1JUJ.C | TYMS

General Structure Information 1juj TYMS human thymidylate synthase bound to dump and ly231514, a pyrrolo(2,3-d)pyrimidine-based antifolate 3.0Å AUTH P.H.SAYRE,J.S.FINER-MOORE,T.A.FRITZ,D.BIERMANN,AUTH 2 S.B.GATES,W.C.MACKELLAR,V.F.PATEL,R.M.STROUDTITL MULTI-TARGETED ANTIFOLATES AIMED AT AVOIDING DRUGTITL 2 RESISTANCE FORM COVALENT CLOSED INHIBITORYTITL 3 COMPLEXES WITH HUMAN AND ESCHERICHIA COLITITL 4 THYMIDYLATE SYNTHASES.REF J.MOL.BIOL. V. 313 813 2001REFN ISSN 0022-2836PMID 11697906DOI 10.1006/JMBI.2001.5074 Variant Set Distributions […]

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3RCW.E | BRD1

General Structure Information 3rcw BRD1 crystal structure of the bromodomain of human brd1 2.21Å AUTH P.FILIPPAKOPOULOS,S.PICAUD,M.MANGOS,T.KEATES,J.P.LAMBERT,AUTH 2 D.BARSYTE-LOVEJOY,I.FELLETAR,R.VOLKMER,S.MULLER,T.PAWSON,AUTH 3 A.C.GINGRAS,C.H.ARROWSMITH,S.KNAPPTITL HISTONE RECOGNITION AND LARGE-SCALE STRUCTURAL ANALYSIS OFTITL 2 THE HUMAN BROMODOMAIN FAMILY.REF CELL(CAMBRIDGE,MASS.) V. 149 214 2012REFN ISSN 0092-8674PMID 22464331DOI 10.1016/J.CELL.2012.02.013 Variant Set Distributions Mapped Variants

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2D9N.A | CPSF4

General Structure Information 2d9n CPSF4 solution structure of ccch type zinc-finger domain 2 in cleavage and polyadenylation specificity factor -1.0Å AUTH C.ABE,Y.MUTO,M.INOUE,T.KIGAWA,T.TERADA,M.SHIROUZU,AUTH 2 S.YOKOYAMATITL SOLUTION STRUCTURE OF CCCH TYPE ZINC-FINGER DOMAINTITL 2 2 IN CLEAVAGE AND POLYADENYLATION SPECIFICITYTITL 3 FACTORREF TO BE PUBLISHEDREFN Variant Set Distributions Mapped Variants

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6RLX.B | RLN2

General Structure Information 6rlx RLN2 x-ray structure of human relaxin at 1.5 angstroms. comparison to insulin and implications for receptor binding determinants 1.5Å AUTH C.EIGENBROT,M.RANDAL,C.QUAN,J.BURNIER,L.OCONNELL,AUTH 2 E.RINDERKNECHT,A.A.KOSSIAKOFFTITL X-RAY STRUCTURE OF HUMAN RELAXIN AT 1.5 A. COMPARISON TOTITL 2 INSULIN AND IMPLICATIONS FOR RECEPTOR BINDING DETERMINANTS.REF J.MOL.BIOL. V. 221 15 1991REFN ISSN 0022-2836PMID 1656049 Variant Set […]

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1LQ8.G | SERPINA5

General Structure Information 1lq8 SERPINA5 crystal structure of cleaved protein c inhibitor 2.4Å AUTH J.A.HUNTINGTON,M.KJELLBERG,J.STENFLOTITL CRYSTAL STRUCTURE OF PROTEIN C INHIBITOR PROVIDES INSIGHTSTITL 2 INTO HORMONE BINDING AND HEPARIN ACTIVATIONREF STRUCTURE V. 11 205 2003REFN ISSN 0969-2126PMID 12575940DOI 10.1016/S0969-2126(02)00944-9 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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1LQ8.B | SERPINA5

General Structure Information 1lq8 SERPINA5 crystal structure of cleaved protein c inhibitor 2.4Å AUTH J.A.HUNTINGTON,M.KJELLBERG,J.STENFLOTITL CRYSTAL STRUCTURE OF PROTEIN C INHIBITOR PROVIDES INSIGHTSTITL 2 INTO HORMONE BINDING AND HEPARIN ACTIVATIONREF STRUCTURE V. 11 205 2003REFN ISSN 0969-2126PMID 12575940DOI 10.1016/S0969-2126(02)00944-9 Variant Set Distributions Mapped Variants

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2UZP.B | PRKCG

General Structure Information 2uzp PRKCG crystal structure of the c2 domain of human protein kinase c gamma. 2.0Å AUTH A.C.W.PIKE,A.AMOS,C.JOHANSSON,F.SOBOTT,P.SAVITSKY,AUTH 2 G.BERRIDGE,O.FEDOROV,C.UMEANO,F.GORREC,G.BUNKOCZI,AUTH 3 J.DEBRECZENI,F.VON DELFT,C.H.ARROWSMITH,A.EDWARDS,J.WEIGELT,AUTH 4 M.SUNDSTROM,S.KNAPPTITL CRYSTAL STRUCTURE OF C2 DOMAIN OF PROTEIN KINASE C GAMMAREF TO BE PUBLISHEDREFN Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis Mapped Variants

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4F0X.H | MLYCD

General Structure Information 4f0x MLYCD crystal structure of human malonyl-coa decarboxylase (peroxisomal isoform) 3.29Å AUTH D.APARICIO,R.PEREZ-LUQUE,X.CARPENA,M.DIAZ,J.C.FERRER,AUTH 2 P.C.LOEWEN,I.FITATITL STRUCTURAL ASYMMETRY AND DISULFIDE BRIDGES AMONG SUBUNITSTITL 2 MODULATE THE ACTIVITY OF HUMAN MALONYL-COA DECARBOXYLASE.REF J.BIOL.CHEM. V. 288 11907 2013REFN ISSN 0021-9258PMID 23482565DOI 10.1074/JBC.M112.443846 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity Analysis […]

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3SE4.B | IFNW1

General Structure Information 3se4 IFNW1 human ifnw-ifnar ternary complex 3.5Å AUTH C.THOMAS,I.MORAGA,D.LEVIN,P.O.KRUTZIK,Y.PODOPLELOVA,A.TREJO,AUTH 2 C.LEE,G.YARDEN,S.E.VLECK,J.S.GLENN,G.P.NOLAN,J.PIEHLER,AUTH 3 G.SCHREIBER,K.C.GARCIATITL STRUCTURAL LINKAGE BETWEEN LIGAND DISCRIMINATION ANDTITL 2 RECEPTOR ACTIVATION BY TYPE I INTERFERONS.REF CELL(CAMBRIDGE,MASS.) V. 146 621 2011REFN ISSN 0092-8674PMID 21854986DOI 10.1016/J.CELL.2011.06.048 Variant Set Distributions Mapped Variants

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1TPG.A | PLAT

General Structure Information 1tpg PLAT f1-g module pair residues 1-91 (c83s) of tissue-type plasminogen activator (t-pa) (nmr, 298k, ph2.95, representative structure) -1.0Å AUTH B.O.SMITH,A.K.DOWNING,P.C.DRISCOLL,T.J.DUDGEON,AUTH 2 I.D.CAMPBELLTITL THE SOLUTION STRUCTURE AND BACKBONE DYNAMICS OFTITL 2 THE FIBRONECTIN TYPE I AND EPIDERMAL GROWTHTITL 3 FACTOR-LIKE PAIR OF MODULES OF TISSUE-TYPETITL 4 PLASMINOGEN ACTIVATOR.REF STRUCTURE V. 3 823 […]

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