3PS4.C | MAST1

General Structure Information 3ps4 MAST1 pdz domain from human microtubule-associated serine/threonine-protein kinase 1 1.85Å AUTH E.UGOCHUKWU,J.WANG,T.KROJER,J.R.C.MUNIZ,R.SETHI,A.C.W.PIKE,AUTH 2 A.ROOS,E.SALAH,R.COCKING,P.SAVITSKY,D.A.DOYLE,F.VON DELFT,AUTH 3 C.BOUNTRA,C.H.ARROWSMITH,J.WEIGELT,A.EDWARDS,S.KNAPP,AUTH 4 J.M.ELKINS,STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL PDZ DOMAIN FROM HUMAN MICROTUBULE-ASSOCIATEDTITL 2 SERINE/THREONINE-PROTEIN KINASE 1REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2M9X.A | MAST1

General Structure Information 2m9x MAST1 solution nmr structure of microtubule-associated serine/threonine- protein kinase 1 from homo sapiens, northeast structural genomics consortium (nesg) target hr9151a -1.0Å AUTH X.XU,A.ELETSKY,R.SHASTRY,D.LEE,K.HAMILTON,R.XIAO,T.B.ACTON,AUTH 2 J.K.EVERETT,G.T.MONTELIONE,T.SZYPERSKITITL SOLUTION NMR STRUCTURE OF MICROTUBULE-ASSOCIATEDTITL 2 SERINE/THREONINE-PROTEIN KINASE 1 FROM HOMO SAPIENS,TITL 3 NORTHEAST STRUCTURAL GENOMICS CONSORTIUM (NESG) TARGETTITL 4 HR9151AREF TO BE PUBLISHEDREFN Variant Set […]

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3E77.B | PSAT1

General Structure Information 3e77 PSAT1 human phosphoserine aminotransferase in complex with plp 2.5Å AUTH L.LEHTIO,T.KARLBERG,J.ANDERSSON,C.H.ARROWSMITH,H.BERGLUND,AUTH 2 C.BOUNTRA,R.COLLINS,L.G.DAHLGREN,A.M.EDWARDS,S.FLODIN,AUTH 3 A.FLORES,S.GRASLUND,M.HAMMARSTROM,A.JOHANSSON,I.JOHANSSON,AUTH 4 T.KOTENYOVA,M.MOCHE,M.E.NILSSON,P.NORDLUND,T.NYMAN,K.OLESEN,AUTH 5 C.PERSSON,J.SAGEMARK,S.G.THORSELL,L.TRESAUGUES,AUTH 6 S.VAN DEN BERG,M.WELIN,M.WIKSTROM,M.WISNIEWSKA,J.WEIGELT,AUTH 7 H.SCHUELER,STRUCTURAL GENOMICS CONSORTIUM (SGC)TITL HUMAN PHOSPHOSERINE AMINOTRANSFERASE IN COMPLEX WITH PLPREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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2CU1.A | MAP3K2

General Structure Information 2cu1 MAP3K2 solution structure of the pb1 domain of human protein kinase mekk2b -1.0Å AUTH K.INOUE,T.NAGASHIMA,F.HAYASHI,S.YOKOYAMATITL SOLUTION STRUCTURE OF THE PB1 DOMAIN OF HUMANTITL 2 PROTEIN KINASE MEKK2BREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2YHW.A | GNE

General Structure Information 2yhw GNE high-resolution crystal structures of n-acetylmannosamine kinase: insights about substrate specificity, activity and inhibitor modelling. 1.64Å AUTH J.MARTINEZ,L.D.NGUYEN,E.TAUBERGER,S.HINDERLICH,W.REUTTER,AUTH 2 H.FAN,W.SAENGER,S.MONIOTTITL CRYSTAL STRUCTURES OF N-ACETYLMANNOSAMINE KINASE PROVIDETITL 2 INSIGHTS INTO ENZYME SPECIFICITY AND INHIBITIONREF J.BIOL.CHEM. V. 287 13656 2012REFN ISSN 0021-9258PMID 22343627DOI 10.1074/JBC.M111.318170 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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4CFF.B | PRKAB1

General Structure Information 4cff PRKAB1 structure of full length human ampk in complex with a small molecule activator, a thienopyridone derivative (a-769662) 3.92Å AUTH B.XIAO,M.J.SANDERS,D.CARMENA,N.J.BRIGHT,L.F.HAIRE,AUTH 2 E.UNDERWOOD,B.R.PATEL,R.B.HEATH,P.A.WALKER,S.HALLEN,AUTH 3 F.GIORDANETTO,S.R.MARTIN,D.CARLING,S.J.GAMBLINTITL STRUCTURAL BASIS OF AMPK REGULATION BY SMALL MOLECULETITL 2 ACTIVATORS.REF NAT.COMMUN. V. 4 3017 2013REFN ISSN 2041-1723PMID 24352254DOI 10.1038/NCOMMS4017 Variant Set Distributions Mapped Variants

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2EOC.A | PARP3

General Structure Information 2eoc PARP3 solution structure of the wgr domain from human poly [adp- ribose] polymerase-3 -1.0Å AUTH T.NAGASHIMA,F.HAYASHI,S.YOKOYAMATITL SOLUTION STRUCTURE OF THE WGR DOMAIN FROM HUMANTITL 2 POLY [ADP-RIBOSE] POLYMERASE-3REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2WTK.A | CAB39

General Structure Information 2wtk CAB39 structure of the heterotrimeric lkb1-stradalpha-mo25alpha complex 2.65Å AUTH E.ZEQIRAJ,B.M.FILIPPI,M.DEAK,D.R.ALESSI,D.M.F.VAN AALTENTITL STRUCTURE OF THE LKB1-STRAD-MO25 COMPLEX REVEALS ANTITL 2 ALLOSTERIC MECHANISM OF KINASE ACTIVATION.REF SCIENCE V. 326 1707 2009REFN ISSN 0036-8075PMID 19892943DOI 10.1126/SCIENCE.1178377 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3A7H.A | STK24

General Structure Information 3a7h STK24 human mst3 kinase in complex with atp 1.96Å AUTH T.P.KO,W.Y.JENG,C.I.LIU,M.D.LAI,C.L.WU,W.J.CHANG,H.L.SHR,AUTH 2 T.J.LU,A.H.J.WANGTITL STRUCTURES OF HUMAN MST3 KINASE IN COMPLEX WITH ADENINE, ADPTITL 2 AND MN2+.REF ACTA CRYSTALLOGR.,SECT.D V. 66 145 2010REFN ISSN 0907-4449PMID 20124694DOI 10.1107/S0907444909047507 Variant Set Distributions Mapped Variants

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2X18.A | AKT3

General Structure Information 2×18 AKT3 the crystal structure of the ph domain of human akt3 protein kinase 1.46Å AUTH M.VOLLMAR,J.WANG,Y.ZHANG,J.M.ELKINS,N.BURGESS-BROWN,AUTH 2 A.CHAIKUAD,A.C.W.PIKE,F.VON DELFT,C.BOUNTRA,C.H.ARROWSMITH,AUTH 3 J.WEIGELT,A.EDWARDS,S.KNAPPTITL THE CRYSTAL STRUCTURE OF THE PH DOMAIN OF HUMAN AKT3TITL 2 PROTEIN KINASEREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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