3GT8.C | EGFR

General Structure Information 3gt8 EGFR crystal structure of the inactive egfr kinase domain in complex with amp-pnp 2.96Å AUTH N.JURA,N.F.ENDRES,K.ENGEL,S.DEINDL,R.DAS,AUTH 2 M.H.LAMERS,D.E.WEMMER,X.ZHANG,J.KURIYANTITL MECHANISM FOR ACTIVATION OF THE EGF RECEPTORTITL 2 CATALYTIC DOMAIN BY THE JUXTAMEMBRANE SEGMENT.REF CELL(CAMBRIDGE,MASS.) V. 137 1293 2009REFN ISSN 0092-8674PMID 19563760DOI 10.1016/J.CELL.2009.04.025 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

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1WIO.B | CD4

General Structure Information 1wio CD4 structure of t-cell surface glycoprotein cd4, tetragonal crystal form 3.9Å AUTH H.WU,P.D.KWONG,W.A.HENDRICKSONTITL DIMERIC ASSOCIATION AND SEGMENTAL VARIABILITY IN THETITL 2 STRUCTURE OF HUMAN CD4.REF NATURE V. 387 527 1997REFN ISSN 0028-0836PMID 9168119DOI 10.1038/387527A0 Variant Set Distributions Mapped Variants

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1BZK.A | SLC4A1

General Structure Information 1bzk SLC4A1 structural studies on the effects of the deletion in the red cell anion exchanger (band3, ae1) associated with south east asian ovalocytosis. -1.0Å AUTH E.J.CHAMBERS,G.B.BLOOMBERG,S.M.RING,M.J.TANNERTITL STRUCTURAL STUDIES ON THE EFFECTS OF THE DELETIONTITL 2 IN THE RED CELL ANION EXCHANGER (BAND 3, AE1)TITL 3 ASSOCIATED WITH SOUTH EAST ASIAN OVALOCYTOSIS.REF […]

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3T2N.A | HPN

General Structure Information 3t2n HPN human hepsin protease in complex with the fab fragment of an inhibitory antibody 2.55Å AUTH T.KOSCHUBS,S.DENGL,H.DURR,K.KALUZA,G.GEORGES,C.HARTL,AUTH 2 S.JENNEWEIN,M.LANZENDORFER,J.AUER,A.STERN,K.S.HUANG,AUTH 3 K.PACKMAN,U.GUBLER,D.KOSTREWA,S.RIES,S.HANSEN,U.KOHNERT,AUTH 4 P.CRAMER,O.MUNDIGLTITL ALLOSTERIC ANTIBODY INHIBITION OF HUMAN HEPSIN PROTEASE.REF BIOCHEM.J. V. 442 483 2012REFN ISSN 0264-6021PMID 22132769DOI 10.1042/BJ20111317 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity […]

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2KNC.B | ITGB3

General Structure Information 2knc ITGB3 platelet integrin alfaiib-beta3 transmembrane-cytoplasmic heterocomplex -1.0Å AUTH J.YANG,Y.Q.MA,R.C.PAGE,S.MISRA,E.F.PLOW,J.QINTITL STRUCTURE OF AN INTEGRIN ALPHAIIB BETA3TITL 2 TRANSMEMBRANE-CYTOPLASMIC HETEROCOMPLEX PROVIDES INSIGHTTITL 3 INTO INTEGRIN ACTIVATION.REF PROC.NATL.ACAD.SCI.USA V. 106 17729 2009REFN ISSN 0027-8424PMID 19805198DOI 10.1073/PNAS.0909589106 Variant Set Distributions Pathogenic Proximity Analysis Mapped Variants

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3CCZ.B | HMGCR

General Structure Information 3ccz HMGCR thermodynamic and structure guided design of statin hmg-coa reductase inhibitors 1.7Å AUTH R.W.SARVER,E.BILLS,G.BOLTON,L.D.BRATTON,AUTH 2 N.L.CASPERS,J.B.DUNBAR,M.S.HARRIS,R.H.HUTCHINGS,AUTH 3 R.M.KENNEDY,S.D.LARSEN,A.PAVLOVSKY,J.A.PFEFFERKORN,AUTH 4 G.BAINBRIDGETITL THERMODYNAMIC AND STRUCTURE GUIDED DESIGN OFTITL 2 STATIN BASED INHIBITORS OFTITL 3 3-HYDROXY-3-METHYLGLUTARYL COENZYME A REDUCTASE.REF J.MED.CHEM. V. 51 3804 2008REFN ISSN 0022-2623PMID 18540668DOI 10.1021/JM7015057 Variant Set Distributions Mapped Variants

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2V5P.C | IGF2

General Structure Information 2v5p IGF2 complex structure of human igf2r domains 11-13 bound to igf-ii 4.1Å AUTH J.BROWN,C.DELAINE,O.J.ZACCHEO,C.SIEBOLD,AUTH 2 R.J.GILBERT,G.VAN BOXEL,A.DENLEY,J.C.WALLACE,AUTH 3 A.B.HASSAN,B.E.FORBES,E.Y.JONESTITL STRUCTURE AND FUNCTIONAL ANALYSIS OF THETITL 2 IGF-II/IGF2R INTERACTIONREF EMBO J. V. 27 265 2008REFN ISSN 0261-4189PMID 18046459DOI 10.1038/SJ.EMBOJ.7601938 Variant Set Distributions Mapped Variants

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2M20.A | EGFR

General Structure Information 2m20 EGFR egfr transmembrane – juxtamembrane (tm-jm) segment in bicelles: md guided nmr refined structure. -1.0Å AUTH N.F.ENDRES,R.DAS,A.W.SMITH,A.ARKHIPOV,E.KOVACS,Y.HUANG,AUTH 2 J.G.PELTON,Y.SHAN,D.E.SHAW,D.E.WEMMER,J.T.GROVES,J.KURIYANTITL CONFORMATIONAL COUPLING ACROSS THE PLASMA MEMBRANE INTITL 2 ACTIVATION OF THE EGF RECEPTOR.REF CELL(CAMBRIDGE,MASS.) V. 152 543 2013REFN ISSN 0092-8674PMID 23374349DOI 10.1016/J.CELL.2012.12.032 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

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3BE1.A | ERBB2

General Structure Information 3be1 ERBB2 dual specific bh1 fab in complex with the extracellular domain of her2/erbb-2 2.9Å AUTH J.BOSTROM,S.F.YU,D.KAN,B.A.APPLETON,C.V.LEE,K.BILLECI,W.MAN,AUTH 2 F.PEALE,S.ROSS,C.WIESMANN,G.FUHTITL VARIANTS OF THE ANTIBODY HERCEPTIN THAT INTERACT WITH HER2TITL 2 AND VEGF AT THE ANTIGEN BINDING SITEREF SCIENCE V. 323 1610 2009REFN ISSN 0036-8075PMID 19299620DOI 10.1126/SCIENCE.1165480 Variant Set Distributions Ripley’s K Analysis Plots […]

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3IKK.A | VAPB

General Structure Information 3ikk VAPB crystal structure analysis of msp domain 2.5Å AUTH J.SHI,S.LUA,J.S.TONG,J.SONGTITL ELIMINATION OF THE NATIVE STRUCTURE AND SOLUBILITY OF THETITL 2 HVAPB MSP DOMAIN BY THE PRO56SER MUTATION THAT CAUSESTITL 3 AMYOTROPHIC LATERAL SCLEROSIS.REF BIOCHEMISTRY V. 49 3887 2010REFN ISSN 0006-2960PMID 20377183DOI 10.1021/BI902057A Variant Set Distributions Mapped Variants

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