3N3K.A | USP8

General Structure Information 3n3k USP8 the catalytic domain of usp8 in complex with a usp8 specific inhibitor 2.6Å AUTH A.ERNST,G.AVVAKUMOV,J.TONG,Y.FAN,Y.ZHAO,P.ALBERTS,A.PERSAUD,AUTH 2 J.R.WALKER,A.M.NECULAI,D.NECULAI,A.VOROBYOV,P.GARG,L.BEATTY,AUTH 3 P.K.CHAN,Y.C.JUANG,M.C.LANDRY,C.YEH,E.ZEQIRAJ,K.KARAMBOULAS,AUTH 4 A.ALLALI-HASSANI,M.VEDADI,M.TYERS,J.MOFFAT,F.SICHERI,AUTH 5 L.PELLETIER,D.DUROCHER,B.RAUGHT,D.ROTIN,J.YANG,M.F.MORAN,AUTH 6 S.DHE-PAGANON,S.S.SIDHUTITL A STRATEGY FOR MODULATION OF ENZYMES IN THE UBIQUITINTITL 2 SYSTEM.REF SCIENCE V. 339 590 2013REFN ISSN 0036-8075PMID 23287719DOI 10.1126/SCIENCE.1230161 Variant Set Distributions Ripley’s K […]

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2EDB.A | DCC

General Structure Information 2edb DCC solution structure of the fourth fibronectin type iii domain of human netrin receptor dcc -1.0Å AUTH N.TOCHIO,S.KOSHIBA,T.KIGAWA,S.YOKOYAMATITL SOLUTION STRUCTURE OF THE FOURTH FIBRONECTIN TYPETITL 2 III DOMAIN OF HUMAN NETRIN RECEPTOR DCCREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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3RZE.A | HRH1

General Structure Information 3rze HRH1 structure of the human histamine h1 receptor in complex with doxepin 3.1Å AUTH T.SHIMAMURA,M.SHIROISHI,S.WEYAND,H.TSUJIMOTO,G.WINTER,AUTH 2 V.KATRITCH,R.ABAGYAN,V.CHEREZOV,W.LIU,G.W.HAN,T.KOBAYASHI,AUTH 3 R.C.STEVENS,S.IWATATITL STRUCTURE OF THE HUMAN HISTAMINE H1 RECEPTOR COMPLEX WITHTITL 2 DOXEPIN.REF NATURE V. 475 65 2011REFN ISSN 0028-0836PMID 21697825DOI 10.1038/NATURE10236 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity […]

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2LXU.A | HNRNPH1

General Structure Information 2lxu HNRNPH1 solution nmr structure of the eukaryotic rna recognition motif, rrm1, from the heterogeneous nuclear ribonucleoprotein h from homo sapiens, northeast structural genomics consortium (nesg) target hr8614a -1.0Å AUTH T.A.RAMELOT,Y.YANG,K.PEDERSON,R.SHASTRY,E.KOHAN,H.JANJUA,AUTH 2 R.XIAO,T.B.ACTON,J.K.EVERETT,J.H.PRESTEGARD,G.T.MONTELIONE,AUTH 3 M.A.KENNEDYTITL SOLUTION NMR STRUCTURE OF THE EUKARYOTIC RNA RECOGNITIONTITL 2 MOTIF, RRM1, FROM THE HETEROGENEOUS NUCLEARTITL 3 RIBONUCLEOPROTEIN […]

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2JRZ.A | KDM5C

General Structure Information 2jrz KDM5C solution structure of the bright/arid domain from the human jarid1c protein. -1.0Å AUTH C.KOEHLER,S.BISHOP,E.F.DOWLER,P.SCHMIEDER,A.DIEHL,AUTH 2 H.OSCHKINAT,L.J.BALLTITL BACKBONE AND SIDECHAIN 1H, 13C AND 15N RESONANCETITL 2 ASSIGNMENTS OF THE BRIGHT/ARID DOMAIN FROM THETITL 3 HUMAN JARID1C (SMCX) PROTEIN.REF BIOMOL.NMR ASSIGN. V. 2 9 2008REFN ISSN 1874-2718PMID 19636912DOI 10.1007/S12104-007-9071-7 Variant Set Distributions […]

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2XYN.B | ABL2

General Structure Information 2xyn ABL2 human abl2 in complex with aurora kinase inhibitor vx-680 2.81Å AUTH E.SALAH,E.UGOCHUKWU,A.J.BARR,F.VON DELFT,S.KNAPP,AUTH 2 J.M.ELKINSTITL CRYSTAL STRUCTURES OF ABL-RELATED GENE (ABL2) INTITL 2 COMPLEX WITH IMATINIB, TOZASERTIB (VX-680), AND ATITL 3 TYPE I INHIBITOR OF THE TRIAZOLE CARBOTHIOAMIDETITL 4 CLASS.REF J.MED.CHEM. V. 54 2359 2011REFN ISSN 0022-2623PMID 21417343DOI 10.1021/JM101506N Variant […]

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3FDT.A | CBX5

General Structure Information 3fdt CBX5 crystal structure of the complex of human chromobox homolog 5 (cbx5) with h3k9(me)3 peptide 2.0Å AUTH L.KAUSTOV,H.OUYANG,M.AMAYA,A.LEMAK,N.NADY,S.DUAN,G.A.WASNEY,AUTH 2 Z.LI,M.VEDADI,M.SCHAPIRA,J.MIN,C.H.ARROWSMITHTITL RECOGNITION AND SPECIFICITY DETERMINANTS OF THE HUMAN CBXTITL 2 CHROMODOMAINS.REF J.BIOL.CHEM. V. 286 521 2011REFN ISSN 0021-9258PMID 21047797DOI 10.1074/JBC.M110.191411 Variant Set Distributions Mapped Variants

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2I3C.A | ASPA

General Structure Information 2i3c ASPA crystal structure of an aspartoacylase from homo sapiens 2.8Å AUTH E.BITTO,C.A.BINGMAN,G.E.WESENBERG,J.G.MCCOY,AUTH 2 G.N.PHILLIPSTITL STRUCTURE OF ASPARTOACYLASE, THE BRAIN ENZYMETITL 2 IMPAIRED IN CANAVAN DISEASE.REF PROC.NATL.ACAD.SCI.USA V. 104 456 2007REFN ISSN 0027-8424PMID 17194761DOI 10.1073/PNAS.0607817104 Variant Set Distributions Pathogenic Proximity Analysis Mapped Variants

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2LNI.A | STIP1

General Structure Information 2lni STIP1 solution nmr structure of stress-induced-phosphoprotein 1 sti1 from homo sapiens, northeast structural genomics consortium target hr4403e -1.0Å AUTH Y.TANG,G.LIU,K.HAMILTON,C.CICCOSANTI,R.SHASTRY,B.ROST,AUTH 2 T.B.ACTON,R.XIAO,J.K.EVERETT,G.T.MONTELIONETITL NORTHEAST STRUCTURAL GENOMICS CONSORTIUM TARGET HR4403EREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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3IU2.A | NMT1

General Structure Information 3iu2 NMT1 crystal structure of human type-i n-myristoyltransferase with bound myristoyl-coa and inhibitor ddd90096 1.73Å AUTH W.QIU,A.HUTCHINSON,A.WERNIMONT,Y.-H.LIN,A.KANIA,AUTH 2 M.RAVICHANDRAN,I.KOZIERADZKI,D.COSSAR,M.SCHAPIRA,AUTH 3 C.H.ARROWSMITH,C.BOUNTRA,J.WEIGELT,A.M.EDWARDS,P.G.WYATT,AUTH 4 M.A.J.FERGUSON,J.A.FREARSON,S.Y.BRAND,D.A.ROBINSON,AUTH 5 A.BOCHKAREV,R.HUITITL CRYSTAL STRUCTURE OF HUMAN TYPE-I N-MYRISTOYLTRANSFERASETITL 2 WITH BOUND MYRISTOYL-COA AND INHIBITOR DDD90096REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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