1DIG.B | MTHFD1

General Structure Information 1dig MTHFD1 human methylenetetrahydrofolate dehydrogenase / cyclohydrolase complexed with nadp and inhibitor ly374571 2.2Å AUTH A.SCHMIDT,H.WU,R.E.MACKENZIE,V.J.CHEN,J.R.BEWLY,AUTH 2 J.E.RAY,J.E.TOTH,M.CYGLERTITL STRUCTURES OF THREE INHIBITOR COMPLEXES PROVIDETITL 2 INSIGHT INTO THE REACTION MECHANISM OF THE HUMANTITL 3 METHYLENETETRAHYDROFOLATETITL 4 DEHYDROGENASE/CYCLOHYDROLASE.REF BIOCHEMISTRY V. 39 6325 2000REFN ISSN 0006-2960PMID 10828945DOI 10.1021/BI992734Y Variant Set Distributions Mapped Variants

See Details
1U3T.B | ADH1A

General Structure Information 1u3t ADH1A crystal structure of human alcohol dehydrogenase alpha- alpha isoform complexed with n-cyclopentyl-n- cyclobutylformamide determined to 2.5 angstrom resolution 2.49Å AUTH B.J.GIBBONS,T.D.HURLEYTITL STRUCTURE OF THREE CLASS I HUMAN ALCOHOLTITL 2 DEHYDROGENASES COMPLEXED WITH ISOENZYME SPECIFICTITL 3 FORMAMIDE INHIBITORSREF BIOCHEMISTRY V. 43 12555 2004REFN ISSN 0006-2960PMID 15449945DOI 10.1021/BI0489107 Variant Set Distributions Ripley’s […]

See Details
3COS.D | ADH4

General Structure Information 3cos ADH4 crystal structure of human class ii alcohol dehydrogenase (adh4) in complex with nad and zn 2.1Å AUTH K.L.KAVANAGH,N.SHAFQAT,W.YUE,F.VON DELFT,S.BISHOP,A.ROOS,AUTH 2 J.MURRAY,A.M.EDWARDS,C.H.ARROWSMITH,C.BOUNTRA,U.OPPERMANNTITL CRYSTAL STRUCTURE OF HUMAN CLASS II ALCOHOL DEHYDROGENASETITL 2 (ADH4) IN COMPLEX WITH NAD AND ZN.REF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

See Details
1T2F.C | LDHB

General Structure Information 1t2f LDHB human b lactate dehydrogenase complexed with nad+ and 4- hydroxy-1,2,5-oxadiazole-3-carboxylic acid 3.0Å AUTH A.CAMERON,J.READ,R.TRANTER,V.J.WINTER,R.B.SESSIONS,AUTH 2 R.L.BRADY,L.VIVAS,A.EASTON,H.KENDRICK,S.L.CROFT,AUTH 3 D.BARROS,J.L.LAVANDERA,J.J.MARTIN,F.RISCO,AUTH 4 S.GARCIA-OCHOA,F.J.GAMO,L.SANZ,L.LEON,J.R.RUIZ,AUTH 5 R.GABARRO,A.MALLO,F.G.DE LAS HERASTITL IDENTIFICATION AND ACTIVITY OF A SERIES OFTITL 2 AZOLE-BASED COMPOUNDS WITH LACTATETITL 3 DEHYDROGENASE-DIRECTED ANTI-MALARIAL ACTIVITY.REF J.BIOL.CHEM. V. 279 31429 2004REFN ISSN 0021-9258PMID 15117937DOI 10.1074/JBC.M402433200 Variant […]

See Details
1ZMD.A | DLD

General Structure Information 1zmd DLD crystal structure of human dihydrolipoamide dehydrogenase complexed to nadh 2.08Å AUTH C.A.BRAUTIGAM,J.L.CHUANG,D.R.TOMCHICK,M.MACHIUS,AUTH 2 D.T.CHUANGTITL CRYSTAL STRUCTURE OF HUMAN DIHYDROLIPOAMIDETITL 2 DEHYDROGENASE: NAD+/NADH BINDING AND THETITL 3 STRUCTURAL BASIS OF DISEASE-CAUSING MUTATIONSREF J.MOL.BIOL. V. 350 543 2005REFN ISSN 0022-2836PMID 15946682DOI 10.1016/J.JMB.2005.05.014 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons […]

See Details
2F8A.B | GPX1

General Structure Information 2f8a GPX1 crystal structure of the selenocysteine to glycine mutant of human glutathione peroxidase 1 1.5Å AUTH K.L.KAVANAGH,C.JOHANSSON,C.SMEE,O.GILEADI,F.VON DELFT,AUTH 2 U.OPPERMANNTITL CRYSTAL STRUCTURE OF THE SELENOCYSTEINE TO GLYCINE MUTANT OFTITL 2 HUMAN GLUTATHIONE PEROXIDASE 1REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

See Details
3EQM.A | CYP19A1

General Structure Information 3eqm CYP19A1 crystal structure of human placental aromatase cytochrome p450 in complex with androstenedione 2.9Å AUTH D.GHOSH,J.GRISWOLD,M.ERMAN,W.PANGBORNTITL STRUCTURAL BASIS FOR ANDROGEN SPECIFICITY AND OESTROGENTITL 2 SYNTHESIS IN HUMAN AROMATASE.REF NATURE V. 457 219 2009REFN ISSN 0028-0836PMID 19129847DOI 10.1038/NATURE07614 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped […]

See Details
1ERV.A | TXN

General Structure Information 1erv TXN human thioredoxin mutant with cys 73 replaced by ser (reduced form) 1.65Å AUTH A.WEICHSEL,J.R.GASDASKA,G.POWIS,W.R.MONTFORTTITL CRYSTAL STRUCTURES OF REDUCED, OXIDIZED, ANDTITL 2 MUTATED HUMAN THIOREDOXINS: EVIDENCE FOR ATITL 3 REGULATORY HOMODIMER.REF STRUCTURE V. 4 735 1996REFN ISSN 0969-2126PMID 8805557DOI 10.1016/S0969-2126(96)00079-2 Variant Set Distributions Mapped Variants

See Details
1OG2.A | CYP2C9

General Structure Information 1og2 CYP2C9 structure of human cytochrome p450 cyp2c9 2.6Å AUTH P.A.WILLIAMS,J.COSME,A.WARD,H.C.ANGOVE,AUTH 2 D.MATAK VINKOVIC,H.JHOTITITL CRYSTAL STRUCTURE OF HUMAN CYTOCHROME P450 2C9TITL 2 WITH BOUND WARFARINREF NATURE V. 424 464 2003REFN ISSN 0028-0836PMID 12861225DOI 10.1038/NATURE01862 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

See Details
2OZL.A | PDHA1

General Structure Information 2ozl PDHA1 human pyruvate dehydrogenase s264e variant 1.9Å AUTH F.SEIFERT,E.M.CISZAK,L.G.KOROTCHKINA,R.GOLBIK,AUTH 2 M.SPINKA,P.M.DOMINIAK,S.SIDHU,J.BRAUER,M.S.PATEL,AUTH 3 K.TITTMANNTITL PHOSPHORYLATION OF SERINE 264 IMPEDES ACTIVE SITETITL 2 ACCESSIBILITY IN THE E1 COMPONENT OF THE HUMANTITL 3 PYRUVATE DEHYDROGENASE MULTIENZYME COMPLEXREF BIOCHEMISTRY V. 46 6277 2007REFN ISSN 0006-2960PMID 17474719DOI 10.1021/BI700083Z Variant Set Distributions Ripley’s K Analysis Plots Variant […]

See Details