1B0F.A | ELANE

General Structure Information 1b0f ELANE crystal structure of human neutrophil elastase with mdl 101, 146 3.0Å AUTH R.J.CREGGE,S.L.DURHAM,R.A.FARR,S.L.GALLION,C.M.HARE,AUTH 2 R.V.HOFFMAN,M.J.JANUSZ,H.O.KIM,J.R.KOEHL,S.MEHDI,W.A.METZ,AUTH 3 N.P.PEET,J.T.PELTON,H.A.SCHREUDER,S.SUNDER,C.TARDIFTITL INHIBITION OF HUMAN NEUTROPHIL ELASTASE. 4. DESIGN,TITL 2 SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, ANDTITL 3 STRUCTURE-ACTIVITY RELATIONSHIPS FOR A SERIES OFTITL 4 P2-MODIFIED, ORALLY ACTIVE PEPTIDYL PENTAFLUOROETHYLTITL 5 KETONES.REF J.MED.CHEM. V. 41 2461 1998REFN […]

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1YGR.B | PTPRC

General Structure Information 1ygr PTPRC crystal structure of the tandem phosphatase domain of rptp cd45 2.9Å AUTH H.J.NAM,F.POY,H.SAITO,C.A.FREDERICKTITL STRUCTURAL BASIS FOR THE FUNCTION AND REGULATIONTITL 2 OF THE RECEPTOR PROTEIN TYROSINE PHOSPHATASE CD45.REF J.EXP.MED. V. 201 441 2005REFN ISSN 0022-1007PMID 15684325DOI 10.1084/JEM.20041890 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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2XWB.A | C3

General Structure Information 2xwb C3 crystal structure of complement c3b in complex with factors b and d 3.49Å AUTH F.FORNERIS,D.RICKLIN,J.WU,A.TZEKOU,R.S.WALLACE,J.D.LAMBRIS,AUTH 2 P.GROSTITL STRUCTURES OF C3B IN COMPLEX WITH FACTORS B AND D GIVETITL 2 INSIGHT INTO COMPLEMENT CONVERTASE FORMATION.REF SCIENCE V. 330 1816 2010REFN ISSN 0036-8075PMID 21205667DOI 10.1126/SCIENCE.1195821 Variant Set Distributions Ripley’s K Analysis Plots […]

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2XWB.H | CFB

General Structure Information 2xwb CFB crystal structure of complement c3b in complex with factors b and d 3.49Å AUTH F.FORNERIS,D.RICKLIN,J.WU,A.TZEKOU,R.S.WALLACE,J.D.LAMBRIS,AUTH 2 P.GROSTITL STRUCTURES OF C3B IN COMPLEX WITH FACTORS B AND D GIVETITL 2 INSIGHT INTO COMPLEMENT CONVERTASE FORMATION.REF SCIENCE V. 330 1816 2010REFN ISSN 0036-8075PMID 21205667DOI 10.1126/SCIENCE.1195821 Variant Set Distributions Ripley’s K Analysis Plots […]

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1KSN.B | F10

General Structure Information 1ksn F10 crystal structure of human coagulation factor xa complexed with fxv673 2.1Å AUTH K.R.GUERTIN,C.J.GARDNER,S.I.KLEIN,A.L.ZULLI,AUTH 2 M.CZEKAJ,Y.GONG,A.P.SPADA,D.L.CHENEY,S.MAIGNAN,AUTH 3 J.P.GUILLOTEAU,K.D.BROWN,D.J.COLUSSI,V.CHU,AUTH 4 C.L.HERAN,S.R.MORGAN,R.G.BENTLEY,C.T.DUNWIDDIE,AUTH 5 R.J.LEADLEY,H.W.PAULSTITL OPTIMIZATION OF THE BETA-AMINOESTER CLASS OFTITL 2 FACTOR XA INHIBITORS. PART 2: IDENTIFICATION OFTITL 3 FXV673 AS A POTENT AND SELECTIVE INHIBITOR WITHTITL 4 EXCELLENT IN VIVO ANTICOAGULANT ACTIVITY.REF […]

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1NB3.I | CSTA

General Structure Information 1nb3 CSTA crystal structure of stefin a in complex with cathepsin h: n-terminal residues of inhibitors can adapt to the active sites of endo-and exopeptidases 2.8Å AUTH S.JENKO,I.DOLENC,G.GUNCAR,A.DOBERSEK,M.PODOBNIK,D.TURKTITL CRYSTAL STRUCTURE OF STEFIN A IN COMPLEX WITH CATHEPSIN H:TITL 2 N-TERMINAL RESIDUES OF INHIBITORS CAN ADAPT TO THE ACTIVETITL 3 SITES OF ENDO- […]

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3NXP.A | F2

General Structure Information 3nxp F2 crystal structure of human prethrombin-1 2.2Å AUTH Z.CHEN,L.A.PELC,E.DI CERATITL CRYSTAL STRUCTURE OF PRETHROMBIN-1.REF PROC.NATL.ACAD.SCI.USA V. 107 19278 2010REFN ISSN 0027-8424PMID 20974933DOI 10.1073/PNAS.1010262107 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3Q91.D | NUDT14

General Structure Information 3q91 NUDT14 crystal structure of human uridine diphosphate glucose pyrophosphatase (nudt14) 2.7Å AUTH L.TRESAUGUES,M.I.SIPONEN,C.H.ARROWSMITH,H.BERGLUND,AUTH 2 C.BOUNTRA,R.COLLINS,A.M.EDWARDS,T.EKBLAD,S.FLODIN,A.FLORES,AUTH 3 S.GRASLUND,M.HAMMARSTROM,I.JOHANSSON,T.KARLBERG,S.KOL,AUTH 4 T.KOTENYOVA,E.KOUZNETSOVA,M.MOCHE,T.NYMAN,C.PERSSON,AUTH 5 H.SCHULER,P.SCHUTZ,A.G.THORSELL,S.VAN DER BERG,E.WAHLBERG,AUTH 6 J.WEIGELT,M.WELIN,P.NORDLUNDTITL CRYSTAL STRUCTURE OF HUMAN URIDINE DIPHOSPHATE GLUCOSETITL 2 PYROPHOSPHATASE (NUDT14)REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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2F83.A | F11

General Structure Information 2f83 F11 crystal structure at 2.9 angstroms resolution of human plasma coagulation factor xi zymogen 2.87Å AUTH E.PAPAGRIGORIOU,P.A.MCEWAN,P.N.WALSH,J.EMSLEYTITL CRYSTAL STRUCTURE OF THE FACTOR XI ZYMOGEN REVEALS A PATHWAYTITL 2 FOR TRANSACTIVATION.REF NAT.STRUCT.MOL.BIOL. V. 13 557 2006REFN ISSN 1545-9993PMID 16699514DOI 10.1038/NSMB1095 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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2WEF.A | BPNT1

General Structure Information 2wef BPNT1 human 3(2), 5-bisphosphate nucleotidase 1 (bpnt1) in complex with amp, po4 and magnesium 1.8Å AUTH M.MOCHE,P.SCHUTZ,C.H.ARROWSMITH,H.BERGLUND,AUTH 2 C.BOUNTRA,R.COLLINS,L.G.DAHLGREN,A.M.EDWARDS,AUTH 3 S.FLODIN,A.FLORES,S.GRASLUND,M.HAMMARSTROM,AUTH 4 A.JOHANSSON,I.JOHANSSON,T.KARLBERG,T.KOTENYOVA,AUTH 5 M.E.NILSSON,T.NYMAN,C.PERSSON,J.SAGEMARK,AUTH 6 H.SCHUELER,M.I.SIPONEN,A.G.THORSELL,L.TRESAUGUES,AUTH 7 S.VAN DEN BERG,J.WEIGELT,M.WELIN,M.WISNIEWSKA,AUTH 8 P.NORDLUNDTITL HUMAN 3(2), 5-BISPHOSPHATE NUCLEOTIDASE 1 (TITL 2 BPNT1) IN COMPLEX WITH AMP, PO4 AND MAGNESIUMREF TO BE PUBLISHEDREFN […]

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