2RJP.C | ADAMTS4

General Structure Information 2rjp ADAMTS4 crystal structure of adamts4 with inhibitor bound 2.8Å AUTH L.MOSYAK,K.GEORGIADIS,T.SHANE,K.SVENSON,T.HEBERT,AUTH 2 T.MCDONAGH,S.MACKIE,S.OLLAND,L.LIN,X.ZHONG,R.KRIZ,AUTH 3 E.L.REIFENBERG,L.A.COLLINS-RACIE,C.CORCORAN,AUTH 4 B.FREEMAN,R.ZOLLNER,T.MARVELL,M.VERA,P.E.SUM,AUTH 5 E.R.LAVALLIE,M.STAHL,W.SOMERSTITL CRYSTAL STRUCTURES OF THE TWO MAJOR AGGRECANTITL 2 DEGRADING ENZYMES, ADAMTS4 AND ADAMTS5.REF PROTEIN SCI. V. 17 16 2008REFN ISSN 0961-8368PMID 18042673DOI 10.1110/PS.073287008 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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1FJ2.A | LYPLA1

General Structure Information 1fj2 LYPLA1 crystal structure of the human acyl protein thioesterase 1 at 1.5 a resolution 1.5Å AUTH Y.DEVEDJIEV,Z.DAUTER,S.R.KUZNETSOV,T.L.JONES,Z.S.DEREWENDATITL CRYSTAL STRUCTURE OF THE HUMAN ACYL PROTEIN THIOESTERASE ITITL 2 FROM A SINGLE X-RAY DATA SET TO 1.5 A.REF STRUCTURE FOLD.DES. V. 8 1137 2000REFN ISSN 0969-2126PMID 11080636DOI 10.1016/S0969-2126(00)00529-3 Variant Set Distributions Ripley’s K […]

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4AW6.E | ZMPSTE24

General Structure Information 4aw6 ZMPSTE24 crystal structure of the human nuclear membrane zinc metalloprotease zmpste24 (face1) 3.4Å AUTH A.QUIGLEY,Y.Y.DONG,A.C.W.PIKE,L.DONG,L.SHRESTHA,G.BERRIDGE,AUTH 2 P.J.STANSFELD,M.S.P.SANSOM,A.M.EDWARDS,C.BOUNTRA,AUTH 3 F.VON DELFT,A.N.BULLOCK,N.A.BURGESS-BROWN,E.P.CARPENTERTITL THE STRUCTURAL BASIS OF ZMPSTE24-DEPENDENT LAMINOPATHIES.REF SCIENCE V. 339 1604 2013REFN ISSN 0036-8075PMID 23539603DOI 10.1126/SCIENCE.1231513 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2JAJ.B | DDAH1

General Structure Information 2jaj DDAH1 ddah1 complexed with l-257 2.0Å AUTH J.LEIPER,M.NANDI,B.TORONDEL,J.MURRAY-RUST,M.MALAKI,B.OHARA,AUTH 2 S.ROSSITER,S.ANTHONY,M.MADHANI,D.SELWOOD,C.SMITH,AUTH 3 B.WOJCIAK-STOTHARD,A.RUDIGER,R.STIDWILL,N.Q.MCDONALD,AUTH 4 P.VALLANCETITL DISRUPTION OF METHYLARGININE METABOLISM IMPAIRS VASCULARTITL 2 HOMEOSTASIS.REF NAT.MED. (N.Y.) V. 13 198 2007REFN ISSN 1078-8956PMID 17273169DOI 10.1038/NM1543 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3B4V.H | FSTL3

General Structure Information 3b4v FSTL3 x-ray structure of activin in complex with fstl3 2.48Å AUTH R.STAMLER,H.T.KEUTMANN,Y.SIDIS,C.KATTAMURI,A.SCHNEYER,AUTH 2 T.B.THOMPSONTITL THE STRUCTURE OF FSTL3.ACTIVIN A COMPLEX. DIFFERENTIALTITL 2 BINDING OF N-TERMINAL DOMAINS INFLUENCES FOLLISTATIN-TYPETITL 3 ANTAGONIST SPECIFICITY.REF J.BIOL.CHEM. V. 283 32831 2008REFN ISSN 0021-9258PMID 18768470DOI 10.1074/JBC.M801266200 Variant Set Distributions Mapped Variants

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3QYB.A | TBC1D4

General Structure Information 3qyb TBC1D4 x-ray crystal structure of human tbc1d4 (as160) rabgap domain 3.5Å AUTH S.Y.PARK,W.JIN,J.R.WOO,S.E.SHOELSONTITL CRYSTAL STRUCTURES OF HUMAN TBC1D1 AND TBC1D4 (AS160)TITL 2 RABGTPASE-ACTIVATING PROTEIN (RABGAP) DOMAINS REVEALTITL 3 CRITICAL ELEMENTS FOR GLUT4 TRANSLOCATION.REF J.BIOL.CHEM. V. 286 18130 2011REFN ISSN 0021-9258PMID 21454505DOI 10.1074/JBC.M110.217323 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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2WFH.B | SLIT2

General Structure Information 2wfh SLIT2 the human slit 2 dimerization domain d4 1.8Å AUTH E.SEIRADAKE,A.C.VON PHILIPSBORN,M.HENRY,M.FRITZ,AUTH 2 H.LORTAT-JACOB,M.JAMIN,W.HEMRIKA,M.BASTMEYER,S.CUSACK,AUTH 3 A.A.MCCARTHYTITL STRUCTURE AND FUNCTIONAL RELEVANCE OF THE SLIT2TITL 2 HOMODIMERIZATION DOMAIN.REF EMBO REP. V. 10 736 2009REFN ISSN 1469-221XPMID 19498462DOI 10.1038/EMBOR.2009.95 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2DL5.A | FCHSD2

General Structure Information 2dl5 FCHSD2 solution structure of the first sh3 domain of human kiaa0769 protein -1.0Å AUTH X.R.QIN,K.IZUMI,M.YOSHIDA,F.HAYASHI,S.YOKOYAMATITL SOLUTION STRUCTURE OF THE FIRST SH3 DOMAIN OFTITL 2 HUMAN KIAA0769 PROTEINREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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3Q3J.A | PLXNA2

General Structure Information 3q3j PLXNA2 crystal structure of plexin a2 rbd in complex with rnd1 1.97Å AUTH H.WANG,W.TEMPEL,Y.TONG,X.GUAN,L.SHEN,L.BUREN,N.ZHANG,AUTH 2 A.K.WERNIMONT,L.CROMBET,C.H.ARROWSMITH,A.M.EDWARDS,AUTH 3 C.BOUNTRA,J.WEIGELT,H.PARKTITL CRYSTAL STRUCTURE OF PLEXIN A2 RBD IN COMPLEX WITH RND1REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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4E90.B | PDE9A

General Structure Information 4e90 PDE9A human phosphodiesterase 9 in complex with inhibitors 2.5Å AUTH M.M.CLAFFEY,C.J.HELAL,P.R.VERHOEST,Z.KANG,K.S.FORS,S.JUNG,AUTH 2 J.ZHONG,M.W.BUNDESMANN,X.HOU,S.LUI,R.J.KLEIMAN,AUTH 3 M.VANASE-FRAWLEY,A.W.SCHMIDT,F.MENNITI,C.J.SCHMIDT,AUTH 4 W.E.HOFFMAN,M.HAJOS,L.MCDOWELL,R.E.OCONNOR,AUTH 5 M.MACDOUGALL-MURPHY,K.R.FONSECA,S.L.BECKER,F.R.NELSON,AUTH 6 S.LIRASTITL APPLICATION OF STRUCTURE-BASED DRUG DESIGN AND PARALLELTITL 2 CHEMISTRY TO IDENTIFY SELECTIVE, BRAIN PENETRANT, IN VIVOTITL 3 ACTIVE PHOSPHODIESTERASE 9A INHIBITORS.REF J.MED.CHEM. V. 55 9055 2012REFN ISSN 0022-2623PMID 23025719DOI 10.1021/JM3009635 […]

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