4HWT.B | TARS

General Structure Information 4hwt TARS crystal structure of human threonyl-trna synthetase bound to a novel inhibitor 2.3Å AUTH M.TENG,M.T.HILGERS,M.L.CUNNINGHAM,A.BORCHARDT,J.B.LOCKE,AUTH 2 S.ABRAHAM,G.HALEY,B.P.KWAN,C.HALL,G.W.HOUGH,K.J.SHAW,J.FINNTITL IDENTIFICATION OF BACTERIA-SELECTIVE THREONYL-TRNATITL 2 SYNTHETASE SUBSTRATE INHIBITORS BY STRUCTURE-BASED DESIGN.REF J.MED.CHEM. V. 56 1748 2013REFN ISSN 0022-2623PMID 23362938DOI 10.1021/JM301756M Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Mapped Variants

See Details
3TDC.A | ACACB

General Structure Information 3tdc ACACB crystal structure of human acetyl-coa carboxylase 2 2.41Å AUTH T.YAMASHITA,M.KAMATA,S.ENDO,M.YAMAMOTO,K.KAKEGAWA,AUTH 2 H.WATANABE,K.MIWA,T.YAMANO,M.FUNATA,J.SAKAMOTO,A.TANI,AUTH 3 C.D.MOL,H.ZOU,D.R.DOUGAN,B.SANG,G.SNELL,K.FUKATSUTITL DESIGN, SYNTHESIS, AND STRUCTURE-ACTIVITY RELATIONSHIPS OFTITL 2 SPIROLACTONES BEARING 2-UREIDOBENZOTHIOPHENE AS ACETYL-COATITL 3 CARBOXYLASES INHIBITORS.REF BIOORG.MED.CHEM.LETT. V. 21 6314 2011REFN ISSN 0960-894XPMID 21944854DOI 10.1016/J.BMCL.2011.08.117 Variant Set Distributions Ripley’s K Analysis Plots Variant Set Comparisons Pathogenic Proximity […]

See Details