2M20.A | EGFR

General Structure Information 2m20 EGFR egfr transmembrane – juxtamembrane (tm-jm) segment in bicelles: md guided nmr refined structure. -1.0Å AUTH N.F.ENDRES,R.DAS,A.W.SMITH,A.ARKHIPOV,E.KOVACS,Y.HUANG,AUTH 2 J.G.PELTON,Y.SHAN,D.E.SHAW,D.E.WEMMER,J.T.GROVES,J.KURIYANTITL CONFORMATIONAL COUPLING ACROSS THE PLASMA MEMBRANE INTITL 2 ACTIVATION OF THE EGF RECEPTOR.REF CELL(CAMBRIDGE,MASS.) V. 152 543 2013REFN ISSN 0092-8674PMID 23374349DOI 10.1016/J.CELL.2012.12.032 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

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2HDL.A | CXCL14

General Structure Information 2hdl CXCL14 solution structure of brak/cxcl14 -1.0Å AUTH F.C.PETERSON,J.A.THORPE,A.G.HARDER,B.F.VOLKMAN,AUTH 2 S.R.SCHWARZETITL STRUCTURAL DETERMINANTS INVOLVED IN THE REGULATIONTITL 2 OF CXCL14/BRAK EXPRESSION BY THE 26 S PROTEASOME.REF J.MOL.BIOL. V. 363 813 2006REFN ISSN 0022-2836PMID 16987528DOI 10.1016/J.JMB.2006.08.057 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1R4C.C | CST3

General Structure Information 1r4c CST3 n-truncated human cystatin c; dimeric form with 3d domain swapping 2.18Å AUTH R.JANOWSKI,M.ABRAHAMSON,A.GRUBB,M.JASKOLSKITITL DOMAIN SWAPPING IN N-TRUNCATED HUMAN CYSTATIN C.REF J.MOL.BIOL. V. 341 151 2004REFN ISSN 0022-2836PMID 15312769DOI 10.1016/J.JMB.2004.06.013 Variant Set Distributions Mapped Variants

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3BE1.A | ERBB2

General Structure Information 3be1 ERBB2 dual specific bh1 fab in complex with the extracellular domain of her2/erbb-2 2.9Å AUTH J.BOSTROM,S.F.YU,D.KAN,B.A.APPLETON,C.V.LEE,K.BILLECI,W.MAN,AUTH 2 F.PEALE,S.ROSS,C.WIESMANN,G.FUHTITL VARIANTS OF THE ANTIBODY HERCEPTIN THAT INTERACT WITH HER2TITL 2 AND VEGF AT THE ANTIGEN BINDING SITEREF SCIENCE V. 323 1610 2009REFN ISSN 0036-8075PMID 19299620DOI 10.1126/SCIENCE.1165480 Variant Set Distributions Ripley’s K Analysis Plots […]

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4O0X.A | PAK4

General Structure Information 4o0x PAK4 back pocket flexibility provides group-ii pak selectivity for type 1 kinase inhibitors 2.48Å AUTH S.T.STABEN,J.A.FENG,K.LYLE,M.BELVIN,J.BOGGS,J.D.BURCH,AUTH 2 C.C.CHUA,H.CUI,A.G.DIPASQUALE,L.S.FRIEDMAN,C.HEISE,AUTH 3 H.KOEPPEN,A.KOTEY,R.MINTZER,A.OH,D.A.ROBERTS,L.ROUGE,AUTH 4 J.RUDOLPH,C.TAM,W.WANG,Y.XIAO,A.YOUNG,Y.ZHANG,K.P.HOEFLICHTITL BACK POCKET FLEXIBILITY PROVIDES GROUP II P21-ACTIVATEDTITL 2 KINASE (PAK) SELECTIVITY FOR TYPE I 1/2 KINASE INHIBITORS.REF J.MED.CHEM. V. 57 1033 2014REFN ISSN 0022-2623PMID 24432870DOI 10.1021/JM401768T Variant Set Distributions […]

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1W4R.G | TK1

General Structure Information 1w4r TK1 structure of a type ii thymidine kinase with bound dttp 1.83Å AUTH M.S.BIRRINGER,M.T.CLAUS,G.FOLKERS,D.P.KLOER,G.E.SCHULZ,AUTH 2 L.SCAPOZZATITL STRUCTURE OF A TYPE II THYMIDINE KINASE WITH BOUND DTTPREF FEBS LETT. V. 579 1376 2005REFN ISSN 0014-5793PMID 15733844DOI 10.1016/J.FEBSLET.2005.01.034 Variant Set Distributions Mapped Variants

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1XDM.D | ALDOB

General Structure Information 1xdm ALDOB structure of human aldolase b associated with hereditary fructose intolerance (a149p), at 291k 3.0Å AUTH A.D.MALAY,K.N.ALLEN,D.R.TOLANTITL STRUCTURE OF THE THERMOLABILE MUTANT ALDOLASE B,TITL 2 A149P: MOLECULAR BASIS OF HEREDITARY FRUCTOSETITL 3 INTOLERANCE.REF J.MOL.BIOL. V. 347 135 2005REFN ISSN 0022-2836PMID 15733923DOI 10.1016/J.JMB.2005.01.008 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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1LHW.A | SHBG

General Structure Information 1lhw SHBG crystal structure of the n-terminal lg-domain of shbg in complex with 2-methoxyestradiol 1.75Å AUTH G.V.AVVAKUMOV,I.GRISHKOVSKAYA,Y.A.MULLER,AUTH 2 G.L.HAMMONDTITL CRYSTAL STRUCTURE OF HUMAN SEX HORMONE-BINDINGTITL 2 GLOBULIN IN COMPLEX WITH 2-METHOXYESTRADIOLTITL 3 REVEALS THE MOLECULAR BASIS FOR HIGH AFFINITYTITL 4 INTERACTIONS WITH C-2 DERIVATIVES OF ESTRADIOL.REF J.BIOL.CHEM. V. 277 45219 2002REFN ISSN […]

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1MFV.A | AMY1B

General Structure Information 1mfv AMY1B probing the role of a mobile loop in human slaivary amylase: structural studies on the loop-deleted enzyme 2.0Å AUTH N.RAMASUBBU,C.RAGUNATH,P.J.MISHRATITL PROBING THE ROLE OF A MOBILE LOOP IN SUBSTRATETITL 2 BINDING AND ENZYME ACTIVITY OF HUMAN SALIVARYTITL 3 AMYLASE.REF J.MOL.BIOL. V. 325 1061 2003REFN ISSN 0022-2836PMID 12527308DOI 10.1016/S0022-2836(02)01326-8 Variant Set […]

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1MFV.A | AMY1C

General Structure Information 1mfv AMY1C probing the role of a mobile loop in human slaivary amylase: structural studies on the loop-deleted enzyme 2.0Å AUTH N.RAMASUBBU,C.RAGUNATH,P.J.MISHRATITL PROBING THE ROLE OF A MOBILE LOOP IN SUBSTRATETITL 2 BINDING AND ENZYME ACTIVITY OF HUMAN SALIVARYTITL 3 AMYLASE.REF J.MOL.BIOL. V. 325 1061 2003REFN ISSN 0022-2836PMID 12527308DOI 10.1016/S0022-2836(02)01326-8 Variant Set […]

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