2LWI.A | HRAS

General Structure Information 2lwi HRAS solution structure of h-rast35s mutant protein in complex with kobe2601 -1.0Å AUTH F.SHIMA,Y.YOSHIKAWA,M.YE,M.ARAKI,S.MATSUMOTO,J.LIAO,L.HU,AUTH 2 T.SUGIMOTO,Y.IJIRI,A.TAKEDA,Y.NISHIYAMA,C.SATO,S.MURAOKA,AUTH 3 A.TAMURA,T.OSODA,K.I.TSUDA,T.MIYAKAWA,H.FUKUNISHI,J.SHIMADA,AUTH 4 T.KUMASAKA,M.YAMAMOTO,T.KATAOKATITL IN SILICO DISCOVERY OF SMALL-MOLECULE RAS INHIBITORS THATTITL 2 DISPLAY ANTITUMOR ACTIVITY BY BLOCKING THE RAS-EFFECTORTITL 3 INTERACTION.REF PROC.NATL.ACAD.SCI.USA 2013REFN ESSN 1091-6490PMID 23630290DOI 10.1073/PNAS.1217730110 Variant Set Distributions Ripley’s K Analysis Plots […]

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4MZR.B | TP53

General Structure Information 4mzr TP53 crystal structure of a polypeptide p53 mutant bound to dna 2.9Å AUTH S.EMAMZADAH,L.TROPIA,I.VINCENTI,B.FALQUET,T.D.HALAZONETISTITL REVERSAL OF THE DNA-BINDING-INDUCED LOOP L1 CONFORMATIONALTITL 2 SWITCH IN AN ENGINEERED HUMAN P53 PROTEIN.REF J.MOL.BIOL. V. 426 936 2014REFN ISSN 0022-2836PMID 24374182DOI 10.1016/J.JMB.2013.12.020 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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1ZNQ.O | GAPDH

General Structure Information 1znq GAPDH crsytal structure of human liver gapdh 2.5Å AUTH S.A.ISMAIL,H.W.PARKTITL CRYSTAL STRUCTURE ANALYSIS OF HUMAN LIVER GAPDHREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2J3T.B | TRAPPC6A

General Structure Information 2j3t TRAPPC6A the crystal structure of the bet3-trs33-bet5-trs23 complex. 2.4Å AUTH Y.KIM,S.RAUNSER,C.MUNGER,J.WAGNER,Y.SONG,M.CYGLER,T.WALZ,AUTH 2 B.OH,M.SACHERTITL THE ARCHITECTURE OF THE MULTISUBUNIT TRAPP I COMPLEXTITL 2 SUGGESTS A MODEL FOR VESICLE TETHERING.REF CELL(CAMBRIDGE,MASS.) V. 127 817 2006REFN ISSN 0092-8674PMID 17110339DOI 10.1016/J.CELL.2006.09.029 Variant Set Distributions Mapped Variants

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3S2K.C | DKK1

General Structure Information 3s2k DKK1 structural basis of wnt signaling inhibition by dickkopf binding to lrp5/6. 2.8Å AUTH V.E.AHN,M.L.CHU,H.J.CHOI,D.TRAN,A.ABO,W.I.WEISTITL STRUCTURAL BASIS OF WNT SIGNALING INHIBITION BY DICKKOPFTITL 2 BINDING TO LRP5/6.REF DEV.CELL V. 21 862 2011REFN ISSN 1534-5807PMID 22000856DOI 10.1016/J.DEVCEL.2011.09.003 Variant Set Distributions Mapped Variants

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3S2K.A | LRP6

General Structure Information 3s2k LRP6 structural basis of wnt signaling inhibition by dickkopf binding to lrp5/6. 2.8Å AUTH V.E.AHN,M.L.CHU,H.J.CHOI,D.TRAN,A.ABO,W.I.WEISTITL STRUCTURAL BASIS OF WNT SIGNALING INHIBITION BY DICKKOPFTITL 2 BINDING TO LRP5/6.REF DEV.CELL V. 21 862 2011REFN ISSN 1534-5807PMID 22000856DOI 10.1016/J.DEVCEL.2011.09.003 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2YTV.A | CSDE1

General Structure Information 2ytv CSDE1 solution structure of the fifth cold-shock domain of the human kiaa0885 protein (unr protein) -1.0Å AUTH A.K.GORONCY,S.KOSHIBA,N.TOCHIO,T.TOMIZAWA,M.INOUE,AUTH 2 S.WATANABE,T.HARADA,A.TANAKA,O.OHARA,T.KIGAWA,S.YOKOYAMATITL THE NMR SOLUTION STRUCTURES OF THE FIVE CONSTITUENTTITL 2 COLD-SHOCK DOMAINS (CSD) OF THE HUMAN UNR (UPSTREAM OFTITL 3 N-RAS) PROTEIN.REF J.STRUCT.FUNCT.GENOM. V. 11 181 2010REFN ISSN 1345-711XPMID 20213426DOI 10.1007/S10969-010-9081-Z Variant […]

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2GQM.A | SCO1

General Structure Information 2gqm SCO1 solution structure of human cu(i)-sco1 -1.0Å AUTH L.BANCI,I.BERTINI,V.CALDERONE,S.CIOFI-BAFFONI,AUTH 2 S.MANGANI,M.MARTINELLI,P.PALUMAA,S.WANGTITL A HINT FOR THE FUNCTION OF HUMAN SCO1 FROMTITL 2 DIFFERENT STRUCTURES.REF PROC.NATL.ACAD.SCI.USA V. 103 8595 2006REFN ISSN 0027-8424PMID 16735468DOI 10.1073/PNAS.0601375103 Variant Set Distributions Mapped Variants

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2XAH.A | KDM1A

General Structure Information 2xah KDM1A crystal structure of lsd1-corest in complex with (+)- trans-2-phenylcyclopropyl-1-amine 3.1Å AUTH C.BINDA,S.VALENTE,M.ROMANENGHI,S.PILOTTO,R.CIRILLI,AUTH 2 A.KARYTINOS,G.CIOSSANI,O.A.BOTRUGNO,F.FORNERIS,AUTH 3 M.TARDUGNO,D.E.EDMONDSON,S.MINUCCI,A.MATTEVI,A.MAITITL BIOCHEMICAL, STRUCTURAL, AND BIOLOGICAL EVALUATIONTITL 2 OF TRANYLCYPROMINE DERIVATIVES AS INHIBITORS OFTITL 3 HISTONE DEMETHYLASES LSD1 AND LSD2.REF J.AM.CHEM.SOC. V. 132 6827 2010REFN ISSN 0002-7863PMID 20415477DOI 10.1021/JA101557K Variant Set Distributions Ripley’s K Analysis Plots […]

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3UO9.D | GLS

General Structure Information 3uo9 GLS crystal structure of human gac in complex with glutamate and bptes 2.3Å AUTH B.DELABARRE,S.GROSS,C.FANG,Y.GAO,A.JHA,F.JIANG,J.SONG J,AUTH 2 W.WEI,J.B.HUROVTITL FULL-LENGTH HUMAN GLUTAMINASE IN COMPLEX WITH AN ALLOSTERICTITL 2 INHIBITOR.REF BIOCHEMISTRY V. 50 10764 2011REFN ISSN 0006-2960PMID 22049910DOI 10.1021/BI201613D Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped […]

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