1YC0.A | HGFAC

General Structure Information 1yc0 HGFAC short form hgfa with first kunitz domain from hai-1 2.6Å AUTH S.SHIA,J.STAMOS,D.KIRCHHOFER,B.FAN,J.WU,R.T.CORPUZ,AUTH 2 L.SANTELL,R.A.LAZARUS,C.EIGENBROTTITL CONFORMATIONAL LABILITY IN SERINE PROTEASE ACTIVE SITES:TITL 2 STRUCTURES OF HEPATOCYTE GROWTH FACTOR ACTIVATOR (HGFA)TITL 3 ALONE AND WITH THE INHIBITORY DOMAIN FROM HGFA INHIBITOR-1B.REF J.MOL.BIOL. V. 346 1335 2005REFN ISSN 0022-2836PMID 15713485DOI 10.1016/J.JMB.2004.12.048 Variant Set […]

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1YC0.A | HGFAC

General Structure Information 1yc0 HGFAC short form hgfa with first kunitz domain from hai-1 2.6Å AUTH S.SHIA,J.STAMOS,D.KIRCHHOFER,B.FAN,J.WU,R.T.CORPUZ,AUTH 2 L.SANTELL,R.A.LAZARUS,C.EIGENBROTTITL CONFORMATIONAL LABILITY IN SERINE PROTEASE ACTIVE SITES:TITL 2 STRUCTURES OF HEPATOCYTE GROWTH FACTOR ACTIVATOR (HGFA)TITL 3 ALONE AND WITH THE INHIBITORY DOMAIN FROM HGFA INHIBITOR-1B.REF J.MOL.BIOL. V. 346 1335 2005REFN ISSN 0022-2836PMID 15713485DOI 10.1016/J.JMB.2004.12.048 Variant Set […]

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1GMY.A | CTSB

General Structure Information 1gmy CTSB cathepsin b complexed with dipeptidyl nitrile inhibitor 1.9Å AUTH P.D.GREENSPAN,K.L.CLARK,R.A.TOMMASI,S.D.COWEN,AUTH 2 L.W.MCQUIRE,D.L.FARLEY,J.H.VAN DUZER,R.L.GOLDBERG,AUTH 3 H.ZHOU,Z.DU,J.J.FITT,D.E.COPPA,Z.FANG,W.MACCHIA,AUTH 4 L.ZHU,M.P.CAPPARELLI,R.GOLDSTEIN,A.M.WIGG,AUTH 5 J.R.DOUGHTY,R.S BOHACEK,A.K.KNAPTITL IDENTIFICATION OF DIPEPTIDYL NITRILES AS POTENTTITL 2 AND SELECTIVE INHIBITORS OF CATHEPSIN B THROUGHTITL 3 STRUCTURE-BASED DRUG DESIGNREF J.MED.CHEM. V. 44 4524 2001REFN ISSN 0022-2623PMID 11741472DOI 10.1021/JM010206Q Variant Set Distributions […]

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