2YHW.A | GNE

General Structure Information 2yhw GNE high-resolution crystal structures of n-acetylmannosamine kinase: insights about substrate specificity, activity and inhibitor modelling. 1.64Å AUTH J.MARTINEZ,L.D.NGUYEN,E.TAUBERGER,S.HINDERLICH,W.REUTTER,AUTH 2 H.FAN,W.SAENGER,S.MONIOTTITL CRYSTAL STRUCTURES OF N-ACETYLMANNOSAMINE KINASE PROVIDETITL 2 INSIGHTS INTO ENZYME SPECIFICITY AND INHIBITIONREF J.BIOL.CHEM. V. 287 13656 2012REFN ISSN 0021-9258PMID 22343627DOI 10.1074/JBC.M111.318170 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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4NCS.A | NEU2

General Structure Information 4ncs NEU2 human sialidase 2 in complex with 2,3-difluorosialic acid (covalent intermediate) 2.2Å AUTH S.BUCHINI,F.X.GALLAT,I.R.GREIG,J.H.KIM,S.WAKATSUKI,AUTH 2 L.M.CHAVAS,S.G.WITHERSTITL TUNING MECHANISM-BASED INACTIVATORS OF NEURAMINIDASES:TITL 2 MECHANISTIC AND STRUCTURAL INSIGHTS.REF ANGEW.CHEM.INT.ED.ENGL. V. 53 3382 2014REFN ISSN 1433-7851PMID 24591206DOI 10.1002/ANIE.201309675 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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2DF3.A | SIGLEC7

General Structure Information 2df3 SIGLEC7 the structure of siglec-7 in complex with alpha(2,3)/alpha(2,6) disialyl lactotetraosyl 2-(trimethylsilyl)ethyl 1.9Å AUTH H.ATTRILL,H.TAKAZAWA,S.WITT,S.KELM,R.ISECKE,R.BROSSMER,AUTH 2 T.ANDO,H.ISHIDA,M.KISO,P.R.CROCKER,D.M.F.VAN AALTENTITL THE STRUCTURE OF SIGLEC-7 IN COMPLEX WITH SIALOSIDES: LEADSTITL 2 FOR RATIONAL STRUCTURE-BASED INHIBITOR DESIGNREF BIOCHEM.J. V. 397 271 2006REFN ISSN 0264-6021PMID 16623661DOI 10.1042/BJ20060103 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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3JTC.A | PROCR

General Structure Information 3jtc PROCR importance of mg2+ in the ca2+-dependent folding of the gamma- carboxyglutamic acid domains of vitamin k-dependent clotting and anticlotting proteins 1.6Å AUTH K.VADIVEL,S.AGAH,A.S.MESSER,D.CASCIO,M.S.BAJAJ,AUTH 2 S.KRISHNASWAMY,C.T.ESMON,K.PADMANABHAN,S.P.BAJAJTITL STRUCTURAL AND FUNCTIONAL STUDIES OF GAMMA-CARBOXYGLUTAMICTITL 2 ACID DOMAINS OF FACTOR VIIA AND ACTIVATED PROTEIN C: ROLE OFTITL 3 MAGNESIUM AT PHYSIOLOGICAL CALCIUM.REF J.MOL.BIOL. V. […]

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1WJP.A | ZBTB21

General Structure Information 1wjp ZBTB21 solution structure of zf-c2h2 domains from human zinc finger protein 295 -1.0Å AUTH T.TOMIZAWA,T.KIGAWA,K.SAITO,S.KOSHIBA,M.INOUE,AUTH 2 S.YOKOYAMATITL SOLUTION STRUCTURE OF ZF-C2H2 DOMAINS FROM HUMANTITL 2 ZINC FINGER PROTEIN 295REF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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3H5C.A | SERPINA10

General Structure Information 3h5c SERPINA10 x-ray structure of protein z-protein z inhibitor complex 3.26Å AUTH X.HUANG,A.DEMENTIEV,S.T.OLSON,P.G.GETTINSTITL BASIS FOR THE SPECIFICITY AND ACTIVATION OF THE SERPINTITL 2 PROTEIN Z-DEPENDENT PROTEINASE INHIBITOR (ZPI) AS ANTITL 3 INHIBITOR OF MEMBRANE-ASSOCIATED FACTOR XA.REF J.BIOL.CHEM. V. 285 20399 2010REFN ISSN 0021-9258PMID 20427285DOI 10.1074/JBC.M110.112748 Variant Set Distributions Ripley’s K Analysis Plots […]

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2IWZ.B | OXSM

General Structure Information 2iwz OXSM human mitochondrial beta-ketoacyl acp synthase complexed with hexanoic acid 1.65Å AUTH C.E.CHRISTENSEN,B.B.KRAGELUND,P.VON WETTSTEIN-KNOWLES,AUTH 2 A.HENRIKSENTITL STRUCTURE OF THE HUMAN BETA-KETOACYL [ACP] SYNTHASE FROMTITL 2 THE MITOCHONDRIAL TYPE II FATTY ACID SYNTHASE.REF PROTEIN SCI. V. 16 261 2007REFN ISSN 0961-8368PMID 17242430DOI 10.1110/PS.062473707 Variant Set Distributions Ripley’s K Analysis Plots Variant Set […]

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1WVO.A | NANS

General Structure Information 1wvo NANS solution structure of rsgi ruh-029, an antifreeze protein like domain in human n-acetylneuraminic acid phosphate synthase gene. -1.0Å AUTH T.HAMADA,Y.ITO,T.ABE,F.HAYASHI,P.GUNTERT,M.INOUE,AUTH 2 T.KIGAWA,T.TERADA,M.SHIROUZU,M.YOSHIDA,A.TANAKA,AUTH 3 S.SUGANO,S.YOKOYAMA,H.HIROTATITL SOLUTION STRUCTURE OF THE ANTIFREEZE-LIKE DOMAINTITL 2 OF HUMAN SIALIC ACID SYNTHASEREF PROTEIN SCI. V. 15 1010 2006REFN ISSN 0961-8368PMID 16597820DOI 10.1110/PS.051700406 Variant Set Distributions Mapped […]

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2C43.A | AASDHPPT

General Structure Information 2c43 AASDHPPT structure of aminoadipate-semialdehyde dehydrogenase- phosphopantetheinyl transferase in complex with coenzyme a 1.93Å AUTH G.BUNKOCZI,S.PASTA,A.JOSHI,X.WU,K.L.KAVANAGH,S.SMITH,AUTH 2 U.OPPERMANNTITL MECHANISM AND SUBSTRATE RECOGNITION OF HUMAN HOLO ACPTITL 2 SYNTHASE.REF CHEM.BIOL. V. 14 1243 2007REFN ISSN 1074-5521PMID 18022563DOI 10.1016/J.CHEMBIOL.2007.10.013 Variant Set Distributions Mapped Variants

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4IE5.A | FTO

General Structure Information 4ie5 FTO crystal structure of the human fat mass and obesity associated protein (fto) in complex with n-[(3-hydroxypyridin-2-yl)carbonyl]glycine (md6) 1.95Å AUTH W.S.AIK,M.DEMETRIADES,M.K.K.HAMDAN,E.A.L.BAGG,K.K.YEOH,AUTH 2 C.LEJEUNE,Z.ZHANG,M.A.MCDONOUGH,C.J.SCHOFIELDTITL STRUCTURAL BASIS FOR INHIBITION OF THE FAT MASS AND OBESITYTITL 2 ASSOCIATED PROTEIN (FTO)REF J.MED.CHEM. V. 56 3680 2013REFN ISSN 0022-2623PMID 23547775DOI 10.1021/JM400193D Variant Set Distributions Mapped Variants

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