3VW7.A | F2R

General Structure Information 3vw7 F2R crystal structure of human protease-activated receptor 1 (par1) bound with antagonist vorapaxar at 2.2 angstrom 2.2Å AUTH C.ZHANG,Y.SRINIVASAN,D.H.ARLOW,J.J.FUNG,D.PALMER,Y.ZHENG,AUTH 2 H.F.GREEN,A.PANDEY,R.O.DROR,D.E.SHAW,W.I.WEIS,S.R.COUGHLIN,AUTH 3 B.K.KOBILKATITL HIGH-RESOLUTION CRYSTAL STRUCTURE OF HUMANTITL 2 PROTEASE-ACTIVATED RECEPTOR 1REF NATURE V. 492 387 2012REFN ISSN 0028-0836PMID 23222541DOI 10.1038/NATURE11701 Variant Set Distributions Mapped Variants

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4MQS.A | CHRM2

General Structure Information 4mqs CHRM2 structure of active human m2 muscarinic acetylcholine receptor bound to the agonist iperoxo 3.5Å AUTH A.C.KRUSE,A.M.RING,A.MANGLIK,J.HU,K.HU,K.EITEL,H.HUBNER,AUTH 2 E.PARDON,C.VALANT,P.M.SEXTON,A.CHRISTOPOULOS,C.C.FELDER,AUTH 3 P.GMEINER,J.STEYAERT,W.I.WEIS,K.C.GARCIA,J.WESS,B.K.KOBILKATITL ACTIVATION AND ALLOSTERIC MODULATION OF A MUSCARINICTITL 2 ACETYLCHOLINE RECEPTOR.REF NATURE V. 504 101 2013REFN ISSN 0028-0836PMID 24256733DOI 10.1038/NATURE12735 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped […]

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