3CCZ.B | HMGCR

General Structure Information

PDB ID 3ccz
HGNC Gene Label(s) HMGCR
Structure Name thermodynamic and structure guided design of statin hmg-coa reductase inhibitors
Resolution 1.7Å
Reference AUTH R.W.SARVER,E.BILLS,G.BOLTON,L.D.BRATTON,AUTH 2 N.L.CASPERS,J.B.DUNBAR,M.S.HARRIS,R.H.HUTCHINGS,AUTH 3 R.M.KENNEDY,S.D.LARSEN,A.PAVLOVSKY,J.A.PFEFFERKORN,AUTH 4 G.BAINBRIDGETITL THERMODYNAMIC AND STRUCTURE GUIDED DESIGN OFTITL 2 STATIN BASED INHIBITORS OFTITL 3 3-HYDROXY-3-METHYLGLUTARYL COENZYME A REDUCTASE.REF J.MED.CHEM. V. 51 3804 2008REFN ISSN 0022-2623PMID 18540668DOI 10.1021/JM7015057

Variant Set Distributions

ExAC Variants

Number Of Residues 405
Number Of SNVs 49
Number Of Permutations 44446
Optimal Distance Threshold 16.0
K Statistic 0.127
p-value 0.793

Mapped Variants

[+] ExAC Missense Variants