3FUK.A | LTA4H

General Structure Information 3fuk LTA4H leukotriene a4 hydrolase in complex with 1-[2-(1h-indol-5- yloxy)ethyl]piperidine-4-carboxylic acid 1.95Å AUTH D.R.DAVIES,B.MAMAT,O.T.MAGNUSSON,J.CHRISTENSEN,AUTH 2 M.H.HARALDSSON,R.MISHRA,B.PEASE,E.HANSEN,J.SINGH,AUTH 3 D.ZEMBOWER,H.KIM,A.S.KISELYOV,A.B.BURGIN,AUTH 4 M.E.GURNEY,L.J.STEWARTTITL DISCOVERY OF LEUKOTRIENE A4 HYDROLASE INHIBITORSTITL 2 USING METABOLOMICS BIASED FRAGMENT CRYSTALLOGRAPHY.REF J.MED.CHEM. V. 52 4694 2009REFN ISSN 0022-2623PMID 19618939DOI 10.1021/JM900259H Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic […]

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2X2M.B | RET

General Structure Information 2x2m RET crystal structure of phosphorylated ret tyrosine kinase domain with inhibitor 2.5Å AUTH L.MOLOGNI,R.ROSTAGNO,S.BRUSSOLO,P.P.KNOWLES,AUTH 2 S.KJAER,J.MURRAY-RUST,E.ROSSO,A.ZAMBON,L.SCAPOZZA,AUTH 3 N.Q.MCDONALD,V.LUCCHINI,C.GAMBACORTI-PASSERINITITL SYNTHESIS, STRUCTURE-ACTIVITY RELATIONSHIP ANDTITL 2 CRYSTALLOGRAPHIC STUDIES OF 3-SUBSTITUTED INDOLIN-TITL 3 2-ONE RET INHIBITORS.REF BIOORG.MED.CHEM. V. 18 1482 2010REFN ISSN 0968-0896PMID 20117004DOI 10.1016/J.BMC.2010.01.011 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

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1BHG.A | GUSB

General Structure Information 1bhg GUSB human beta-glucuronidase at 2.6 a resolution 2.53Å AUTH S.JAIN,W.B.DRENDEL,Z.W.CHEN,F.S.MATHEWS,W.S.SLY,J.H.GRUBBTITL STRUCTURE OF HUMAN BETA-GLUCURONIDASE REVEALS CANDIDATETITL 2 LYSOSOMAL TARGETING AND ACTIVE-SITE MOTIFS.REF NAT.STRUCT.BIOL. V. 3 375 1996REFN ISSN 1072-8368PMID 8599764DOI 10.1038/NSB0496-375 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1Z10.D | CYP2A6

General Structure Information 1z10 CYP2A6 crystal structure of human microsomal p450 2a6 with coumarin bound 1.9Å AUTH J.K.YANO,M.H.HSU,K.J.GRIFFIN,C.D.STOUT,E.F.JOHNSONTITL STRUCTURES OF HUMAN MICROSOMAL CYTOCHROME P450 2A6 COMPLEXEDTITL 2 WITH COUMARIN AND METHOXSALENREF NAT.STRUCT.MOL.BIOL. V. 12 822 2005REFN ISSN 1545-9993PMID 16086027DOI 10.1038/NSMB971 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1EGD.A | ACADM

General Structure Information 1egd ACADM structure of t255e, e376g mutant of human medium chain acyl- coa dehydrogenase 2.4Å AUTH H.J.LEE,M.WANG,R.PASCHKE,A.NANDY,S.GHISLA,J.J.KIMTITL CRYSTAL STRUCTURES OF THE WILD TYPE AND THETITL 2 GLU376GLY/THR255GLU MUTANT OF HUMAN MEDIUM-CHAINTITL 3 ACYL-COA DEHYDROGENASE: INFLUENCE OF THE LOCATIONTITL 4 OF THE CATALYTIC BASE ON SUBSTRATE SPECIFICITY.REF BIOCHEMISTRY V. 35 12412 1996REFN ISSN […]

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1Q68.B | LCK

General Structure Information 1q68 LCK solution structure of t-cell surface glycoprotein cd4 and proto-oncogene tyrosine-protein kinase lck fragments -1.0Å AUTH P.W.KIM,Z.Y.SUN,S.C.BLACKLOW,G.WAGNER,M.J.ECKTITL A ZINC CLASP STRUCTURE TETHERS LCK TO T CELLTITL 2 CORECEPTORS CD4 AND CD8.REF SCIENCE V. 301 1725 2003REFN ISSN 0036-8075PMID 14500983DOI 10.1126/SCIENCE.1085643 Variant Set Distributions Mapped Variants

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1KF9.C | GHR

General Structure Information 1kf9 GHR phage display derived variant of human growth hormone complexed with two copies of the extracellular domain of its receptor 2.6Å AUTH C.A.SCHIFFER,M.ULTSCH,S.WALSH,W.SOMERS,A.M.DE VOS,AUTH 2 A.A.KOSSIAKOFFTITL STRUCTURE OF A PHAGE DISPLAY DERIVED VARIANT OFTITL 2 HUMAN GROWTH HORMONE COMPLEXED TO TWO COPIES OFTITL 3 THE EXTRACELLULAR DOMAIN OF ITS RECEPTOR: EVIDENCETITL […]

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2Y5B.F | UBB

General Structure Information 2y5b UBB structure of usp21 in complex with linear diubiquitin-aldehyde 2.7Å AUTH Y.YE,M.AKUTSU,F.REYES-TURCU,R.I.ENCHEV,K.D.WILKINSON,AUTH 2 D.KOMANDERTITL POLYUBIQUITIN BINDING AND CROSS-REACTIVITY IN THE USPTITL 2 DOMAIN DEUBIQUITINASE USP21.REF EMBO REP. V. 12 350 2011REFN ISSN 1469-221XPMID 21399617DOI 10.1038/EMBOR.2011.17 Variant Set Distributions Mapped Variants

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2FJ9.A | DBI

General Structure Information 2fj9 DBI high resolution crystal structure of the unliganded human acbp 1.6Å AUTH J.P.TASKINEN,D.M.VAN AALTEN,J.KNUDSEN,R.K.WIERENGATITL HIGH RESOLUTION CRYSTAL STRUCTURES OF UNLIGANDED ANDTITL 2 LIGANDED HUMAN LIVER ACBP REVEAL A NEW MODE OF BINDING FORTITL 3 THE ACYL-COA LIGAND.REF PROTEINS V. 66 229 2006REFN ISSN 0887-3585PMID 17044054DOI 10.1002/PROT.21124 Variant Set Distributions Mapped Variants

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1TRN.A | PRSS1

General Structure Information 1trn PRSS1 crystal structure of human trypsin 1: unexpected phosphorylation of tyrosine 151 2.2Å AUTH C.GABORIAUD,L.SERRE,O.GUY-CROTTE,E.FOREST,AUTH 2 J.C.FONTECILLA-CAMPSTITL CRYSTAL STRUCTURE OF HUMAN TRYPSIN 1: UNEXPECTEDTITL 2 PHOSPHORYLATION OF TYR151.REF J.MOL.BIOL. V. 259 995 1996REFN ISSN 0022-2836PMID 8683601DOI 10.1006/JMBI.1996.0376 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped […]

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