4N4W.A | SMO

General Structure Information 4n4w SMO structure of the human smoothened receptor in complex with sant-1. 2.8Å AUTH C.WANG,H.WU,T.EVRON,E.VARDY,G.W.HAN,X.P.HUANG,S.J.HUFEISEN,AUTH 2 T.J.MANGANO,D.J.URBAN,V.KATRITCH,V.CHEREZOV,M.G.CARON,AUTH 3 B.L.ROTH,R.C.STEVENSTITL STRUCTURAL BASIS FOR SMOOTHENED RECEPTOR MODULATION ANDTITL 2 CHEMORESISTANCE TO ANTICANCER DRUGS.REF NAT COMMUN V. 5 4355 2014REFN ESSN 2041-1723PMID 25008467DOI 10.1038/NCOMMS5355 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped […]

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4AJ5.Q | SKA2

General Structure Information 4aj5 SKA2 crystal structure of the ska core complex 3.32Å AUTH A.A.JEYAPRAKASH,A.SANTAMARIA,U.JAYACHANDRAN,Y.W.CHAN,AUTH 2 C.BENDA,E.A.NIGG,E.CONTITITL STRUCTURAL AND FUNCTIONAL ORGANIZATION OF THE SKA COMPLEX,TITL 2 A KEY COMPONENT OF THE KINETOCHORE-MICROTUBULE INTERFACE.REF MOL.CELL V. 46 274 2012REFN ISSN 1097-2765PMID 22483620DOI 10.1016/J.MOLCEL.2012.03.005 Variant Set Distributions Mapped Variants

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4AJ5.U | SKA3

General Structure Information 4aj5 SKA3 crystal structure of the ska core complex 3.32Å AUTH A.A.JEYAPRAKASH,A.SANTAMARIA,U.JAYACHANDRAN,Y.W.CHAN,AUTH 2 C.BENDA,E.A.NIGG,E.CONTITITL STRUCTURAL AND FUNCTIONAL ORGANIZATION OF THE SKA COMPLEX,TITL 2 A KEY COMPONENT OF THE KINETOCHORE-MICROTUBULE INTERFACE.REF MOL.CELL V. 46 274 2012REFN ISSN 1097-2765PMID 22483620DOI 10.1016/J.MOLCEL.2012.03.005 Variant Set Distributions Mapped Variants

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3QXY.A | SETD6

General Structure Information 3qxy SETD6 human setd6 in complex with rela lys310 2.09Å AUTH Y.CHANG,D.LEVY,J.R.HORTON,J.PENG,X.ZHANG,O.GOZANI,X.CHENGTITL STRUCTURAL BASIS OF SETD6-MEDIATED REGULATION OF THE NF-KBTITL 2 NETWORK VIA METHYL-LYSINE SIGNALING.REF NUCLEIC ACIDS RES. V. 39 6380 2011REFN ISSN 0305-1048PMID 21515635DOI 10.1093/NAR/GKR256 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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4OR2.B | GRM1

General Structure Information 4or2 GRM1 human class c g protein-coupled metabotropic glutamate receptor 1 in complex with a negative allosteric modulator 2.8Å AUTH H.WU,C.WANG,K.J.GREGORY,G.W.HAN,H.P.CHO,Y.XIA,C.M.NISWENDER,AUTH 2 V.KATRITCH,J.MEILER,V.CHEREZOV,P.J.CONN,R.C.STEVENSTITL STRUCTURE OF A CLASS C GPCR METABOTROPIC GLUTAMATE RECEPTORTITL 2 1 BOUND TO AN ALLOSTERIC MODULATORREF SCIENCE V. 344 58 2014REFN ISSN 0036-8075PMID 24603153DOI 10.1126/SCIENCE.1249489 Variant Set Distributions Ripley’s […]

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4OR2.B | GRM1

General Structure Information 4or2 GRM1 human class c g protein-coupled metabotropic glutamate receptor 1 in complex with a negative allosteric modulator 2.8Å AUTH H.WU,C.WANG,K.J.GREGORY,G.W.HAN,H.P.CHO,Y.XIA,C.M.NISWENDER,AUTH 2 V.KATRITCH,J.MEILER,V.CHEREZOV,P.J.CONN,R.C.STEVENSTITL STRUCTURE OF A CLASS C GPCR METABOTROPIC GLUTAMATE RECEPTORTITL 2 1 BOUND TO AN ALLOSTERIC MODULATORREF SCIENCE V. 344 58 2014REFN ISSN 0036-8075PMID 24603153DOI 10.1126/SCIENCE.1249489 Variant Set Distributions Ripley’s […]

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4OR2.B | GRM1

General Structure Information 4or2 GRM1 human class c g protein-coupled metabotropic glutamate receptor 1 in complex with a negative allosteric modulator 2.8Å AUTH H.WU,C.WANG,K.J.GREGORY,G.W.HAN,H.P.CHO,Y.XIA,C.M.NISWENDER,AUTH 2 V.KATRITCH,J.MEILER,V.CHEREZOV,P.J.CONN,R.C.STEVENSTITL STRUCTURE OF A CLASS C GPCR METABOTROPIC GLUTAMATE RECEPTORTITL 2 1 BOUND TO AN ALLOSTERIC MODULATORREF SCIENCE V. 344 58 2014REFN ISSN 0036-8075PMID 24603153DOI 10.1126/SCIENCE.1249489 Variant Set Distributions Ripley’s […]

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3OE8.B | CXCR4

General Structure Information 3oe8 CXCR4 crystal structure of the cxcr4 chemokine receptor in complex with a small molecule antagonist it1t in p1 spacegroup 3.1Å AUTH B.WU,E.Y.CHIEN,C.D.MOL,G.FENALTI,W.LIU,V.KATRITCH,R.ABAGYAN,AUTH 2 A.BROOUN,P.WELLS,F.C.BI,D.J.HAMEL,P.KUHN,T.M.HANDEL,AUTH 3 V.CHEREZOV,R.C.STEVENSTITL STRUCTURES OF THE CXCR4 CHEMOKINE GPCR WITH SMALL-MOLECULETITL 2 AND CYCLIC PEPTIDE ANTAGONISTS.REF SCIENCE V. 330 1066 2010REFN ISSN 0036-8075PMID 20929726DOI 10.1126/SCIENCE.1194396 Variant Set Distributions […]

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3OE8.B | CXCR4

General Structure Information 3oe8 CXCR4 crystal structure of the cxcr4 chemokine receptor in complex with a small molecule antagonist it1t in p1 spacegroup 3.1Å AUTH B.WU,E.Y.CHIEN,C.D.MOL,G.FENALTI,W.LIU,V.KATRITCH,R.ABAGYAN,AUTH 2 A.BROOUN,P.WELLS,F.C.BI,D.J.HAMEL,P.KUHN,T.M.HANDEL,AUTH 3 V.CHEREZOV,R.C.STEVENSTITL STRUCTURES OF THE CXCR4 CHEMOKINE GPCR WITH SMALL-MOLECULETITL 2 AND CYCLIC PEPTIDE ANTAGONISTS.REF SCIENCE V. 330 1066 2010REFN ISSN 0036-8075PMID 20929726DOI 10.1126/SCIENCE.1194396 Variant Set Distributions […]

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4MBS.B | CCR5

General Structure Information 4mbs CCR5 crystal structure of the ccr5 chemokine receptor 2.71Å AUTH Q.TAN,Y.ZHU,J.LI,Z.CHEN,G.W.HAN,I.KUFAREVA,T.LI,L.MA,AUTH 2 G.FENALTI,J.LI,W.ZHANG,X.XIE,H.YANG,H.JIANG,V.CHEREZOV,AUTH 3 H.LIU,R.C.STEVENS,Q.ZHAO,B.WUTITL STRUCTURE OF THE CCR5 CHEMOKINE RECEPTOR-HIV ENTRY INHIBITORTITL 2 MARAVIROC COMPLEX.REF SCIENCE V. 341 1387 2013REFN ISSN 0036-8075PMID 24030490DOI 10.1126/SCIENCE.1241475 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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