2CCI.B | CCNA2

General Structure Information 2cci CCNA2 crystal structure of phospho-cdk2 cyclin a in complex with a peptide containing both the substrate and recruitment sites of cdc6 2.7Å AUTH K.Y.CHENG,M.E.M.NOBLE,V.SKAMNAKI,N.R.BROWN,E.D.LOWE,AUTH 2 L.KONTOGIANNIS,K.SHEN,P.A.COLE,G.SILIGARDI,L.N.JOHNSONTITL THE ROLE OF THE PHOSPHO-CDK2/CYCLIN A RECRUITMENT SITE INTITL 2 SUBSTRATE RECOGNITIONREF J.BIOL.CHEM. V. 281 23167 2006REFN ISSN 0021-9258PMID 16707497DOI 10.1074/JBC.M600480200 Variant Set Distributions Mapped […]

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4ELJ.A | RB1

General Structure Information 4elj RB1 crystal structure of the inactive retinoblastoma protein phosphorylated at t373 2.7Å AUTH J.R.BURKE,G.L.HURA,S.M.RUBINTITL STRUCTURES OF INACTIVE RETINOBLASTOMA PROTEIN REVEALTITL 2 MULTIPLE MECHANISMS FOR CELL CYCLE CONTROL.REF GENES DEV. V. 26 1156 2012REFN ISSN 0890-9369PMID 22569856DOI 10.1101/GAD.189837.112 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped […]

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2AZE.C | RB1

General Structure Information 2aze RB1 structure of the rb c-terminal domain bound to an e2f1-dp1 heterodimer 2.55Å AUTH S.M.RUBIN,A.L.GALL,N.ZHENG,N.P.PAVLETICHTITL STRUCTURE OF THE RB C-TERMINAL DOMAIN BOUND TOTITL 2 E2F1-DP1: A MECHANISM FOR PHOSPHORYLATION-INDUCEDTITL 3 E2F RELEASE.REF CELL(CAMBRIDGE,MASS.) V. 123 1093 2005REFN ISSN 0092-8674PMID 16360038DOI 10.1016/J.CELL.2005.09.044 Variant Set Distributions Mapped Variants

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3E04.C | FH

General Structure Information 3e04 FH crystal structure of human fumarate hydratase 1.95Å AUTH K.L.KAVANAGH,S.PICAUD,E.S.PILKA,W.W.YUE,A.K.ROOS,AUTH 2 P.FILIPPAKOPOULOS,F.VON DELFT,C.H.ARROWSMITH,M.WIKSTROM,AUTH 3 A.M.EDWARDS,C.BOUNTRA,U.OPPERMANN,AUTH 4 STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL CRYSTAL STRUCTURE OF HUMAN FUMARATE HYDRATASEREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3GT8.C | EGFR

General Structure Information 3gt8 EGFR crystal structure of the inactive egfr kinase domain in complex with amp-pnp 2.96Å AUTH N.JURA,N.F.ENDRES,K.ENGEL,S.DEINDL,R.DAS,AUTH 2 M.H.LAMERS,D.E.WEMMER,X.ZHANG,J.KURIYANTITL MECHANISM FOR ACTIVATION OF THE EGF RECEPTORTITL 2 CATALYTIC DOMAIN BY THE JUXTAMEMBRANE SEGMENT.REF CELL(CAMBRIDGE,MASS.) V. 137 1293 2009REFN ISSN 0092-8674PMID 19563760DOI 10.1016/J.CELL.2009.04.025 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

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2P5X.A | ASMTL

General Structure Information 2p5x ASMTL crystal structure of maf domain of human n-acetylserotonin o- methyltransferase-like protein 2.0Å AUTH A.TCHIGVINTSEV,D.TCHIGVINTSEV,R.FLICK,A.POPOVIC,A.DONG,X.XU,AUTH 2 G.BROWN,W.LU,H.WU,H.CUI,L.DOMBROWSKI,J.C.JOO,N.BELOGLAZOVA,AUTH 3 J.MIN,A.SAVCHENKO,A.A.CAUDY,J.D.RABINOWITZ,A.G.MURZIN,AUTH 4 A.F.YAKUNINTITL BIOCHEMICAL AND STRUCTURAL STUDIES OF CONSERVED MAF PROTEINSTITL 2 REVEALED NUCLEOTIDE PYROPHOSPHATASES WITH A PREFERENCE FORTITL 3 MODIFIED NUCLEOTIDES.REF CHEM.BIOL. V. 20 1386 2013REFN ISSN 1074-5521PMID 24210219DOI 10.1016/J.CHEMBIOL.2013.09.011 Variant Set […]

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3RCD.A | ERBB2

General Structure Information 3rcd ERBB2 her2 kinase domain complexed with tak-285 3.21Å AUTH T.ISHIKAWA,M.SETO,H.BANNO,Y.KAWAKITA,M.OORUI,T.TANIGUCHI,AUTH 2 Y.OHTA,T.TAMURA,A.NAKAYAMA,H.MIKI,H.KAMIGUCHI,T.TANAKA,AUTH 3 N.HABUKA,S.SOGABE,J.YANO,K.AERTGEERTS,K.KAMIYAMATITL DESIGN AND SYNTHESIS OF NOVEL HUMAN EPIDERMAL GROWTH FACTORTITL 2 RECEPTOR 2 (HER2)/EPIDERMAL GROWTH FACTOR RECEPTOR (EGFR)TITL 3 DUAL INHIBITORS BEARING A PYRROLO[3,2-D]PYRIMIDINE SCAFFOLD.REF J.MED.CHEM. V. 54 8030 2011REFN ISSN 0022-2623PMID 22003817DOI 10.1021/JM2008634 Variant Set Distributions Ripley’s […]

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2D68.A | FGFR1OP

General Structure Information 2d68 FGFR1OP structure of the n-terminal domain of fop (fgfr1op) protein 1.6Å AUTH A.MIKOLAJKA,X.YAN,G.M.POPOWICZ,P.SMIALOWSKI,AUTH 2 E.A.NIGG,T.A.HOLAKTITL STRUCTURE OF THE N-TERMINAL DOMAIN OF THE FOPTITL 2 (FGFR1OP) PROTEIN AND IMPLICATIONS FOR ITSTITL 3 DIMERIZATION AND CENTROSOMAL LOCALIZATION.REF J.MOL.BIOL. V. 359 863 2006REFN ISSN 0022-2836PMID 16690081DOI 10.1016/J.JMB.2006.03.070 Variant Set Distributions Mapped Variants

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3I6W.H | CHEK2

General Structure Information 3i6w CHEK2 structure and activation mechanism of the chk2 dna-damage checkpoint kinase 3.25Å AUTH Z.CAI,N.H.CHEHAB,N.P.PAVLETICHTITL STRUCTURE AND ACTIVATION MECHANISM OF THE CHK2 DNA DAMAGETITL 2 CHECKPOINT KINASE.REF MOL.CELL V. 35 818 2009REFN ISSN 1097-2765PMID 19782031DOI 10.1016/J.MOLCEL.2009.09.007 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3SI5.B | BUB1B

General Structure Information 3si5 BUB1B kinetochore-bubr1 kinase complex 2.2Å AUTH V.M.BOLANOS-GARCIA,T.LISCHETTI,D.MATAK-VINKOVIC,E.COTA,AUTH 2 P.J.SIMPSON,D.Y.CHIRGADZE,D.R.SPRING,C.V.ROBINSON,J.NILSSON,AUTH 3 T.L.BLUNDELLTITL STRUCTURE OF A BLINKIN-BUBR1 COMPLEX REVEALS AN INTERACTIONTITL 2 CRUCIAL FOR KINETOCHORE-MITOTIC CHECKPOINT REGULATION VIA ANTITL 3 UNANTICIPATED BINDING SITE.REF STRUCTURE V. 19 1691 2011REFN ISSN 0969-2126PMID 22000412DOI 10.1016/J.STR.2011.09.017 Variant Set Distributions Mapped Variants

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