4O0X.A | PAK4

General Structure Information 4o0x PAK4 back pocket flexibility provides group-ii pak selectivity for type 1 kinase inhibitors 2.48Å AUTH S.T.STABEN,J.A.FENG,K.LYLE,M.BELVIN,J.BOGGS,J.D.BURCH,AUTH 2 C.C.CHUA,H.CUI,A.G.DIPASQUALE,L.S.FRIEDMAN,C.HEISE,AUTH 3 H.KOEPPEN,A.KOTEY,R.MINTZER,A.OH,D.A.ROBERTS,L.ROUGE,AUTH 4 J.RUDOLPH,C.TAM,W.WANG,Y.XIAO,A.YOUNG,Y.ZHANG,K.P.HOEFLICHTITL BACK POCKET FLEXIBILITY PROVIDES GROUP II P21-ACTIVATEDTITL 2 KINASE (PAK) SELECTIVITY FOR TYPE I 1/2 KINASE INHIBITORS.REF J.MED.CHEM. V. 57 1033 2014REFN ISSN 0022-2623PMID 24432870DOI 10.1021/JM401768T Variant Set Distributions […]

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