4K0V.A | TEK

General Structure Information 4k0v TEK structural basis for angiopoietin-1 mediated signaling initiation 4.51Å AUTH X.YU,T.C.SEEGAR,A.C.DALTON,D.TZVETKOVA-ROBEV,Y.GOLDGUR,AUTH 2 K.R.RAJASHANKAR,D.B.NIKOLOV,W.A.BARTONTITL STRUCTURAL BASIS FOR ANGIOPOIETIN-1-MEDIATED SIGNALINGTITL 2 INITIATION.REF PROC.NATL.ACAD.SCI.USA V. 110 7205 2013REFN ISSN 0027-8424PMID 23592718DOI 10.1073/PNAS.1216890110 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2DBJ.A | MERTK

General Structure Information 2dbj MERTK solution structures of the fn3 domain of human proto- oncogene tyrosine-protein kinase mer precursor -1.0Å AUTH M.SATO,N.TOCHIO,S.KOSHIBA,M.INOUE,T.KIGAWA,AUTH 2 S.YOKOYAMATITL SOLUTION STRUCTURES OF THE FN3 DOMAIN OF HUMANTITL 2 PROTO-ONCOGENE TYROSINE-PROTEIN KINASE MERTITL 3 PRECURSORREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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1AWW.A | BTK

General Structure Information 1aww BTK sh3 domain from brutons tyrosine kinase, nmr, 42 structures -1.0Å AUTH H.HANSSON,P.T.MATTSSON,P.ALLARD,P.HAAPANIEMI,AUTH 2 M.VIHINEN,C.I.SMITH,T.HARDTITL SOLUTION STRUCTURE OF THE SH3 DOMAIN FROM BRUTONSTITL 2 TYROSINE KINASE.REF BIOCHEMISTRY V. 37 2912 1998REFN ISSN 0006-2960PMID 9485443DOI 10.1021/BI972409F Variant Set Distributions Mapped Variants

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1K2P.A | BTK

General Structure Information 1k2p BTK crystal structure of brutons tyrosine kinase domain 2.1Å AUTH C.MAO,M.ZHOU,F.M.UCKUNTITL CRYSTAL STRUCTURE OF BRUTONS TYROSINE KINASETITL 2 DOMAIN SUGGESTS A NOVEL PATHWAY FOR ACTIVATION ANDTITL 3 PROVIDES INSIGHTS INTO THE MOLECULAR BASIS OFTITL 4 X-LINKED AGAMMAGLOBULINEMIA.REF J.BIOL.CHEM. V. 276 41435 2001REFN ISSN 0021-9258PMID 11527964DOI 10.1074/JBC.M104828200 Variant Set Distributions Ripley’s K […]

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2VD5.A | DMPK

General Structure Information 2vd5 DMPK structure of human myotonic dystrophy protein kinase in complex with the bisindoylmaleide inhibitor bim viii 2.8Å AUTH J.ELKINS,A.AMOS,F.NIESEN,A.C.W.PIKE,O.FEDOROV,S.KNAPPTITL STRUCTURE OF DYSTROPHIA MYOTONICA PROTEIN KINASE.REF PROTEIN SCI. V. 18 782 2009REFN ISSN 0961-8368PMID 19309729DOI 10.1002/PRO.82 Variant Set Distributions Mapped Variants

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3DTC.A | MAP3K9

General Structure Information 3dtc MAP3K9 crystal structure of mixed-lineage kinase mlk1 complexed with compound 16 2.6Å AUTH R.L.HUDKINS,J.L.DIEBOLD,M.TAO,K.A.JOSEF,C.H.PARK,AUTH 2 T.S.ANGELES,L.D.AIMONE,J.HUSTEN,M.A.ATOR,S.L.MEYER,AUTH 3 B.P.HOLSKIN,J.T.DURKIN,A.A.FEDOROV,E.V.FEDOROV,AUTH 4 S.C.ALMO,J.R.MATHIASEN,D.BOZYCZKO-COYNE,AUTH 5 M.S.SAPORITO,R.W.SCOTT,J.P.MALLAMOTITL MIXED-LINEAGE KINASE 1 AND MIXED-LINEAGE KINASE 3TITL 2 SUBTYPE-SELECTIVETITL 3 DIHYDRONAPHTHYL[3,4-A]PYRROLO[3,4-C]CARBAZOLE-5-TITL 4 ONES: OPTIMIZATION, MIXED-LINEAGE KINASE 1TITL 5 CRYSTALLOGRAPHY, AND ORAL IN VIVO ACTIVITY INTITL 6 1-METHYL-4-PHENYLTETRAHYDROPYRIDINE MODELS.REF J.MED.CHEM. […]

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3U9C.A | CSNK2A1

General Structure Information 3u9c CSNK2A1 structure of a c-terminal deletion mutant of human protein kinase ck2 catalytic subunit with the atp-competitive inhibitor resorufin 3.2Å AUTH K.KLOPFFLEISCH,O.G.ISSINGER,K.NIEFINDTITL LOW-DENSITY CRYSTAL PACKING OF HUMAN PROTEIN KINASE CK2TITL 2 CATALYTIC SUBUNIT IN COMPLEX WITH RESORUFIN OR OTHERTITL 3 LIGANDS: A TOOL TO STUDY THE UNIQUE HINGE-REGION PLASTICITYTITL 4 OF […]

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3MTL.A | CDK16

General Structure Information 3mtl CDK16 crystal structure of the pctaire1 kinase in complex with indirubin e804 2.4Å AUTH T.KROJER,T.D.SHARPE,A.ROOS,P.SAVITSKY,A.AMOS,V.AYINAMPUDI,AUTH 2 G.BERRIDGE,O.FEDOROV,T.KEATES,C.PHILLIPS,N.BURGESS-BROWN,AUTH 3 Y.ZHANG,A.C.W.PIKE,J.MUNIZ,M.VOLLMAR,C.THANGARATNARAJAH,AUTH 4 P.RELLOS,E.UGOCHUKWU,P.FILIPPAKOPOULOS,W.YUE,S.DAS,AUTH 5 F.VON DELFT,A.EDWARDS,C.H.ARROWSMITH,J.WEIGELT,C.BOUNTRA,AUTH 6 S.KNAPP,A.BULLOCKTITL CRYSTAL STRUCTURE OF THE PCTAIRE1 KINASE IN COMPLEX WITHTITL 2 INDIRUBIN E804REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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1UNL.B | CDK5

General Structure Information 1unl CDK5 structural mechanism for the inhibition of cd5-p25 from the roscovitine, aloisine and indirubin. 2.2Å AUTH M.MAPELLI,L.MASSIMILINAO,C.CROVACE,M.A.SEELIGER,L.-H.TSAI,AUTH 2 L.MEIJER,A.MUSACCHIOTITL MECHANISM OF CDK5/P25 BINDING BY CDK INHIBITORSREF J.MED.CHEM. V. 48 671 2005REFN ISSN 0022-2623PMID 15689152DOI 10.1021/JM049323M Variant Set Distributions Mapped Variants

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1FVR.A | TEK

General Structure Information 1fvr TEK tie2 kinase domain 2.2Å AUTH L.M.SHEWCHUK,A.M.HASSELL,B.ELLIS,W.D.HOLMES,AUTH 2 R.DAVIS,E.L.HORNE,S.H.KADWELL,D.D.MCKEE,J.T.MOORETITL STRUCTURE OF THE TIE2 RTK DOMAIN: SELF-INHIBITIONTITL 2 BY THE NUCLEOTIDE BINDING LOOP, ACTIVATION LOOP,TITL 3 AND C-TERMINAL TAIL.REF STRUCTURE FOLD.DES. V. 8 1105 2000REFN ISSN 0969-2126PMID 11080633DOI 10.1016/S0969-2126(00)00516-5 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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