3B1U.A | PADI4

General Structure Information 3b1u PADI4 crystal structure of human peptidylarginine deiminase 4 in complex with o-f-amidine 2.1Å AUTH C.P.CAUSEY,J.E.JONES,J.L.SLACK,D.KAMEI,L.E.JONES JR,AUTH 2 V.SUBRAMANIAN,B.KNUCKLEY,P.EBRAHIMI,A.A.CHUMANEVICH,Y.LUO,AUTH 3 H.HASHIMOTO,M.SATO,L.J.HOFSETH,P.R.THOMPSONTITL THE DEVELOPMENT OFTITL 2 N-ALPHA-(2-CARBOXYL)BENZOYL-N(5)-(2-FLUORO-1-IMINOETHYL)-L-TITL 3 ORNITHINE AMIDE (O-F-AMIDINE) ANDTITL 4 N-ALPHA-(2-CARBOXYL)BENZOYL-N(5)-(2-CHLORO-1-IMINOETHYL)-L-TITL 5 ORNITHINE AMIDE (O-CL-AMIDINE) AS SECOND GENERATION PROTEINTITL 6 ARGININE DEIMINASE (PAD) INHIBITORSREF J.MED.CHEM. V. 54 6919 2011REFN ISSN […]

See Details
1UUC.A | SPINK5

General Structure Information 1uuc SPINK5 solution structure of a chimeric lekti-domain -1.0Å AUTH H.TIDOW,T.LAUBER,K.VITZITHUM,C.SOMMERHOFF,P.ROESCH,AUTH 2 U.C.MARXTITL THE SOLUTION STRUCTURE OF A CHIMERIC LEKTI DOMAINTITL 2 REVEALS A CHAMELEON SEQUENCEREF BIOCHEMISTRY V. 43 11238 2004REFN ISSN 0006-2960PMID 15366933DOI 10.1021/BI0492399 Variant Set Distributions Mapped Variants

See Details
3UA9.B | TNKS2

General Structure Information 3ua9 TNKS2 crystal structure of human tankyrase 2 in complex with a selective inhibitor 2.15Å AUTH M.NARWAL,H.VENKANNAGARI,L.LEHTIOTITL STRUCTURAL BASIS OF SELECTIVE INHIBITION OF HUMANTITL 2 TANKYRASES.REF J.MED.CHEM. V. 55 1360 2012REFN ISSN 0022-2623PMID 22233320DOI 10.1021/JM201510P Variant Set Distributions Mapped Variants

See Details
3MK6.A | PANK3

General Structure Information 3mk6 PANK3 substrate and inhibitor binding to pank 1.98Å AUTH R.LEONARDI,Y.M.ZHANG,M.K.YUN,R.ZHOU,F.Y.ZENG,W.LIN,J.CUI,AUTH 2 T.CHEN,C.O.ROCK,S.W.WHITE,S.JACKOWSKITITL MODULATION OF PANTOTHENATE KINASE 3 ACTIVITY BY SMALLTITL 2 MOLECULES THAT INTERACT WITH THE SUBSTRATE/ALLOSTERICTITL 3 REGULATORY DOMAIN.REF CHEM.BIOL. V. 17 892 2010REFN ISSN 1074-5521PMID 20797618DOI 10.1016/J.CHEMBIOL.2010.06.006 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity […]

See Details
3CEG.A | BIRC6

General Structure Information 3ceg BIRC6 crystal structure of the ubc domain of baculoviral iap repeat- containing protein 6 2.01Å AUTH Y.SHENG,J.H.HONG,R.DOHERTY,T.SRIKUMAR,J.SHLOUSH,AUTH 2 G.V.AVVAKUMOV,J.R.WALKER,S.XUE,D.NECULAI,J.W.WAN,S.K.KIM,AUTH 3 C.H.ARROWSMITH,B.RAUGHT,S.DHE-PAGANONTITL A HUMAN UBIQUITIN CONJUGATING ENZYME (E2)-HECT E3 LIGASETITL 2 STRUCTURE-FUNCTION SCREEN.REF MOL CELL PROTEOMICS V. 11 329 2012REFNPMID 22496338DOI 10.1074/MCP.O111.013706 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

See Details
4KS7.A | PAK6

General Structure Information 4ks7 PAK6 pak6 kinase domain in complex with pf-3758309 1.4Å AUTH J.GAO,B.H.HA,H.J.LOU,E.M.MORSE,R.ZHANG,D.A.CALDERWOOD,AUTH 2 B.E.TURK,T.J.BOGGONTITL SUBSTRATE AND INHIBITOR SPECIFICITY OF THE TYPE IITITL 2 P21-ACTIVATED KINASE, PAK6.REF PLOS ONE V. 8 77818 2013REFN ESSN 1932-6203PMID 24204982DOI 10.1371/JOURNAL.PONE.0077818 Variant Set Distributions Mapped Variants

See Details
3PB9.X | QPCTL

General Structure Information 3pb9 QPCTL crystal structure of the catalytic domain of human golgi-resident glutaminyl cyclase in complex with 1-benzylimidazole 1.12Å AUTH K.F.HUANG,S.S.LIAW,W.L.HUANG,C.Y.CHIA,Y.C.LO,Y.L.CHEN,AUTH 2 A.H.J.WANGTITL STRUCTURES OF HUMAN GOLGI-RESIDENT GLUTAMINYL CYCLASE ANDTITL 2 ITS COMPLEXES WITH INHIBITORS REVEAL A LARGE LOOP MOVEMENTTITL 3 UPON INHIBITOR BINDINGREF J.BIOL.CHEM. V. 286 12439 2011REFN ISSN 0021-9258PMID 21288892DOI 10.1074/JBC.M110.208595 […]

See Details
3T6J.A | DPP3

General Structure Information 3t6j DPP3 structure of human dppiii in complex with the opioid peptide tynorphin, at 3.0 angstroms 2.98Å AUTH G.A.BEZERRA,E.DOBROVETSKY,R.VIERTLMAYR,A.DONG,A.BINTER,AUTH 2 M.ABRAMIC,P.MACHEROUX,S.DHE-PAGANON,K.GRUBERTITL ENTROPY-DRIVEN BINDING OF OPIOID PEPTIDES INDUCES A LARGETITL 2 DOMAIN MOTION IN HUMAN DIPEPTIDYL PEPTIDASE III.REF PROC.NATL.ACAD.SCI.USA V. 109 6525 2012REFN ISSN 0027-8424PMID 22493238DOI 10.1073/PNAS.1118005109 Variant Set Distributions Ripley’s K Analysis […]

See Details
1UVG.A | SPINK5

General Structure Information 1uvg SPINK5 solution structure of the 15th domain of lekti -1.0Å AUTH H.TIDOW,T.LAUBER,K.VITZITHUM,C.SOMMERHOFF,P.ROESCH,AUTH 2 U.C.MARXTITL THE SOLUTION STRUCTURE OF A CHIMERIC LEKTI DOMAINTITL 2 REVEALS A CHAMELEON SEQUENCEREF BIOCHEMISTRY V. 43 11238 2004REFN ISSN 0006-2960PMID 15366933DOI 10.1021/BI0492399 Variant Set Distributions Mapped Variants

See Details
3D8C.A | HIF1AN

General Structure Information 3d8c HIF1AN factor inhibiting hif-1 alpha d201g mutant in complex with zn(ii), alpha-ketoglutarate and hif-1 alpha 19mer 2.1Å AUTH K.S.HEWITSON,S.L.HOLMES,D.EHRISMANN,A.P.HARDY,R.CHOWDHURY,AUTH 2 C.J.SCHOFIELD,M.A.MCDONOUGHTITL EVIDENCE THAT TWO ENZYME-DERIVED HISTIDINE LIGANDS ARETITL 2 SUFFICIENT FOR IRON BINDING AND CATALYSIS BY FACTORTITL 3 INHIBITING HIF (FIH).REF J.BIOL.CHEM. V. 283 25971 2008REFN ISSN 0021-9258PMID 18611856DOI 10.1074/JBC.M804999200 Variant […]

See Details