2XAH.A | KDM1A

General Structure Information 2xah KDM1A crystal structure of lsd1-corest in complex with (+)- trans-2-phenylcyclopropyl-1-amine 3.1Å AUTH C.BINDA,S.VALENTE,M.ROMANENGHI,S.PILOTTO,R.CIRILLI,AUTH 2 A.KARYTINOS,G.CIOSSANI,O.A.BOTRUGNO,F.FORNERIS,AUTH 3 M.TARDUGNO,D.E.EDMONDSON,S.MINUCCI,A.MATTEVI,A.MAITITL BIOCHEMICAL, STRUCTURAL, AND BIOLOGICAL EVALUATIONTITL 2 OF TRANYLCYPROMINE DERIVATIVES AS INHIBITORS OFTITL 3 HISTONE DEMETHYLASES LSD1 AND LSD2.REF J.AM.CHEM.SOC. V. 132 6827 2010REFN ISSN 0002-7863PMID 20415477DOI 10.1021/JA101557K Variant Set Distributions Ripley’s K Analysis Plots […]

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2Q3E.B | UGDH

General Structure Information 2q3e UGDH structure of human udp-glucose dehydrogenase complexed with nadh and udp-glucose 2.0Å AUTH S.EGGER,A.CHAIKUAD,K.L.KAVANAGH,U.OPPERMANN,B.NIDETZKYTITL STRUCTURE AND MECHANISM OF HUMAN UDP-GLUCOSETITL 2 6-DEHYDROGENASE.REF J.BIOL.CHEM. V. 286 23877 2011REFN ISSN 0021-9258PMID 21502315DOI 10.1074/JBC.M111.234682 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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4C5W.A | BBOX1

General Structure Information 4c5w BBOX1 three dimensional structure of human gamma-butyrobetaine hydroxylase in complex with 4-(ethyldimethylammonio)butanoate 1.7Å AUTH K.TARS,J.LEITANS,A.KAZAKS,D.ZELENCOVA,E.LIEPINSH,J.KUKA,AUTH 2 M.MAKRECKA,D.LOLA,V.ANDRIANOVS,D.GUSTINA,S.GRINBERGA,AUTH 3 E.LIEPINSH,I.KALVINSH,M.DAMBROVA,E.LOZA,O.PUGOVICSTITL TARGETING CARNITINE BIOSYNTHESIS: DISCOVERY OF NEWTITL 2 INHIBITORS AGAINST GAMMA-BUTYROBETAINE HYDROXYLASE.REF J.MED.CHEM. V. 57 2213 2014REFN ISSN 0022-2623PMID 24571165DOI 10.1021/JM401603E Variant Set Distributions Mapped Variants

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1T0L.B | IDH1

General Structure Information 1t0l IDH1 crystal structure of human cytosolic nadp(+)-dependent isocitrate dehydrogenase in complex with nadp, isocitrate, and calcium(2+) 2.41Å AUTH X.XU,J.ZHAO,Z.XU,B.PENG,Q.HUANG,E.ARNOLD,J.DINGTITL STRUCTURES OF HUMAN CYTOSOLIC NADP-DEPENDENTTITL 2 ISOCITRATE DEHYDROGENASE REVEAL A NOVELTITL 3 SELF-REGULATORY MECHANISM OF ACTIVITYREF J.BIOL.CHEM. V. 279 33946 2004REFN ISSN 0021-9258PMID 15173171DOI 10.1074/JBC.M404298200 Variant Set Distributions Ripley’s K Analysis Plots […]

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2CQ8.A | ALDH1L1

General Structure Information 2cq8 ALDH1L1 solution structure of rsgi ruh-033, a pp-binding domain of 10-fthfdh from human cdna -1.0Å AUTH T.ABE,H.HIROTA,F.HAYASHI,S.YOKOYAMATITL SOLUTION STRUCTURE OF RSGI RUH-033, A PP-BINDINGTITL 2 DOMAIN OF 10-FTHFDH FROM HUMAN CDNAREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2CLP.I | AKR7A3

General Structure Information 2clp AKR7A3 crystal structure of human aflatoxin b1 aldehyde reductase member 3 3.0Å AUTH J.E.DEBRECZENI,C.JOHANSSON,K.KAVANAGH,A.TURNBULL,AUTH 2 E.PAPAGRIGORIOU,F.VON DELFT,A.EDWARDS,C.ARROWSMITH,AUTH 3 J.WEIGELT,M.SUNDSTROM,U.OPPERMANNTITL CRYSTAL STRUCTURE OF HUMAN AFLATOXIN B1 ALDEHYDE REDUCTASETITL 2 MEMBER 3REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

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2BW0.A | ALDH1L1

General Structure Information 2bw0 ALDH1L1 crystal structure of the hydrolase domain of human 10-formyltetrahydrofolate 2 dehydrogenase 1.7Å AUTH P.KURSULA,H.SCHULER,S.FLODIN,P.NILSSON-EHLE,AUTH 2 D.J.OGG,P.SAVITSKY,P.NORDLUND,P.STENMARKTITL STRUCTURES OF THE HYDROLASE DOMAIN OF HUMAN 10-TITL 2 FORMYLTETRAHYDROFOLATE DEHYDROGENASE AND ITSTITL 3 COMPLEX WITH A SUBSTRATE ANALOGUE.REF ACTA CRYSTALLOGR.,SECT.D V. 62 1294 2006REFN ISSN 0907-4449PMID 17057331DOI 10.1107/S0907444906026849 Variant Set Distributions Ripley’s K […]

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2I3Y.A | GPX5

General Structure Information 2i3y GPX5 crystal structure of human glutathione peroxidase 5 2.0Å AUTH K.L.KAVANAGH,U.OPPERMANNTITL CRYSTAL STRUCTURE OF HUMAN GLUTATHIONE PEROXIDASE 5REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2YAN.A | GLRX3

General Structure Information 2yan GLRX3 crystal structure of the second glutaredoxin domain of human txnl2 1.9Å AUTH M.VOLLMAR,C.JOHANSSON,R.COCKING,J.R.C.MUNIZ,T.KROJER,AUTH 2 C.ALLERSTON,F.VON DELFT,C.BOUNTRA,C.H.ARROWSMITH,J.WEIGELT,AUTH 3 A.EDWARDS,U.OPPERMANNTITL CRYSTAL STRUCTURE OF THE SECOND GLUTAREDOXIN DOMAIN OFTITL 2 HUMAN TXNL2REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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2HRB.A | CBR3

General Structure Information 2hrb CBR3 crystal structure of human carbonyl reductase 3, complexed with nadp+ 1.9Å AUTH E.S.PILKA,A.ROJKOVA,K.L.KAVANAGH,F.NIESEN,M.SUNDSTROM,AUTH 2 C.ARROWSMITH,J.WEIGELT,A.EDWARDS,U.OPPERMANNTITL CRYSTAL STRUCTURE OF HUMAN CARBONYL REDUCTASE 3, COMPLEXEDTITL 2 WITH NADP+REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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