2NO3.A | MAPK8

General Structure Information 2no3 MAPK8 novel 4-anilinopyrimidines as potent jnk1 inhibitors 3.2Å AUTH M.LIU,S.WANG,J.E.CLAMPIT,R.J.GUM,D.L.HAASCH,AUTH 2 C.M.RONDINONE,J.M.TREVILLYAN,C.ABAD-ZAPATERO,AUTH 3 E.H.FRY,H.L.SHAM,G.LIUTITL DISCOVERY OF A NEW CLASS OF 4-ANILINOPYRIMIDINESTITL 2 AS POTENT C-JUN N-TERMINAL KINASE INHIBITORS:TITL 3 SYNTHESIS AND SAR STUDIES.REF BIOORG.MED.CHEM.LETT. V. 17 668 2007REFN ISSN 0960-894XPMID 17107797DOI 10.1016/J.BMCL.2006.10.093 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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4EKC.D | RGS2

General Structure Information 4ekc RGS2 structure of human regulator of g protein signaling 2 (rgs2) in complex with murine galpha-q(r183c) 7.4Å AUTH M.R.NANCE,B.KREUTZ,V.M.TESMER,R.STERNE-MARR,T.KOZASA,AUTH 2 J.J.TESMERTITL STRUCTURAL AND FUNCTIONAL ANALYSIS OF THE REGULATOR OF GTITL 2 PROTEIN SIGNALING 2-G ALPHA Q COMPLEX.REF STRUCTURE V. 21 438 2013REFN ISSN 0969-2126PMID 23434405DOI 10.1016/J.STR.2012.12.016 Variant Set Distributions Mapped Variants

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2OZO.A | ZAP70

General Structure Information 2ozo ZAP70 autoinhibited intact human zap-70 2.6Å AUTH S.DEINDL,T.A.KADLECEK,T.BRDICKA,X.CAO,A.WEISS,AUTH 2 J.KURIYANTITL STRUCTURAL BASIS FOR THE INHIBITION OF TYROSINETITL 2 KINASE ACTIVITY OF ZAP-70.REF CELL(CAMBRIDGE,MASS.) V. 129 735 2007REFN ISSN 0092-8674PMID 17512407DOI 10.1016/J.CELL.2007.03.039 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1IMV.A | SERPINF1

General Structure Information 1imv SERPINF1 2.85 a crystal structure of pedf 2.85Å AUTH M.SIMONOVIC,P.G.GETTINS,K.VOLZTITL CRYSTAL STRUCTURE OF HUMAN PEDF, A POTENT ANTI-ANGIOGENICTITL 2 AND NEURITE GROWTH-PROMOTING FACTOR.REF PROC.NATL.ACAD.SCI.USA V. 98 11131 2001REFN ISSN 0027-8424PMID 11562499DOI 10.1073/PNAS.211268598 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1NWT.A | CHI3L1

General Structure Information 1nwt CHI3L1 crystal structure of human cartilage gp39 (hc-gp39) in complex with chitopentaose 2.5Å AUTH F.FUSETTI,T.PIJNING,K.H.KALK,E.BOS,B.W.DIJKSTRATITL CRYSTAL STRUCTURE AND CARBOHYDRATE-BINDING PROPERTIES OF THETITL 2 HUMAN CARTILAGE GLYCOPROTEIN-39REF J.BIOL.CHEM. V. 278 37753 2003REFN ISSN 0021-9258PMID 12851408DOI 10.1074/JBC.M303137200 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2C5D.C | AXL

General Structure Information 2c5d AXL structure of a minimal gas6-axl complex 3.3Å AUTH T.SASAKI,P.G.KNYAZEV,N.J.CLOUT,Y.CHEBURKIN,AUTH 2 W.GOEHRING,A.ULLRICH,R.TIMPL,E.HOHENESTERTITL STRUCTURAL BASIS FOR GAS6-AXL SIGNALLING.REF EMBO J. V. 25 80 2006REFN ISSN 0261-4189PMID 16362042DOI 10.1038/SJ.EMBOJ.7600912 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1X6G.A | MATK

General Structure Information 1x6g MATK solution structures of the sh3 domain of human megakaryocyte-associated tyrosine-protein kinase. -1.0Å AUTH M.SATO,S.KOSHIBA,M.INOUE,T.KIGAWA,S.YOKOYAMATITL SOLUTION STRUCTURES OF THE SH3 DOMAIN OF HUMANTITL 2 MEGAKARYOCYTE-ASSOCIATED TYROSINE-PROTEIN KINASE.REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2JOD.A | ADCYAP1R1

General Structure Information 2jod ADCYAP1R1 pac1-rshort n-terminal ec domain pacap(6-38) complex -1.0Å AUTH C.SUN,D.SONG,R.A.DAVIS-TABER,L.W.BARRETT,V.E.SCOTT,AUTH 2 P.L.RICHARDSON,A.PEREDA-LOPEZ,M.E.UCHIC,AUTH 3 L.R.SOLOMON,M.R.LAKE,K.A.WALTER,P.J.HAJDUK,AUTH 4 E.T.OLEJNICZAKTITL SOLUTION STRUCTURE AND MUTATIONAL ANALYSIS OFTITL 2 PITUITARY ADENYLATE CYCLASE-ACTIVATING POLYPEPTIDETITL 3 BINDING TO THE EXTRACELLULAR DOMAIN OF PAC1-RS.REF PROC.NATL.ACAD.SCI.USA V. 104 7875 2007REFN ISSN 0027-8424PMID 17470806DOI 10.1073/PNAS.0611397104 Variant Set Distributions Mapped Variants

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3US4.A | MATK

General Structure Information 3us4 MATK crystal structure of a sh2 domain of a megakaryocyte-associated tyrosine kinase (matk) from homo sapiens at 1.50 a resolution 1.5Å AUTH JOINT CENTER FOR STRUCTURAL GENOMICS (JCSG),AUTH 2 PARTNERSHIP FOR T-CELL BIOLOGY (TCELL)TITL CRYSTAL STRUCTURE OF A SH2 DOMAIN OF ATITL 2 MEGAKARYOCYTE-ASSOCIATED TYROSINE KINASE (MATK) FROM HOMOTITL 3 SAPIENS […]

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4FSS.B | RASA1

General Structure Information 4fss RASA1 crystal structure of a ras p21 protein activator (rasa1) from homo sapiens at 2.25 a resolution 2.25Å AUTH JOINT CENTER FOR STRUCTURAL GENOMICS (JCSG),AUTH 2 PARTNERSHIP FOR T-CELL BIOLOGY (TCELL)TITL CRYSTAL STRUCTURE OF A RAS P21 PROTEIN ACTIVATOR (RASA1)TITL 2 FROM HOMO SAPIENS AT 2.25 A RESOLUTIONREF TO BE PUBLISHEDREFN […]

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