4J1Y.A | C1S

General Structure Information 4j1y C1S the x-ray crystal structure of human complement protease c1s zymogen 2.66Å AUTH A.J.PERRY,L.C.WIJEYEWICKREMA,P.G.WILMANN,M.J.GUNZBURG,AUTH 2 L.DANDREA,J.A.IRVING,S.S.PANG,R.C.DUNCAN,J.A.WILCE,AUTH 3 J.C.WHISSTOCK,R.N.PIKETITL A MOLECULAR SWITCH GOVERNS THE INTERACTION BETWEEN THE HUMANTITL 2 COMPLEMENT PROTEASE C1S AND ITS SUBSTRATE, COMPLEMENT C4.REF J.BIOL.CHEM. V. 288 15821 2013REFN ISSN 0021-9258PMID 23592783DOI 10.1074/JBC.M113.464545 Variant Set Distributions Ripley’s K Analysis […]

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3VI4.A | ITGA5

General Structure Information 3vi4 ITGA5 crystal structure of alpha5beta1 integrin headpiece in complex with rgd peptide 2.9Å AUTH M.NAGAE,S.RE,E.MIHARA,T.NOGI,Y.SUGITA,J.TAKAGITITL CRYSTAL STRUCTURE OF ALPHA5BETA1 INTEGRIN ECTODOMAIN: ATOMICTITL 2 DETAILS OF THE FIBRONECTIN RECEPTORREF J.CELL BIOL. V. 197 131 2012REFN ISSN 0021-9525PMID 22451694DOI 10.1083/JCB.201111077 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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2PIP.L | AR

General Structure Information 2pip AR androgen receptor lbd with small molecule 1.8Å AUTH E.ESTEBANEZ-PERPINA,L.A.ARNOLD,A.A.ARNOLD,P.NGUYEN,AUTH 2 E.D.RODRIGUES,E.MAR,R.BATEMAN,P.PALLAI,K.M.SHOKAT,AUTH 3 J.D.BAXTER,R.K.GUY,P.WEBB,R.J.FLETTERICKTITL A SURFACE ON THE ANDROGEN RECEPTOR THATTITL 2 ALLOSTERICALLY REGULATES COACTIVATOR BINDING.REF PROC.NATL.ACAD.SCI.USA V. 104 16074 2007REFN ISSN 0027-8424PMID 17911242DOI 10.1073/PNAS.0708036104 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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2H4M.D | HNRNPA1

General Structure Information 2h4m HNRNPA1 karyopherin beta2/transportin-m9nls 3.05Å AUTH B.J.LEE,A.E.CANSIZOGLU,T.H.LOUIS,Z.ZHANG,Y.M.CHOOKTITL RULES FOR NUCLEAR LOCALIZATION SEQUENCETITL 2 RECOGNITION BY KARYOPHERIN BETA 2.REF CELL(CAMBRIDGE,MASS.) V. 126 543 2006REFN ISSN 0092-8674PMID 16901787DOI 10.1016/J.CELL.2006.05.049 Variant Set Distributions Pathogenic Proximity Analysis Mapped Variants

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2E9W.A | KIT

General Structure Information 2e9w KIT crystal structure of the extracellular domain of kit in complex with stem cell factor (scf) 3.5Å AUTH S.YUZAWA,Y.OPATOWSKY,Z.ZHANG,V.MANDIYAN,I.LAX,J.SCHLESSINGERTITL STRUCTURAL BASIS FOR ACTIVATION OF THE RECEPTOR TYROSINETITL 2 KINASE KIT BY STEM CELL FACTORREF CELL(CAMBRIDGE,MASS.) V. 130 323 2007REFN ISSN 0092-8674PMID 17662946DOI 10.1016/J.CELL.2007.05.055 Variant Set Distributions Ripley’s K Analysis Plots Variant […]

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1NQ0.A | THRB

General Structure Information 1nq0 THRB tr receptor mutations conferring hormone resistance and reduced corepressor release exhibit decreased stability in the nterminal lbd 2.4Å AUTH B.R.HUBER,M.DESCLOZEAUX,B.L.WEST,S.T.CUNHA-LIMA,H.T.NGUYEN,AUTH 2 J.D.BAXTER,H.A.INGRAHAM,R.J.FLETTERICKTITL THYROID HORMONE RECEPTOR-BETA MUTATIONS CONFERRING HORMONETITL 2 RESISTANCE AND REDUCED COREPRESSOR RELEASE EXHIBIT DECREASEDTITL 3 STABILITY IN THE N-TERMINAL LIGAND-BINDING DOMAINREF MOL.ENDOCRINOL. V. 17 107 2003REFN ISSN 0888-8809PMID […]

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3UJR.A | ENO2

General Structure Information 3ujr ENO2 asymmetric complex of human neuron specific enolase-5-pga/pep 1.4Å AUTH J.QIN,G.CHAI,J.M.BREWER,L.L.LOVELACE,L.LEBIODATITL STRUCTURES OF ASYMMETRIC COMPLEXES OF HUMAN NEURON SPECIFICTITL 2 ENOLASE WITH RESOLVED SUBSTRATE AND PRODUCT AND AN ANALOGOUSTITL 3 COMPLEX WITH TWO INHIBITORS INDICATE SUBUNIT INTERACTION ANDTITL 4 INHIBITOR COOPERATIVITY.REF J.INORG.BIOCHEM. V. 111 187 2012REFN ISSN 0162-0134PMID 22437160DOI 10.1016/J.JINORGBIO.2012.02.011 Variant […]

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1L5S.A | PYGL

General Structure Information 1l5s PYGL human liver glycogen phosphorylase complexed with uric acid, n-acetyl- beta-d-glucopyranosylamine, and cp-403,700 2.1Å AUTH J.L.EKSTROM,T.A.PAULY,M.D.CARTY,W.C.SOELLER,J.CULP,AUTH 2 D.E.DANLEY,D.J.HOOVER,J.L.TREADWAY,E.M.GIBBS,R.J.FLETTERICK,AUTH 3 Y.S.DAY,D.G.MYSZKA,V.L.RATHTITL STRUCTURE-ACTIVITY ANALYSIS OF THE PURINE BINDING SITE OFTITL 2 HUMAN LIVER GLYCOGEN PHOSPHORYLASE.REF CHEM.BIOL. V. 9 915 2002REFN ISSN 1074-5521PMID 12204691DOI 10.1016/S1074-5521(02)00186-2 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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3FCS.C | ITGA2B

General Structure Information 3fcs ITGA2B structure of complete ectodomain of integrin aiibb3 2.55Å AUTH J.ZHU,B.H.LUO,T.XIAO,C.ZHANG,N.NISHIDA,T.A.SPRINGERTITL STRUCTURE OF A COMPLETE INTEGRIN ECTODOMAIN IN A PHYSIOLOGICTITL 2 RESTING STATE AND ACTIVATION AND DEACTIVATION BY APPLIEDTITL 3 FORCES.REF MOL.CELL V. 32 849 2008REFN ISSN 1097-2765PMID 19111664DOI 10.1016/J.MOLCEL.2008.11.018 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped […]

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1ZXN.B | TOP2A

General Structure Information 1zxn TOP2A human dna topoisomerase iia atpase/adp 2.51Å AUTH H.WEI,A.J.RUTHENBURG,S.K.BECHIS,G.L.VERDINETITL NUCLEOTIDE-DEPENDENT DOMAIN MOVEMENT IN THE ATPASE DOMAIN OFTITL 2 A HUMAN TYPE IIA DNA TOPOISOMERASE.REF J.BIOL.CHEM. V. 280 37041 2005REFN ISSN 0021-9258PMID 16100112DOI 10.1074/JBC.M506520200 Variant Set Distributions Mapped Variants

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