2QXI.A | KLK7

General Structure Information 2qxi KLK7 high resolution structure of human kallikrein 7 in complex with suc-ala-ala-pro-phe-chloromethylketone 1.0Å AUTH M.DEBELA,P.HESS,V.MAGDOLEN,N.M.SCHECHTER,T.STEINER,AUTH 2 R.HUBER,W.BODE,P.GOETTIGTITL CHYMOTRYPTIC SPECIFICITY DETERMINANTS IN THE 1.0 ATITL 2 STRUCTURE OF THE ZINC-INHIBITED HUMAN TISSUETITL 3 KALLIKREIN 7.REF PROC.NATL.ACAD.SCI.USA V. 104 16086 2007REFN ISSN 0027-8424PMID 17909180DOI 10.1073/PNAS.0707811104 Variant Set Distributions Ripley’s K Analysis Plots Variant […]

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3E37.A | FNTA

General Structure Information 3e37 FNTA protein farnesyltransferase complexed with bisubstrate ethylenediamine scaffold inhibitor 5 1.8Å AUTH M.A.HAST,S.FLETCHER,C.G.CUMMINGS,E.E.PUSATERI,AUTH 2 M.A.BLASKOVICH,K.RIVAS,M.H.GELB,W.C.VAN VOORHIS,AUTH 3 S.M.SEBTI,A.D.HAMILTON,L.S.BEESETITL STRUCTURAL BASIS FOR BINDING AND SELECTIVITY OFTITL 2 ANTIMALARIAL AND ANTICANCER ETHYLENEDIAMINETITL 3 INHIBITORS TO PROTEIN FARNESYLTRANSFERASE.REF CHEM.BIOL. V. 16 181 2009REFN ISSN 1074-5521PMID 19246009DOI 10.1016/J.CHEMBIOL.2009.01.014 Variant Set Distributions Ripley’s K Analysis Plots […]

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2AOT.B | HNMT

General Structure Information 2aot HNMT histamine methyltransferase complexed with the antihistamine drug diphenhydramine 1.9Å AUTH J.R.HORTON,K.SAWADA,M.NISHIBORI,X.CHENGTITL STRUCTURAL BASIS FOR INHIBITION OF HISTAMINETITL 2 N-METHYLTRANSFERASE BY DIVERSE DRUGSREF J.MOL.BIOL. V. 353 334 2005REFN ISSN 0022-2836PMID 16168438DOI 10.1016/J.JMB.2005.08.040 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3Q2U.A | GLIPR1

General Structure Information 3q2u GLIPR1 structure of human glioma pathogenesis-related protein 1 reveals unique loops and surface motifs. 1.85Å AUTH O.A.ASOJO,R.A.KOSKI,N.BONAFETITL STRUCTURAL STUDIES OF HUMAN GLIOMA PATHOGENESIS-RELATEDTITL 2 PROTEIN 1.REF ACTA CRYSTALLOGR.,SECT.D V. 67 847 2011REFN ISSN 0907-4449PMID 21931216DOI 10.1107/S0907444911028198 Variant Set Distributions Mapped Variants

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1NE7.D | GNPDA1

General Structure Information 1ne7 GNPDA1 human glucosamine-6-phosphate deaminase isomerase at 1.75 a resolution complexed with n-acetyl-glucosamine-6-phosphate and 2-deoxy-2-amino-glucitol-6-phosphate 1.75Å AUTH R.ARREOLA,B.VALDERRAMA,M.L.MORANTE,E.HORJALESTITL TWO MAMMALIAN GLUCOSAMINE-6-PHOSPHATE DEAMINASES:TITL 2 A STRUCTURAL AND GENETIC STUDY.REF FEBS LETT. V. 551 63 2003REFN ISSN 0014-5793PMID 12965206DOI 10.1016/S0014-5793(03)00896-2 Variant Set Distributions Mapped Variants

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2D5R.B | TOB1

General Structure Information 2d5r TOB1 crystal structure of a tob-hcaf1 complex 2.5Å AUTH M.HORIUCHI,K.TAKEUCHI,N.NODA,N.MUROYA,T.SUZUKI,AUTH 2 T.NAKAMURA,J.KAWAMURA-TSUZUKU,K.TAKAHASI,AUTH 3 T.YAMAMOTO,F.INAGAKITITL STRUCTURAL BASIS FOR THE ANTIPROLIFERATIVE ACTIVITYTITL 2 OF THE TOB-HCAF1 COMPLEX.REF J.BIOL.CHEM. V. 284 13244 2009REFN ISSN 0021-9258PMID 19276069DOI 10.1074/JBC.M809250200 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3PFF.A | ACLY

General Structure Information 3pff ACLY truncated human atp-citrate lyase with adp and tartrate bound 2.3Å AUTH T.SUN,K.HAYAKAWA,M.E.FRASERTITL ADP-MG2+ BOUND TO THE ATP-GRASP DOMAIN OF ATP-CITRATE LYASE.REF ACTA CRYSTALLOGR.,SECT.F V. 67 1168 2011REFN ESSN 1744-3091PMID 22102020DOI 10.1107/S1744309111028363 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3FEY.C | KPNA2

General Structure Information 3fey KPNA2 crystal structure of the cbc-importin alpha complex. 2.2Å AUTH S.M.DIAS,K.F.WILSON,K.S.ROJAS,A.L.AMBROSIO,R.A.CERIONETITL THE MOLECULAR BASIS FOR THE REGULATION OF THE CAP-BINDINGTITL 2 COMPLEX BY THE IMPORTINS.REF NAT.STRUCT.MOL.BIOL. V. 16 930 2009REFN ISSN 1545-9993PMID 19668212DOI 10.1038/NSMB.1649 Variant Set Distributions Mapped Variants

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1KO6.A | NUP98

General Structure Information 1ko6 NUP98 crystal structure of c-terminal autoproteolytic domain of nucleoporin nup98 3.0Å AUTH A.E.HODEL,M.R.HODEL,E.R.GRIFFIS,K.A.HENNIG,AUTH 2 G.A.RATNER,S.XU,M.A.POWERSTITL THE THREE-DIMENSIONAL STRUCTURE OF THETITL 2 AUTOPROTEOLYTIC, NUCLEAR PORE-TARGETING DOMAIN OFTITL 3 THE HUMAN NUCLEOPORIN NUP98.REF MOL.CELL V. 10 347 2002REFN ISSN 1097-2765PMID 12191480DOI 10.1016/S1097-2765(02)00589-0 Variant Set Distributions Mapped Variants

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2ZKS.A | GZMM

General Structure Information 2zks GZMM structural insights into the proteolytic machinery of apoptosis- inducing granzyme m 2.7Å AUTH L.WU,L.WANG,G.HUA,K.LIU,X.YANG,Y.ZHAI,M.BARTLAM,F.SUN,Z.FANTITL STRUCTURAL BASIS FOR PROTEOLYTIC SPECIFICITY OF THE HUMANTITL 2 APOPTOSIS-INDUCING GRANZYME MREF J.IMMUNOL. V. 183 421 2009REFN ISSN 0022-1767PMID 19542453DOI 10.4049/JIMMUNOL.0803088 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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