1M3G.A | DUSP2

General Structure Information 1m3g DUSP2 solution structure of the catalytic domain of mapk phosphatase pac-1: insights into substrate-induced enzymatic activation -1.0Å AUTH A.FAROOQ,O.PLOTNIKOVA,G.CHATURVEDI,S.YAN,L.ZENG,AUTH 2 Q.ZHANG,M.-M.ZHOUTITL SOLUTION STRUCTURE OF THE MAPK PHOSPHATASE PAC-1TITL 2 CATALYTIC DOMAIN INSIGHTS INTO SUBSTRATE-INDUCEDTITL 3 ENZYMATIC ACTIVATION OF MKPREF STRUCTURE V. 11 155 2003REFN ISSN 0969-2126PMID 12575935DOI 10.1016/S0969-2126(02)00943-7 Variant Set Distributions […]

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3V5L.A | ITK

General Structure Information 3v5l ITK crystal structure of interleukin-2 inducible t-cell kinase itk catalytic domain with thienopyrazolylindole inhibitor 542 1.86Å AUTH L.R.MCLEAN,Y.ZHANG,N.ZAIDI,X.BI,R.WANG,R.DHARANIPRAGADA,AUTH 2 J.G.JURCAK,T.A.GILLESPY,Z.ZHAO,K.Y.MUSICK,Y.M.CHOI,AUTH 3 M.BARRAGUE,J.PEPPARD,M.SMICKER,M.DUGUID,A.PARKAR,J.FORDHAM,AUTH 4 D.KOMINOSTITL X-RAY CRYSTALLOGRAPHIC STRUCTURE-BASED DESIGN OF SELECTIVETITL 2 THIENOPYRAZOLE INHIBITORS FOR INTERLEUKIN-2-INDUCIBLETITL 3 TYROSINE KINASE.REF BIOORG.MED.CHEM.LETT. V. 22 3296 2012REFN ISSN 0960-894XPMID 22464456DOI 10.1016/J.BMCL.2012.03.016 Variant Set Distributions Ripley’s […]

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3W7R.A | DHODH

General Structure Information 3w7r DHODH structure of human dihydroorotate dehydrogenase in complex with mii-4- 097 1.68Å AUTH D.K.INAOKA,M.IIDA,T.TABUCHI,N.LEE,S.HASHIMOTO,S.MATSUOKA,AUTH 2 T.KURANAGA,T.SHIBA,K.SAKAMOTO,S.SUZUKI,E.O.BALOGUN,T.NARA,AUTH 3 T.AOKI,M.INOUE,T.HONMA,A.TANAKA,S.HARADA,K.KITATITL STRUCTURE OF HUMAN DIHYDROOROTATE DEHYDROGENASE IN COMPLEXTITL 2 WITH MII-4-097REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3W7R.A | DHODH

General Structure Information 3w7r DHODH structure of human dihydroorotate dehydrogenase in complex with mii-4- 097 1.68Å AUTH D.K.INAOKA,M.IIDA,T.TABUCHI,N.LEE,S.HASHIMOTO,S.MATSUOKA,AUTH 2 T.KURANAGA,T.SHIBA,K.SAKAMOTO,S.SUZUKI,E.O.BALOGUN,T.NARA,AUTH 3 T.AOKI,M.INOUE,T.HONMA,A.TANAKA,S.HARADA,K.KITATITL STRUCTURE OF HUMAN DIHYDROOROTATE DEHYDROGENASE IN COMPLEXTITL 2 WITH MII-4-097REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3W7R.A | DHODH

General Structure Information 3w7r DHODH structure of human dihydroorotate dehydrogenase in complex with mii-4- 097 1.68Å AUTH D.K.INAOKA,M.IIDA,T.TABUCHI,N.LEE,S.HASHIMOTO,S.MATSUOKA,AUTH 2 T.KURANAGA,T.SHIBA,K.SAKAMOTO,S.SUZUKI,E.O.BALOGUN,T.NARA,AUTH 3 T.AOKI,M.INOUE,T.HONMA,A.TANAKA,S.HARADA,K.KITATITL STRUCTURE OF HUMAN DIHYDROOROTATE DEHYDROGENASE IN COMPLEXTITL 2 WITH MII-4-097REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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4NR2.D | STK4

General Structure Information 4nr2 STK4 crystal structure of stk4 (mst1) sarah domain 2.0Å AUTH A.CHAIKUAD,T.KROJER,J.KOPEC,F.VON DELFT,C.H.ARROWSMITH,AUTH 2 A.M.EDWARDS,C.BOUNTRA,S.KNAPP,AUTH 3 STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL CRYSTAL STRUCTURE OF STK4 (MST1) SARAH DOMAINREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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4NR2.D | STK4

General Structure Information 4nr2 STK4 crystal structure of stk4 (mst1) sarah domain 2.0Å AUTH A.CHAIKUAD,T.KROJER,J.KOPEC,F.VON DELFT,C.H.ARROWSMITH,AUTH 2 A.M.EDWARDS,C.BOUNTRA,S.KNAPP,AUTH 3 STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL CRYSTAL STRUCTURE OF STK4 (MST1) SARAH DOMAINREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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4NR2.D | STK4

General Structure Information 4nr2 STK4 crystal structure of stk4 (mst1) sarah domain 2.0Å AUTH A.CHAIKUAD,T.KROJER,J.KOPEC,F.VON DELFT,C.H.ARROWSMITH,AUTH 2 A.M.EDWARDS,C.BOUNTRA,S.KNAPP,AUTH 3 STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL CRYSTAL STRUCTURE OF STK4 (MST1) SARAH DOMAINREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2ENN.A | PRKCQ

General Structure Information 2enn PRKCQ solution structure of the first c1 domain from human protein kinase c theta -1.0Å AUTH T.NAGASHIMA,F.HAYASHI,S.YOKOYAMATITL SOLUTION STRUCTURE OF THE FIRST C1 DOMAIN FROMTITL 2 HUMAN PROTEIN KINASE C THETAREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1YRK.A | PRKCD

General Structure Information 1yrk PRKCD the c2 domain of pkc is a new phospho-tyrosine binding domain 1.7Å AUTH C.H.BENES,N.WU,A.E.ELIA,T.DHARIA,L.C.CANTLEY,AUTH 2 S.P.SOLTOFFTITL THE C2 DOMAIN OF PKCDELTA IS A PHOSPHOTYROSINETITL 2 BINDING DOMAIN.REF CELL(CAMBRIDGE,MASS.) V. 121 271 2005REFN ISSN 0092-8674PMID 15851022DOI 10.1016/J.CELL.2005.02.019 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped […]

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