4AEL.B | PDE10A

General Structure Information 4ael PDE10A pde10a in complex with the inhibitor az5 2.2Å AUTH U.BAUER,F.GIORDANETTO,M.BAUER,G.OMAHONY,K.E.JOHANSSON,AUTH 2 W.KNECHT,J.HARTLEIB-GESCHWINDNER,E.T.CARLSSON,C.ENROTHTITL DISCOVERY OF 4-HYDROXY-1,6-NAPHTHYRIDINE-3-CARBONITRILETITL 2 DERIVATIVES AS NOVEL PDE10A INHIBITORS.REF BIOORG.MED.CHEM.LETT. V. 22 1944 2012REFN ISSN 0960-894XPMID 22321214DOI 10.1016/J.BMCL.2012.01.046 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3H3S.B | COL4A3BP

General Structure Information 3h3s COL4A3BP crystal structure of the cert start domain in complex with hpa-15 1.66Å AUTH N.KUDO,K.KUMAGAI,R.MATSUBARA,S.KOBAYASHI,K.HANADA,AUTH 2 S.WAKATSUKI,R.KATOTITL CRYSTAL STRUCTURES OF THE CERT START DOMAIN WITHTITL 2 INHIBITORS PROVIDE INSIGHTS INTO THE MECHANISM OFTITL 3 CERAMIDE TRANSFER.REF J.MOL.BIOL. V. 396 245 2010REFN ISSN 0022-2836PMID 20036255DOI 10.1016/J.JMB.2009.12.029 Variant Set Distributions Ripley’s K Analysis […]

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1R4X.A | COPG1

General Structure Information 1r4x COPG1 crystal structure analys of the gamma-copi appendage domain 1.9Å AUTH P.J.WATSON,G.FRIGERIO,B.M.COLLINS,R.DUDEN,D.J.OWENTITL GAMMA-COP APPENDAGE DOMAIN – STRUCTURE AND FUNCTIONREF TRAFFIC V. 5 79 2004REFN ISSN 1398-9219PMID 14690497DOI 10.1111/J.1600-0854.2004.00158.X Variant Set Distributions Mapped Variants

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3NAU.A | ZHX2

General Structure Information 3nau ZHX2 crystal structure of zhx2 hd2 (zinc-fingers and homeoboxes protein 2, homeodomain 2) 2.7Å AUTH L.E.BIRD,J.REN,J.E.NETTLESHIP,G.E.FOLKERS,R.J.OWENS,AUTH 2 D.K.STAMMERSTITL NOVEL STRUCTURAL FEATURES IN TWO ZHX HOMEODOMAINS DERIVEDTITL 2 FROM A SYSTEMATIC STUDY OF SINGLE AND MULTIPLE DOMAINSREF BMC STRUCT.BIOL. V. 10 13 2010REFN ESSN 1472-6807PMID 20509910DOI 10.1186/1472-6807-10-13 Variant Set Distributions Mapped Variants

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3E77.B | PSAT1

General Structure Information 3e77 PSAT1 human phosphoserine aminotransferase in complex with plp 2.5Å AUTH L.LEHTIO,T.KARLBERG,J.ANDERSSON,C.H.ARROWSMITH,H.BERGLUND,AUTH 2 C.BOUNTRA,R.COLLINS,L.G.DAHLGREN,A.M.EDWARDS,S.FLODIN,AUTH 3 A.FLORES,S.GRASLUND,M.HAMMARSTROM,A.JOHANSSON,I.JOHANSSON,AUTH 4 T.KOTENYOVA,M.MOCHE,M.E.NILSSON,P.NORDLUND,T.NYMAN,K.OLESEN,AUTH 5 C.PERSSON,J.SAGEMARK,S.G.THORSELL,L.TRESAUGUES,AUTH 6 S.VAN DEN BERG,M.WELIN,M.WIKSTROM,M.WISNIEWSKA,J.WEIGELT,AUTH 7 H.SCHUELER,STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL HUMAN PHOSPHOSERINE AMINOTRANSFERASE IN COMPLEX WITH PLPREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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2CU1.A | MAP3K2

General Structure Information 2cu1 MAP3K2 solution structure of the pb1 domain of human protein kinase mekk2b -1.0Å AUTH K.INOUE,T.NAGASHIMA,F.HAYASHI,S.YOKOYAMATITL SOLUTION STRUCTURE OF THE PB1 DOMAIN OF HUMANTITL 2 PROTEIN KINASE MEKK2BREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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4CC9.A | VPRBP

General Structure Information 4cc9 VPRBP crystal structure of human samhd1 (amino acid residues 582- 626) bound to vpx isolated from sooty mangabey and human dcaf1 (amino acid residues 1058-1396) 2.47Å AUTH D.SCHWEFEL,H.C.T.GROOM,V.C.BOUCHERIT,E.CHRISTODOULOU,AUTH 2 P.A.WALKER,J.P.STOYE,K.N.BISHOP,I.A.TAYLORTITL STRUCTURAL BASIS OF LENTIVIRAL SUBVERSION OF A CELLULARTITL 2 PROTEIN DEGRADATION PATHWAY.REF NATURE V. 505 234 2014REFN ISSN 0028-0836PMID 24336198DOI 10.1038/NATURE12815 […]

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2NYT.A | APOBEC2

General Structure Information 2nyt APOBEC2 the apobec2 crystal structure and functional implications for aid 2.5Å AUTH C.PROCHNOW,R.BRANSTEITTER,M.G.KLEIN,M.F.GOODMAN,AUTH 2 X.S.CHENTITL THE APOBEC-2 CRYSTAL STRUCTURE AND FUNCTIONALTITL 2 IMPLICATIONS FOR THE DEAMINASE AID.REF NATURE V. 445 447 2007REFN ISSN 0028-0836PMID 17187054DOI 10.1038/NATURE05492 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1X5X.A | FNDC3A

General Structure Information 1x5x FNDC3A solution structure of the fibronectin type-iii domain of human fibronectin type iii domain containing protein 3 -1.0Å AUTH M.YONEYAMA,N.TOCHIO,S.KOSHIBA,M.INOUE,T.KIGAWA,AUTH 2 S.YOKOYAMATITL SOLUTION STRUCTURE OF THE FIBRONECTIN TYPE-IIITITL 2 DOMAIN OF HUMAN FIBRONECTIN TYPE III DOMAINTITL 3 CONTAINING PROTEIN 3REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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3ENP.B | TPRKB

General Structure Information 3enp TPRKB crystal structure of human cgi121 2.48Å AUTH D.Y.MAO,D.NECULAI,M.DOWNEY,S.ORLICKY,Y.Z.HAFFANI,AUTH 2 D.F.CECCARELLI,J.S.HO,R.K.SZILARD,W.ZHANG,C.S.HO,L.WAN,AUTH 3 C.FARES,S.RUMPEL,I.KURINOV,C.H.ARROWSMITH,D.DUROCHER,AUTH 4 F.SICHERITITL ATOMIC STRUCTURE OF THE KEOPS COMPLEX: AN ANCIENT PROTEINTITL 2 KINASE-CONTAINING MOLECULAR MACHINE.REF MOL.CELL V. 32 259 2008REFN ISSN 1097-2765PMID 18951093DOI 10.1016/J.MOLCEL.2008.10.002 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped […]

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