO,Y.DOU,AUTH 2 H.Y.CHANG,M.LEITITL CRYSTAL STRUCTURE OF THE N-TERMINAL REGION OF HUMAN ASH2LTITL 2 SHOWS A WINGED-HELIX MOTIF INVOLVED IN DNA BINDING.REF EMBO REP. V. 12 797 2011REFN ISSN 1469-221XPMID 21660059DOI 10.1038/EMBOR.2011.101 Variant Set Distributions Mapped Variants

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4GMJ.D | CNOT7

General Structure Information 4gmj CNOT7 structure of human not1 mif4g domain co-crystallized with caf1 2.7Å AUTH A.P.PETIT,L.WOHLBOLD,P.BAWANKAR,E.HUNTZINGER,S.SCHMIDT,AUTH 2 E.IZAURRALDE,O.WEICHENRIEDERTITL THE STRUCTURAL BASIS FOR THE INTERACTION BETWEEN THE CAF1TITL 2 NUCLEASE AND THE NOT1 SCAFFOLD OF THE HUMAN CCR4-NOTTITL 3 DEADENYLASE COMPLEXREF NUCLEIC ACIDS RES. V. 40 11058 2012REFN ISSN 0305-1048PMID 22977175DOI 10.1093/NAR/GKS883 Variant Set Distributions […]

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2CQE.A | ZC3H4

General Structure Information 2cqe ZC3H4 solution structure of the zinc-finger domain in kiaa1064 protein -1.0Å AUTH T.SOMEYA,Y.MUTO,M.INOUE,T.KIGAWA,T.TERADA,AUTH 2 M.SHIROUZU,S.YOKOYAMATITL SOLUTION STRUCTURE OF THE ZINC-FINGER DOMAIN INTITL 2 KIAA1064 PROTEINREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2EM6.A | ZNF224

General Structure Information 2em6 ZNF224 solution structure of the c2h2 type zinc finger (region 199- 231) of human zinc finger protein 224 -1.0Å AUTH N.TOCHIO,T.TOMIZAWA,H.ABE,K.SAITO,H.LI,M.SATO,AUTH 2 S.KOSHIBA,N.KOBAYASHI,T.KIGAWA,S.YOKOYAMATITL SOLUTION STRUCTURE OF THE C2H2 TYPE ZINC FINGERTITL 2 (REGION 199-231) OF HUMAN ZINC FINGER PROTEIN 224REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2DZR.A | GTF2IRD1

General Structure Information 2dzr GTF2IRD1 solution structure of rsgi ruh-067, a gtf2i domain in human cdna -1.0Å AUTH Y.DOI-KATAYAMA,H.HIROTA,Y.MUTO,S.YOKOYAMATITL SOLUTION STRUCTURE OF RSGI RUH-067, A GTF2I DOMAINTITL 2 IN HUMAN CDNAREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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3TOJ.B | ASH2L

General Structure Information 3toj ASH2L structure of the spry domain of human ash2l 2.07Å AUTH Y.CHEN,F.CAO,B.WAN,Y.DOU,M.LEITITL STRUCTURE OF THE SPRY DOMAIN OF HUMAN ASH2L AND ITSTITL 2 INTERACTIONS WITH RBBP5 AND DPY30.REF CELL RES. V. 22 598 2012REFN ISSN 1001-0602PMID 22231628DOI 10.1038/CR.2012.9 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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4BLD.B | SUFU

General Structure Information 4bld SUFU crystal structure of a human suppressor of fused (sufu)- gli3p complex 2.8Å AUTH A.L.CHERRY,C.FINTA,M.KARLSTROM,Q.JIN,T.SCHWEND,AUTH 2 J.ASTORGA-WELLS,R.A.ZUBAREV,M.DEL CAMPO,A.R.CRISWELL,AUTH 3 D.DE SANCTIS,L.JOVINE,R.TOFTGARDTITL STRUCTURAL BASIS OF SUFU-GLI INTERACTION IN HEDGEHOGTITL 2 SIGNALLING REGULATIONREF ACTA CRYSTALLOGR.,SECT.D V. 69 2579 2013REFN ISSN 0907-4449PMID 24311597DOI 10.1107/S0907444913028473 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

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