1KIV.A | LPA

General Structure Information 1kiv LPA recombinant kringle iv-10/m66 variant of human apolipoprotein(a) 2.1Å AUTH I.MOCHALKIN,B.CHENG,O.KLEZOVITCH,A.M.SCANU,AUTH 2 A.TULINSKYTITL RECOMBINANT KRINGLE IV-10 MODULES OF HUMANTITL 2 APOLIPOPROTEIN(A): STRUCTURE, LIGAND BINDINGTITL 3 MODES, AND BIOLOGICAL RELEVANCE.REF BIOCHEMISTRY V. 38 1990 1999REFN ISSN 0006-2960PMID 10026282DOI 10.1021/BI9820558 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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1LSL.A | THBS1

General Structure Information 1lsl THBS1 crystal structure of the thrombospondin-1 type 1 repeats 1.9Å AUTH K.TAN,M.DUQUETTE,J.H.LIU,Y.DONG,R.ZHANG,AUTH 2 A.JOACHIMIAK,J.LAWLER,J.H.WANGTITL CRYSTAL STRUCTURE OF THE TSP-1 TYPE 1 REPEATS: ATITL 2 NOVEL LAYERED FOLD AND ITS BIOLOGICAL IMPLICATION.REF J.CELL BIOL. V. 159 373 2002REFN ISSN 0021-9525PMID 12391027DOI 10.1083/JCB.200206062 Variant Set Distributions Mapped Variants

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1GZW.B | LGALS1

General Structure Information 1gzw LGALS1 x-ray crystal structure of human galectin-1 1.7Å AUTH M.I.F.LOPEZ-LUCENDO,D.SOLIS,S.ANDRE,J.HIRABAYASHI,AUTH 2 K.KASAI,H.KALTNER,H.J.GABIUS,A.ROMEROTITL GROWTH-REGULATORY HUMAN GALECTIN-1:TITL 2 CRYSTALLOGRAPHIC CHARACTERISATION OF THETITL 3 STRUCTURAL CHANGES INDUCED BY SINGLE-SITETITL 4 MUTATIONS AND THEIR IMPACT ON THE THERMODYNAMICSTITL 5 OF LIGAND BINDINGREF J.MOL.BIOL. V. 343 957 2004REFN ISSN 0022-2836PMID 15476813DOI 10.1016/J.JMB.2004.08.078 Variant Set Distributions Mapped […]

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3LCO.A | CSF1R

General Structure Information 3lco CSF1R inhibitor bound to a dfg-out structure of the kinase domain of csf-1r 3.4Å AUTH M.J.MEYERS,M.PELC,S.KAMTEKAR,J.DAY,G.I.PODA,M.K.HALL,AUTH 2 M.L.MICHENER,B.A.REITZ,K.J.MATHIS,B.S.PIERCE,M.D.PARIKH,AUTH 3 D.A.MISCHKE,S.A.LONG,J.J.PARLOW,D.R.ANDERSON,A.THORARENSENTITL STRUCTURE-BASED DRUG DESIGN ENABLES CONVERSION OF A DFG-INTITL 2 BINDING CSF-1R KINASE INHIBITOR TO A DFG-OUT BINDING MODE.REF BIOORG.MED.CHEM.LETT. V. 20 1543 2010REFN ISSN 0960-894XPMID 20137931DOI 10.1016/J.BMCL.2010.01.078 Variant Set Distributions Pathogenic […]

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3KQS.B | PNMT

General Structure Information 3kqs PNMT crystal structure of hpnmt in complex adohcy and 2-aminobenzimidazole 2.0Å AUTH N.DRINKWATER,H.VU,K.M.LOVELL,K.R.CRISCIONE,B.M.COLLINS,AUTH 2 T.E.PRISINZANO,S.A.POULSEN,M.J.MCLEISH,G.L.GRUNEWALD,AUTH 3 J.L.MARTINTITL FRAGMENT-BASED SCREENING BY X-RAY CRYSTALLOGRAPHY, MS ANDTITL 2 ISOTHERMAL TITRATION CALORIMETRY TO IDENTIFY PNMTTITL 3 (PHENYLETHANOLAMINE N-METHYLTRANSFERASE) INHIBITORS.REF BIOCHEM.J. V. 431 51 2010REFN ISSN 0264-6021PMID 20642456DOI 10.1042/BJ20100651 Variant Set Distributions Ripley’s K Analysis Plots […]

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1I0E.B | CKM

General Structure Information 1i0e CKM crystal structure of creatine kinase from human muscle 3.5Å AUTH Y.Q.SHEN,L.TANG,H.M.ZHOU,Z.J.LINTITL STRUCTURE OF HUMAN MUSCLE CREATINE KINASE.REF ACTA CRYSTALLOGR.,SECT.D V. 57 1196 2001REFN ISSN 0907-4449PMID 11517911 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2JDF.A | CRYGB

General Structure Information 2jdf CRYGB human gamma-b crystallin 1.7Å AUTH H.EBERSBACH,E.FIEDLER,T.SCHEUERMANN,M.FIEDLER,AUTH 2 M.T.STUBBS,C.REIMANN,G.PROETZEL,R.RUDOLPH,U.FIEDLERTITL AFFILIN-NOVEL BINDING MOLECULES BASED ON HUMANTITL 2 GAMMA-B-CRYSTALLIN, AN ALL BETA-SHEET PROTEIN.REF J.MOL.BIOL. V. 372 172 2007REFN ISSN 0022-2836PMID 17628592DOI 10.1016/J.JMB.2007.06.045 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2NLL.B | THRB

General Structure Information 2nll THRB retinoid x receptor-thyroid hormone receptor dna-binding domain heterodimer bound to thyroid response element dna 1.9Å AUTH F.RASTINEJAD,T.PERLMANN,R.M.EVANS,P.B.SIGLERTITL STRUCTURAL DETERMINANTS OF NUCLEAR RECEPTORTITL 2 ASSEMBLY ON DNA DIRECT REPEATS.REF NATURE V. 375 203 1995REFN ISSN 0028-0836PMID 7746322DOI 10.1038/375203A0 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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1G83.B | FYN

General Structure Information 1g83 FYN crystal structure of fyn sh3-sh2 2.6Å AUTH S.T.AROLD,T.S.ULMER,T.D.MULHERN,J.M.WERNER,AUTH 2 J.E.LADBURY,I.D.CAMPBELL,M.E.NOBLETITL THE ROLE OF THE SRC HOMOLOGY 3-SRC HOMOLOGY 2TITL 2 INTERFACE IN THE REGULATION OF SRC KINASES.REF J.BIOL.CHEM. V. 276 17199 2001REFN ISSN 0021-9258PMID 11278857DOI 10.1074/JBC.M011185200 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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3Q6N.E | HSP90AA1

General Structure Information 3q6n HSP90AA1 crystal structure of human mc-hsp90 in p21 space group 3.05Å AUTH C.C.LEE,T.W.LIN,T.P.KO,A.H.-J.WANGTITL THE HEXAMERIC STRUCTURES OF HUMAN HEAT SHOCK PROTEIN 90REF PLOS ONE V. 6 19961 2011REFN ESSN 1932-6203PMID 21647436DOI 10.1371/JOURNAL.PONE.0019961 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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